Invention Grant
- Patent Title: Method of forming methyl penam derivatives
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Application No.: US15311146Application Date: 2015-05-14
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Publication No.: US09963465B2Publication Date: 2018-05-08
- Inventor: Andrea Faini , Marco Forzatti , Giovanni Fogliato , Stefano Biondi
- Applicant: Allecra Therapeutics SAS
- Applicant Address: FR Saint Louis
- Assignee: Allecra Therapeutics SAS
- Current Assignee: Allecra Therapeutics SAS
- Current Assignee Address: FR Saint Louis
- Agency: Marshall, Gerstein & Borun LLP
- Priority: GB1408649.0 20140515
- International Application: PCT/EP2015/060733 WO 20150514
- International Announcement: WO2015/173378 WO 20151119
- Main IPC: C07D499/87
- IPC: C07D499/87

Abstract:
A method of forming a compound of formula (IIIa): wherein: R1 in each occurrence is independently selected from H, halogen, amino, C1-5 alkyl, C1-5 alkenyl and C1-5 alkynyl; R2 in each occurrence is independently selected from H, halogen, amino, C1-5 alkyl, C1-5 alkenyl and C1-5 alkynyl; R4 is C1-5 alkyl; and R6 is a C1-5 fluoroalkyl; and PG is a protecting group, the method comprising the step of reacting a compound of formula (IIa) with a compound of formula (VIII):
Public/Granted literature
- US20170101421A1 METHOD Public/Granted day:2017-04-13
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