Invention Grant
- Patent Title: Process for the regioselective synthesis of pyrazoles
-
Application No.: US15104094Application Date: 2014-12-23
-
Publication No.: US09676726B2Publication Date: 2017-06-13
- Inventor: Giovanni Meazza , Laura Sillani , Pierangelo Mereghetti , Daniele Forgia
- Applicant: ISAGRO S.P.A.
- Applicant Address: IT Milan
- Assignee: ISAGRO S.P.A.
- Current Assignee: ISAGRO S.P.A.
- Current Assignee Address: IT Milan
- Agency: Florek & Endres PLLC
- Priority: ITMI2013A2201 20131223
- International Application: PCT/IB2014/067258 WO 20141223
- International Announcement: WO2015/097658 WO 20150702
- Main IPC: C07D231/14
- IPC: C07D231/14 ; C07C243/28

Abstract:
A process is described for the synthesis of pyrazoles having general formula (I) which comprises the steps of mixing a compound having general formula (II) and a 1,2-disubstituted hydrazine having general formula (III) to form a reaction intermediate having general formula (IV) and the reaction mixture obtained in step i), in an acid environment, cyclizes to form a pyrazole having general formula (I), according to reaction scheme 1
Public/Granted literature
- US20160318874A1 PROCESS FOR THE REGIOSELECTIVE SYNTHESIS OF PYRAZOLES Public/Granted day:2016-11-03
Information query