AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES
    3.
    发明申请
    AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES 审中-公开
    氨基取代的苯并(杂环)环状衍生物

    公开(公告)号:WO2004080170A3

    公开(公告)日:2004-11-04

    申请号:PCT/EP2004001677

    申请日:2004-02-20

    CPC classification number: A01N43/72 A01N43/60

    Abstract: Use of compounds Formula (I), A = a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R = OH, SH, NH2, CN, NO2, halogen, C1-C6-alkyl, C1-C6-haloalkyl; C1-C6- alkoxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C2-C6-alkenyl, C2-C6-alkenyloxy, C2-C6-alkenylthio, C2-C6-alkynyl, C2-C6­alkynyloxy, C2-C6-alkynylthio, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C2-C6-alkenylsulfonyl, C2-C6-alkynylsulfoxyl, C1-C6-alkylcarbonyl, C1-C6- alkoxycarbonyl, C1-C6-alkylcarbonyloxy; R = C1-C6-alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C1-C6-alkylene or C1-C6-alkyleneoxy linkage to A or fused to A and which may be substituted; R , R = H, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylamino, C1-C6-alkoxy, C3-C6 cycloalkyl, or R and R together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system con-taining 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitro-gen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R and R together form the chains -(CH2)2N (O-)(CH2)2- or -(CH2)3N (O )(CH2)2 ; m = 0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.

    Abstract translation: 式(I)化合物的用途,A =可含有1-3个杂原子且可以是饱和或部分或完全不饱和的5至7元环; R 1 = OH,SH,NH 2,CN,NO 2,卤素,C 1 -C 6烷基,C 1 -C 6卤代烷基; C 1 -C 6烷氧基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基,C 1 -C 6卤代烷硫基,C 2 -C 6烯基,C 2 -C 6烯氧基,C 2 -C 6烯硫基, C 1 -C 6烷基磺酰基,C 1 -C 6烷基亚磺酰基,C 2 -C 6烯基磺酰基,C 2 -C 6炔基亚磺酰基,C 1 -C 6烷基羰基,C 1 -C 6烷氧基羰基, R 2 = C 1 -C 6烷基或可含有1至4个杂原子并且直接键合或通过O,S,C 1 -C 6亚烷基键合的单环或双环5至10元芳环体系或 与A相连的C1-C6-亚烷氧基键或者与A相连并可以被取代的; R 3,R 4 = H,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6烷基氨基,C 1 -C 6烷氧基,C 3 -C 6环烷基或R 3和 R 4与它们所连接的氮原子一起形成饱和或部分饱和的含有1至3个杂原子的5至10元环系统或含有1至4个硝基的5元杂芳基 其中环系统中的碳和/或氮原子可以被取代或者可以被取代的苯基或苄基; 或者R 3和R 4一起形成链 - (CH 2)2 N +(O-)(CH 2)2 - 或 - (CH 2)3 N +(O-)(CH 2)2 < - >; m = 0至4; n是0至4; 以及用于防治昆虫,蛛形纲动物或线虫的对映异构体,非对映异构体,顺式/反式异构体或其盐,控制这些害虫的方法以及通过施用农药有效量的式(I)化合物来保护生长中的植物对这些害虫的侵袭或侵染 (I),制备它们的方法以及包含它们的组合物。

    2-ARYLOXY-6-PYRAZOLYL-PYRIDINES
    4.
    发明申请
    2-ARYLOXY-6-PYRAZOLYL-PYRIDINES 审中-公开
    2-芳氧基-6-吡唑基 - 吡啶

    公开(公告)号:WO03029243A3

    公开(公告)日:2003-09-12

    申请号:PCT/EP0210322

    申请日:2002-09-14

    CPC classification number: C07D401/04 A01N43/56

    Abstract: The invention relates to 2-aryloxy-6-pyrazolyl-pyridines of formula (I), in which the variables are defined as follows: A represents phenyl, which is optionally substituted, an optionally substituted 5 or 6-membered heteroaryl comprising between one and four N, O and/or S atoms, or 2,2-difluorobenzo[1.3]dioxol-4-yl or 2,2-difluorobenzo[1.3]dioxol-5-yl; X represents O, S, CH2-0 or CH2-S; R represents hydrogen, halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy; R represents hydrogen, halogen, cyano, cycloalkyl, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkoxyalkyl, alkylamino, dialkylamino, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl or COR ; R represents halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy; R represents hydrogen, halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl or alkoxyalkyl; R represents hydrogen, halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl or haloalkylsulfonyl; R represents hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl or cycloalkyl; R represents hydrogen, hydroxy, alkyl, alkoxy, amino, alkylamino or dialkylamino. The invention also relates to the agriculturally useful salts of said pyridines, to a method and intermediate products for their production and to the use of said compounds or agents containing said compounds for combating undesirable plants.

