Invention Grant
US09562009B2 Process to manufacture N-[(3S)-1-[4-[(3-fluorophenyl)methoxy]phenyl]-5-oxo-pyrrolidin-3-yl]acetamide
有权
制备N - [(3S)-1- [4 - [(3-氟苯基)甲氧基]苯基] -5-氧代 - 吡咯烷-3-基]乙酰胺
- Patent Title: Process to manufacture N-[(3S)-1-[4-[(3-fluorophenyl)methoxy]phenyl]-5-oxo-pyrrolidin-3-yl]acetamide
- Patent Title (中): 制备N - [(3S)-1- [4 - [(3-氟苯基)甲氧基]苯基] -5-氧代 - 吡咯烷-3-基]乙酰胺
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Application No.: US15139668Application Date: 2016-04-27
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Publication No.: US09562009B2Publication Date: 2017-02-07
- Inventor: Olaf Grassmann , Stefan Hildbrand , Roland Meier , Michelangelo Scalone , Urs Schwitter , Beat Wirz , Ulrich Zutter
- Applicant: Hoffmann-La Roche Inc.
- Applicant Address: US NJ Little Falls
- Assignee: Hoffmann-La Roche Inc.
- Current Assignee: Hoffmann-La Roche Inc.
- Current Assignee Address: US NJ Little Falls
- Priority: EP13190612 20131029
- Main IPC: C07D207/273
- IPC: C07D207/273 ; C07C237/22
![Process to manufacture N-[(3S)-1-[4-[(3-fluorophenyl)methoxy]phenyl]-5-oxo-pyrrolidin-3-yl]acetamide](/abs-image/US/2017/02/07/US09562009B2/abs.jpg.150x150.jpg)
Abstract:
The present invention provides processes to manufacture crystalline N-[(3S)-1-[4-[(3-fluorophenyl)methoxy]phenyl]-5-oxo-pyrrolidin-3-yl]acetamide. Also disclosed are compounds useful as intermediates in the methods of the invention.
Public/Granted literature
- US20160237032A1 PROCESS TO MANUFACTURE N-[(3S)-1-[4-[(3-FLUOROPHENYL)METHOXY]PHENYL]-5-OXO-PYRROLIDIN-3-YL]ACETAMIDE Public/Granted day:2016-08-18
Information query
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