Invention Grant
- Patent Title: Structural variants of mycolactones for use in modulating inflammation, immunity and pain
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Application No.: US14358501Application Date: 2012-11-16
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Publication No.: US09598393B2Publication Date: 2017-03-21
- Inventor: Caroline Demangel , Nicolas Blanchard , Georges Bismuth , Jacques Eustache , Virginie Casarotto , Anne-Caroline Chany , Laure Guenin-Mace
- Applicant: INSTITUT PASTEUR
- Applicant Address: FR Paris
- Assignee: Institut Pasteur
- Current Assignee: Institut Pasteur
- Current Assignee Address: FR Paris
- Agency: Foley & Lardner LLP
- Priority: EP11306521 20111118
- International Application: PCT/IB2012/056506 WO 20121116
- International Announcement: WO2013/072896 WO 20130523
- Main IPC: C07D313/00
- IPC: C07D313/00 ; A61K31/335 ; C07C69/76 ; C07D521/00 ; C07C69/732 ; C07C43/15 ; C07C59/135 ; C07F5/02

Abstract:
The present invention is related to variants of mycolactones of formula (I), processes for the preparation thereof, pharmaceutical compositions thereof and their use in modulating inflammation, immunity and pain. Y—O—W (I), wherein Y and W are as defined in claim 1.
Public/Granted literature
- US20140329771A1 STRUCTURAL VARIANTS OF MYCOLACTONES FOR USE IN MODULATING INFLAMMATION, IMMUNITY AND PAIN Public/Granted day:2014-11-06
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