Invention Grant
- Patent Title: 1,3-Disubstituted cyclopentane derivatives
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Application No.: US14908217Application Date: 2014-07-11
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Publication No.: US09718785B2Publication Date: 2017-08-01
- Inventor: Christos Tsaklakidis , Wolfgang Staehle , Birgitta Leuthner , Thomas Fuchss
- Applicant: MERCK PATENT GMBH
- Applicant Address: DE Darmstadt
- Assignee: MERCK PATENT GMBH
- Current Assignee: MERCK PATENT GMBH
- Current Assignee Address: DE Darmstadt
- Agency: Millen White Zelano and Branigan, PC
- Agent John Sopp; Anthony Zelano
- Priority: EP13003769 20130729
- International Application: PCT/EP2014/001912 WO 20140711
- International Announcement: WO2015/014446 WO 20150205
- Main IPC: C07D231/12
- IPC: C07D231/12 ; C07D231/54 ; C07D233/60 ; C07D233/61 ; C07D233/64 ; C07D233/66 ; C07D249/06 ; C07D249/08 ; C07D401/14 ; C07D403/10 ; C07D413/10 ; C07D413/14 ; C07D417/10 ; C07D471/04 ; A61K31/4164 ; A61K31/4178 ; A61K31/4192 ; A61K31/4196 ; A61K31/423 ; A61K31/428 ; A61K31/437

Abstract:
Compounds of the formula I in which R, Y, R1, X1, X2, X3 and q have the meanings indicated in claim 1, are inhibitors of fatty acid synthase, and can be employed, inter alia, for the treatment of diseases such as cancer, cardiovascular diseases, central nervous system injury and different forms of inflammation.
Public/Granted literature
- US20160176824A1 1,3-DISUBSTITUTED CYCLOPENTANE DERIVATIVES Public/Granted day:2016-06-23
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