    Abstract translation: 本发明涉及式(I):其中各变量具有以下含义的2-芳氧基-6-吡唑基 - 吡啶:A是苯基,其任选被取代; 5-或6-元含一个杂至四个N,O和/或S原子,其任选被取代; 2,2-二氟 - 苯并[1.3]二氧杂环戊烯-4-基或2,2-二氟 - 苯并[1.3]二氧杂环戊烯-5-基; X是O,S,或CH 2 -CH 2 -O S; [R 是氢,卤素,氰基,硝基,烷基,卤代烷基,烷氧基或卤代烷 - [R <2>是氢,卤素,氰基,环烷基,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代炔基,烷氧基,链烯氧基,炔氧基,卤代烷氧基 ,烷氧基烷基,烷基氨基,二烷基氨基,烷硫基,卤代烷硫基,烷基亚磺酰基,卤代烷,烷基磺酰基,卤代烷基磺酰基或COR <7>; [R <3>为卤素,氰基,硝基,烷基,卤代烷基,烷氧基或卤代烷氧基; [R <4>是氢,卤素,氰基,硝基,烷基,烯基,炔基,卤代烷基或烷氧基烷基; [R <5>是氢,卤素,氰基,硝基,烷基,烯基,炔基,卤代烷基,烷氧基,烷氧基烷基,卤代烷氧基,烷硫基,卤代烷硫基,烷基亚磺酰基,卤代烷基亚磺酰,烷基磺酰基或卤代烷基磺酰基; [R <6>是氢,氰基,烷基,烯基,炔基,卤代烷基或环烷基; [R <7>是氢,羟基,烷基,烷氧基,氨基,烷基氨基或二烷基氨基; 及其可农用盐,过程和它们的制备中间体; 和使用这些化合物或包含用于控制不希望的Pflangen手段这些化合物。

    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS
    5.
    发明申请
    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-(1,2-二苯基乙基)-3-(2-羟基乙基) - 硫脲化合物,用于组合动物饲料

    公开(公告)号:WO2006125745A3

    公开(公告)日:2007-05-10

    申请号:PCT/EP2006062413

    申请日:2006-05-18

    CPC classification number: C07C335/12 A01N47/28

    Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal at- tack or infestation, with a pesticidally effective amount of at least one 1-(1 ,2-diphenyl- ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R 3 and R 4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R 7 , R 8 , R 9 and R 10 are H or optionally substituted C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 - alkylamino, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, phenyl or benzyl and the variables R 1 , R 2 , R 5 and R 6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

    Abstract translation: 本发明涉及一种防治动物害虫的方法,包括使动物害虫,其习惯,繁殖地,食物供应,植物,种子,土壤,区域,动物害虫生长或可能生长的物质或环境接触;或 防止动物死亡或侵染的材料,植物,种子,土壤,表面或空间,具有杀虫有效量的至少一种1-(1,2-二苯基 - 乙基)-3-(2-羟乙基 ) - 硫脲化合物I或其农业上可接受的盐,其中m为0至5,n为0至5,R 3和R 4为H或任选取代的烷基 ,卤代烷基,环烷基,苯基或苄基,R 7,R 8,R 9和R 10是H 或任选取代的C 1 -C 6 - 烷基,C 1 -C 6 - 卤代烷基,C 1,R 2,R 5和R 6如权利要求中所定义。 本发明还涉及一种保护作物免受动物害虫侵袭或侵袭的方法,一种保护非生物材料免受动物害虫侵袭或侵染的方法,新的1-(1,2-二苯基 - 乙基)-3-( 2-羟乙基) - 硫脲化合物I及其农业上可接受的盐,以及包含1-(1,2-二苯基 - 乙基)-3-(2-羟乙基) - 硫脲化合物I或其盐的农业组合物。

    RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES
    8.
    发明申请
    RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
    RESORCINE衍生物及其作为杀虫剂的用途

    公开(公告)号:WO2007054558A2

    公开(公告)日:2007-05-18

    申请号:PCT/EP2006068329

    申请日:2006-11-10

    CPC classification number: C07D213/64 C07D277/34 C07D307/80

    Abstract: This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)Ra, -C(=G)ORa, -C(=G)NRa2, -C(=G)[N=SRa2], -C(=NORa)Ra, -C(=NORa)NRa2, -C(=NNRa2)Ra , -OC(=G)-OC(=G)ORa, N=SRa2, -NRaC(=G)Ra, -N[C(=G)Ra]2, - NRaC(=G)ORa, -C(=G)NRa-NRa2, -C(=G)NRa-NRa [C(=G)Ra], -NRa-C(=G)NRa2, -NRa-NRaC(=G)Ra, -NRa-N[C(=G)Ra]2, -N[(C=G)Ra]-NRa2, -NRa-NRa[(C=G)GRa], -NRa[(C=G)NRa2, -NRa[C=NRa]Ra, -NRa(C=NRa)NRa2, -O-NRa2, -O-NRa(C=G)Ra, - SO2NRa2, -NRaSO2Ra, -S(=O)Ra, -S(=O)2Ra, -SO2ORa, or -OSO2Ra, wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

