Invention Grant
US09573943B2 Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use
有权
吡唑-4-基 - 杂环基甲酰胺化合物及其使用方法
- Patent Title: Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use
- Patent Title (中): 吡唑-4-基 - 杂环基甲酰胺化合物及其使用方法
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Application No.: US14153891Application Date: 2014-01-13
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Publication No.: US09573943B2Publication Date: 2017-02-21
- Inventor: Xiaojing Wang
- Applicant: Genentech, Inc.
- Applicant Address: US CA South San Francisco
- Assignee: Genentech, Inc.
- Current Assignee: Genentech, Inc.
- Current Assignee Address: US CA South San Francisco
- Agency: Alston & Bird LLP
- Main IPC: A61K31/4155
- IPC: A61K31/4155 ; C07D401/14 ; C07D403/14 ; C07D417/14 ; C07D401/12 ; C07D403/12 ; C07D417/12

Abstract:
Pyrazol-4-yl-heterocyclyl-carboxamide compounds of Formula I, including stereoisomers, geometric isomers, tautomers, and pharmaceutically acceptable salts thereof, wherein X is a thiazolyl, picolinyl, pyridinyl, or pyrimidinyl, are useful for inhibiting Pim kinase, and for treating disorders such as cancer mediated by Pim kinase. Methods of using compounds of Formula I for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions, are disclosed.
Public/Granted literature
- US20140128376A1 PYRAZOL-4-YL-HETEROCYCLYL-CARBOXAMIDE COMPOUNDS AND METHODS OF USE Public/Granted day:2014-05-08
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