Invention Grant
- Patent Title: Process for manufacturing 5-(2,6-di-4-morpholinyl-4-pyrimidinyl)-4-trifluoromethylpyridin-2-amine
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Application No.: US14437177Application Date: 2013-10-21
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Publication No.: US09637468B2Publication Date: 2017-05-02
- Inventor: Dietmar Flubacher , Nicole Bieri , Murat Acemoglu , Pascal Michel , Rasmus Mose , Hans Stettler , Maria Caterina Testa , Joerg Brozio , Frank Schaefer
- Applicant: Dietmar Flubacher , Nicole Bieri , Murat Acemoglu , Pascal Michel , Rasmus Mose , Hans Stettler , Maria Caterina Testa , Joerg Brozio , Frank Schaefer
- Applicant Address: CH Basel
- Assignee: Novartis AG
- Current Assignee: Novartis AG
- Current Assignee Address: CH Basel
- Agent Sandra Rueck
- International Application: PCT/EP2013/071996 WO 20131021
- International Announcement: WO2014/064058 WO 20140501
- Main IPC: C07D401/04
- IPC: C07D401/04 ; C07D213/75 ; C07F5/02 ; C07D413/14 ; A61K31/5377 ; A61K31/506 ; A61K31/4433 ; A61K31/444 ; C07D401/14 ; C07D239/28 ; C07D239/42

Abstract:
The invention discloses improved processes for manufacturing a compound, 5-(2,6-Di-4-morpholinyl-4-pyrimidinyl)-4-trifluoromethylpyridin-2-amine, its monohydrochloride salt and intermediates thereof.
Public/Granted literature
- US20150246897A1 Process for Manufacturing 5-(2,6-Di-4-morpholinyl-4-pyrimidinyl)-4-trifluoromethylpyridin-2-amine Public/Granted day:2015-09-03
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