    Abstract translation: 本发明涉及其中R 1为苯基或可含有1-3个选自氧,氮和硫的杂原子的5至6元杂芳环的式(I)的间苯二酚衍生物,其中苯基 或杂芳环可以与选自苯基和5-至6-元饱和,部分不饱和或芳族杂环的环稠合,所述杂环可以含有1-3个选自氧,氮和硫的杂原子,其中苯基或5- 至6元杂芳环或相应的稠环体系可以是未取代的或被1至6个任选取代的基团R 3 3的任何组合取代,其中R 3是卤素, 氰基,硝基,羟基,巯基,氨基,烷基,烯基,炔基,环烷基,环烯基,卤代烷基,卤代烯基,卤代炔基,卤代环烷基,卤代环烯基,烷氧基,烯氧基,炔氧基,卤代烷氧基,卤代烯氧基,卤代炔氧基,烷硫基,烯硫基,炔硫基,卤代烷硫基, H 烯基氨基,炔基氨基,二烷基氨基,二链烷基氨基,二炔基氨基,烷基 - 链烯基氨基,烷基 - 炔基氨基,烯基 - 炔基氨基,三烷基甲硅烷基或苯基或5至7元饱和或部分不饱和的杂环, 至3个选自氧,硫和氮的杂原子或5至6元杂芳环体系,其可以含有1至4个选自氧,氮和硫的杂原子,该苯基和杂芳环可以通过氧或 硫原子或-C(= G)R a,-C(= G)OR a,-C(= G)NR a 2,-C(= G)[N = SR a 2] (= NORa)NRa2,-C(= NNRa2)Ra,-OC(= G)-OC(= G)ORa,N = SRa2,-NRaC(= G)Ra,-N [C(= G)Ra] 2,-NR a C(= G)OR a,-C(= G)NR a -NR a 2,-C(= G)NR a -NR a [C(= G)R a] -NRaC(= G)Ra,-NRa-N [C(= G)Ra] 2,-N [(C = G)Ra] -NRa2,-NRa-NRa [(C = G) [(C = G)NRa2,-NRa [C = NRa] Ra,-NRa(C = NRa)NRa2,-O-NRa2,-O-NRa(C = G)Ra,-SO2NRa2,-NRaSO2Ra,-S (= O)R a,-S(= O)2 R a,-SO 2 OR a或-O SO 2 R a,其中G是氧或硫,Ra如说明书中所定义,R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基,烷氧基或卤代烷氧基, x是2,3,4,5,6或7,或其非对映异构体,对映异构体,盐或N-氧化物,条件是R 1不是5-氯-2,2 ,当R 2是氢并且x是3或4时,制备化合物I的方法和中间体,使用化合物I,其中R 1,R 2,R 3, 用于防治昆虫,螨虫或线虫,以及用化合物I治疗,控制,预防或保护动物免受寄生虫侵袭或感染的方法。

    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS
    9.
    发明申请
    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    新型2-氰基-3-(卤代)烷氧基苯磺酰胺化合物用于防治动物病虫害

    公开(公告)号:WO2006056433A2

    公开(公告)日:2006-06-01

    申请号:PCT/EP2005012561

    申请日:2005-11-24

    CPC classification number: C07C319/20 A01N41/06 C07C311/29 C07C323/62

    Abstract: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds (I), where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to: the use of compounds (I) and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula (I) and/or at least one agriculturally useful salt of (I) and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula (I) and/or at least one agriculturally acceptable salt thereof; a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula (I).

    Abstract translation: 本发明涉及2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物(I),其中变量Alk和R1-R5如权利要求1中所定义,和/或其可农用盐。 此外,本发明涉及:化合物(I)和/或其盐用于对抗动物害虫的用途; 包含这种量的至少一种通式(I)的化合物和/或至少一种(I)的农业上有用的盐和至少一种惰性液体和/或固体农艺上可接受的载体的农业组合物,其具有杀虫作用 和如果需要的话,至少一种表面活性剂; 以及防治动物害虫的方法,其包括使动物害虫,其习性,繁殖场,食物供应,植物,种子,土壤,面积,动物害虫正在生长或可能生长的材料或环境,或材料,植物 (I)的至少一种2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物和/或至少一种农业上受到保护的种子,土壤,表面或空间免于动物攻击或侵染 其可接受的盐; 一种用于保护种子免受土壤昆虫以及所得植物的根和茎由土壤和叶面昆虫引起的方法,包括在播种之前和/或在萌芽后使种子与2-氰基-3-(卤代)烷氧基 - 苯磺酰胺 通式(I)的化合物。

    1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thioureacompounds for combating animal pests.

    公开(公告)号:EG25049A

    公开(公告)日:2011-07-19

    申请号:EGNA2007001264

    申请日:2007-11-20

    Applicant: BASF AG

    Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation, with a pesticidally effective amount of at least one 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R 3 and R 4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R 7 , R 8 , R 9 and R 10 are H or optionally substituted C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylamino, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, phenyl or benzyl and the variables R 1 , R 2 , R 5 and R 6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

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