Invention Grant
- Patent Title: Crystalline forms and processes for the preparation of phenyl-pyrazoles useful as modulators of the 5-HT2A serotonin receptor
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Application No.: US14921651Application Date: 2015-10-23
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Publication No.: US09783502B2Publication Date: 2017-10-10
- Inventor: Tawfik Gharbaoui , Dipanjan Sengupta , Ashwin Krishnan , Nainesh Shah , Ryan M. Hart , Mark Macias , Edward A. Lally
- Applicant: Arena Pharmaceuticals, Inc.
- Applicant Address: US CA San Diego
- Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee Address: US CA San Diego
- Agency: Fish & Richardson P.C.
- Agent Lyle W. Spruce
- Main IPC: C07D231/12
- IPC: C07D231/12

Abstract:
The present invention relates to processes for preparing phenyl-pyrazoles of Formula (I) and salts and pharmaceutical compositions thereof, useful as modulators of 5-HT2A serotonin receptor activity. The present invention also relates to intermediates used in the processes, and their preparation. The present invention also relates to crystalline forms of 5-HT2A serotonin receptor modulators, compositions thereof and methods of using the same.
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