Invention Grant
- Patent Title: Imidazoline derivatives, preparation methods thereof, and their applications in medicine
- Patent Title (中): 咪唑啉衍生物及其制备方法及其在药物中的应用
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Application No.: US14425207Application Date: 2013-08-26
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Publication No.: US09586947B2Publication Date: 2017-03-07
- Inventor: Hejun Lu , Piaoyang Sun , Hongbo Fei , Hongjian Jiang , Haowei Wang , Qing Dong
- Applicant: Shanghai Hengrui Pharmaceutical Co., Ltd. , Jiangsu Hengrui Medicine Co., Ltd.
- Applicant Address: CN Shanghai CN Lianyungang, Jiangsu
- Assignee: Shanghai Hengrui Pharmaceutical Co., Ltd.,Jiangsu Hengrui Medicine Co., Ltd.
- Current Assignee: Shanghai Hengrui Pharmaceutical Co., Ltd.,Jiangsu Hengrui Medicine Co., Ltd.
- Current Assignee Address: CN Shanghai CN Lianyungang, Jiangsu
- Agency: Panitch Schwarze Belisario & Nadel LLP
- Priority: CN201210323870 20120904
- International Application: PCT/CN2013/082273 WO 20130826
- International Announcement: WO2014/036897 WO 20140313
- Main IPC: C07D233/86
- IPC: C07D233/86 ; C07D409/12 ; C07D403/12 ; C07D405/14 ; C07D405/12 ; C07D401/04 ; C07D401/12

Abstract:
New imidazoline derivatives represented by formula (I): preparation methods thereof, pharmaceutical compositions comprising such derivatives, and applications of such derivatives in preparing androgen receptor antagonists and medicaments for treating diseases such as prostate cancer are described.
Public/Granted literature
- US20150225381A1 IMIDAZOLINE DERIVATIVES, PREPARATION METHODS THEREOF, AND THEIR APPLICATIONS IN MEDICINE Public/Granted day:2015-08-13
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