Invention Grant
- Patent Title: Pyrazole derivative
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Application No.: US15234730Application Date: 2016-08-11
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Publication No.: US09777000B2Publication Date: 2017-10-03
- Inventor: Akihiro Okano , Kouki Ogawa
- Applicant: MOCHIDA PHARMACEUTICAL CO., LTD.
- Applicant Address: JP Tokyo
- Assignee: MOCHIDA PHARMACEUTICAL CO., LTD.
- Current Assignee: MOCHIDA PHARMACEUTICAL CO., LTD.
- Current Assignee Address: JP Tokyo
- Agency: Birch, Stewart, Kolasch & Birch, LLP
- Priority: JP2013-038030 20130227
- Main IPC: C07D471/04
- IPC: C07D471/04 ; C07D401/04 ; C07D417/04 ; A61K31/437 ; A61K31/444 ; A61K31/497 ; A61K31/501 ; A61K31/506 ; A61K31/5377 ; A61K45/06 ; C07D403/04

Abstract:
It has been desired to develop a pharmaceutical composition, which is used in agents for preventing and/or treating various diseases related to PDE10 (e.g. mental disorder and neurodegenerative disorder). The present invention provides: compounds having PDE10 inhibitory effect, in particular, compounds having a 4-heteroarylpyrazole-5-carboxylic acid amide structure represented by the following formula (I), or their pharmaceutically acceptable salts, or their solvates; pharmaceutical compositions comprising, as active ingredients, the compounds, or their pharmaceutically acceptable salts, or their solvates; and medical use of the compounds, or their pharmaceutically acceptable salts, or their solvates.
Public/Granted literature
- US20160347751A1 NOVEL PYRAZOLE DERIVATIVE Public/Granted day:2016-12-01
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