Invention Grant
- Patent Title: Process for the preparation of Paliperidone palmitate
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Application No.: US15543987Application Date: 2016-01-13
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Publication No.: US09963449B2Publication Date: 2018-05-08
- Inventor: Sandeep Jain , Srikanth Sindhanur , Anil Kumar Jain , Sivakumaran Meenakshisunderam
- Applicant: AUROBINDO PHARMA LIMITED
- Applicant Address: IN Hyderabad
- Assignee: Aurobindo Pharma Ltd
- Current Assignee: Aurobindo Pharma Ltd
- Current Assignee Address: IN Hyderabad
- Agent Jay R. Akhave
- Priority: IN269/CHE/2015 20150119
- International Application: PCT/IB2016/050136 WO 20160113
- International Announcement: WO2016/116831 WO 20160728
- Main IPC: A01N43/90
- IPC: A01N43/90 ; A61K31/519 ; C07D471/04

Abstract:
The present invention relates to a process for the preparation of pure Paliperidone Palmitate, which comprises: (a) providing a solution of Paliperidone Palmitate in an alcoholic solvent; (b) adding the alcoholic solution of Paliperidone palmitate to water or vice versa; and (c) isolating the product to obtain pure Paliperidone Palmitate.
Public/Granted literature
- US20180009802A1 PROCESS FOR THE PREPARATION OF PALIPERIDONE PALMITATE Public/Granted day:2018-01-11
Information query
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