Invention Grant
- Patent Title: Monoamine reuptake inhibitors
- Patent Title (中): 单胺再摄取抑制剂
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Application No.: US13271419Application Date: 2011-10-12
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Publication No.: US09562001B2Publication Date: 2017-02-07
- Inventor: Frank Ivy Carroll , Bruce Edward Blough , Philip Abraham
- Applicant: Frank Ivy Carroll , Bruce Edward Blough , Philip Abraham
- Applicant Address: US NC Research Triangle Park
- Assignee: Research Triangle Institute
- Current Assignee: Research Triangle Institute
- Current Assignee Address: US NC Research Triangle Park
- Agency: Womble Carlyle Sandridge & Rice, LLP
- Main IPC: A61K31/137
- IPC: A61K31/137 ; C07C225/18 ; A61P25/24 ; A61P3/04 ; A61P25/34 ; A61P25/00 ; A61P3/00 ; A61P25/16 ; A61P25/22 ; A61P25/06 ; A61P25/36 ; A01N33/24 ; C07C225/16 ; C07C211/27 ; C07C211/29 ; C07C211/35

Abstract:
The invention provides bupropion analog compounds capable of inhibiting the reuptake of one or more monoamines. The compounds may selectively bind to one or more monoamine transporters, including those for dopamine, norepinephrine, and serotonin. Such compounds may be used to treat conditions that are responsive to inhibition of the reuptake of monoamines, including addiction, depression, and obesity.
Public/Granted literature
- US20120071560A1 MONOAMINE REUPTAKE INHIBITORS Public/Granted day:2012-03-22
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