Invention Grant
- Patent Title: Processes for preparing ASK1 inhibitors
- Patent Title (中): 制备ASK1抑制剂的方法
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Application No.: US14757663Application Date: 2015-12-22
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Publication No.: US09586933B2Publication Date: 2017-03-07
- Inventor: Gregory Notte
- Applicant: Gilead Sciences, Inc.
- Applicant Address: US CA Foster City
- Assignee: Gilead Sciences, Inc.
- Current Assignee: Gilead Sciences, Inc.
- Current Assignee Address: US CA Foster City
- Main IPC: C07D233/64
- IPC: C07D233/64 ; C07D401/14 ; C07D233/56

Abstract:
The present disclosure provides processes for the preparation of a compound of formula: which exhibits apoptosis signal-regulating kinase (“ASK1”) inhibitory activity and is thus useful in the treatment of diseases such as kidney disease, diabetic nephropathy and kidney fibrosis. The disclosure also provides compounds that are synthetic intermediates.
Public/Granted literature
- US20160244430A1 Processes for preparing ASK1 inhibitors Public/Granted day:2016-08-25
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