Invention Grant
- Patent Title: Azaindole derivative
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Application No.: US15112070Application Date: 2015-02-04
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Publication No.: US09676773B2Publication Date: 2017-06-13
- Inventor: Masayuki Nakamura , Hiroyoshi Yamanaka , Kazuaki Shibata , Morihiro Mitsuya , Takafumi Harada
- Applicant: TAIHO PHARMACEUTICAL CO., LTD.
- Applicant Address: JP Chiyoda-ku
- Assignee: TAIHO PHARMACEUTICAL CO., LTD.
- Current Assignee: TAIHO PHARMACEUTICAL CO., LTD.
- Current Assignee Address: JP Chiyoda-ku
- Agency: Oblon, McClelland, Maier & Neustadt, L.L.P.
- Priority: JP2014-019584 20140204
- International Application: PCT/JP2015/053031 WO 20150204
- International Announcement: WO2015/119126 WO 20150813
- Main IPC: C07D401/14
- IPC: C07D401/14 ; A61K31/437 ; C07D471/04

Abstract:
Provided is a novel compound having a selective JAK3-inhibitory effect and also having excellent oral absorbability. Also provided is a pharmaceutical agent, which is based on a JAK3-inhibitory effect and is useful for preventing and/or treating a disease involving the JAK3, and in particular, rheumatoid arthritis or multiple sclerosis.An azaindole derivative having a cycloalkenyl group, which is represented by the following formula (I), or a salt thereof, and a pharmaceutical composition containing the same: where R1 to R4, m and n have the same meanings as those defined in the description.
Public/Granted literature
- US20160340353A1 AZAINDOLE DERIVATIVE Public/Granted day:2016-11-24
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