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1.METHODS AND COMPOUNDS PRODUCING DIPEPTIDYL PEPTIDASE IV INHIBITORS AND INTERMEDIATES THEREOF 审中-公开
Title translation: 制备DIPEPTIDYL PEPTIDASE IV抑制剂的方法和化合物及其中间体公开(公告)号:WO2004052850A3
公开(公告)日:2006-03-02
申请号:PCT/US0338558
申请日:2003-12-04
Applicant: SQUIBB BRISTOL MYERS CO , VU TRUC CHI , BRZOZOWSKI DAVID B , FOX RITA , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , KOLOTUCHIN SERGEI V , MAZZULLO JOHN A JR , PATEL RAMESH N , WANG JIANJI , WONG KWOK , YU JURONG , ZHU JASON , MAGNIN DAVID R , AUGERI DAVID J , HAMANN LAWRENCE G
Inventor: VU TRUC CHI , BRZOZOWSKI DAVID B , FOX RITA , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , KOLOTUCHIN SERGEI V , MAZZULLO JOHN A JR , PATEL RAMESH N , WANG JIANJI , WONG KWOK , YU JURONG , ZHU JASON , MAGNIN DAVID R , AUGERI DAVID J , HAMANN LAWRENCE G
IPC: A61K31/403 , A61K31/435 , C07C62/06 , C07C69/00 , C07C69/716 , C07C229/28 , C07C271/22 , C07D20060101 , C07D201/00 , C07D207/22 , C07D207/277 , C07D209/02 , C07D209/52 , C07D221/02
CPC classification number: C07C69/757 , C07C62/06 , C07C69/635 , C07C69/675 , C07C229/28 , C07C271/22 , C07C2603/74 , C07D207/22 , C07D209/52
Abstract: Methods and compounds for production of cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV are provided.
Abstract translation: 提供了用于制备二肽基肽酶IV的环丙基稠合吡咯烷基抑制剂的方法和化合物。
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2.METHODS AND COMPOUNDS PRODUCING DIPEPTIDYL PEPTIDASE IV INHIBITORS AND INTERMEDIATES THEREOF 有权
Title translation: 生产二肽的方法和化合物肽基肽酶IV抑制剂及其中间体公开(公告)号:EP1581487A4
公开(公告)日:2007-08-08
申请号:EP03812799
申请日:2003-12-04
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: VU TRUC CHI , BRZOZOWSKI DAVID B , FOX RITA , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , KOLOTUCHIN SERGEI V , MAZZULLO JOHN A JR , PATEL RAMESH N , WANG JIANJI , WONG KWOK , YU JURONG , ZHU JASON , MAGNIN DAVID R , AUGERI DAVID J , HAMANN LAWRENCE G
IPC: A61K31/403 , A61K31/435 , C07C62/06 , C07C69/00 , C07C69/716 , C07C229/28 , C07C271/22 , C07D20060101 , C07D201/00 , C07D207/22 , C07D207/277 , C07D209/02 , C07D209/52 , C07D221/02
CPC classification number: C07C69/757 , C07C62/06 , C07C69/635 , C07C69/675 , C07C229/28 , C07C271/22 , C07C2603/74 , C07D207/22 , C07D209/52
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3.
公开(公告)号:AU2003297647A1
公开(公告)日:2004-06-30
申请号:AU2003297647
申请日:2003-12-04
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: VU TRUC CHI , BRZOZOWSKI DAVID B , FOX RITA , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , KOLOTUCHIN SERGEI V , MAZZULLO JOHN A JR , PATEL RAMESH N , WANG JIANJI , WONG KWOK , YU JURONG , ZHU JASON , MAGNIN DAVID R , AUGERI DAVID J , HAMANN LAWRENCE G
IPC: A61K31/403 , A61K31/435 , C07C62/06 , C07C69/00 , C07C69/716 , C07C229/28 , C07C271/22 , C07D20060101 , C07D201/00 , C07D207/22 , C07D207/277 , C07D209/02 , C07D209/52 , C07D221/02
Abstract: Methods and compounds for production of cycloproyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV are provided.
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公开(公告)号:BR0317139A
公开(公告)日:2005-11-29
申请号:BR0317139
申请日:2003-12-04
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: VU TRUC CHI , BRZOZOWSKI DAVID B , FOX RITA , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , KOLOTUCHIN SERGEI V , MAZULLO JOHN A JR , PATEL RAMESH N , WANG JIANJI , WONG KWOK , YU JURONG , ZHU JASON , MAGNIN DAVID R , AUGERI DAVID J , HAMANN LAWRENCE G
IPC: A61K31/403 , A61K31/435 , C07C62/06 , C07C69/00 , C07C69/716 , C07C229/28 , C07C271/22 , C07D20060101 , C07D201/00 , C07D207/22 , C07D207/277 , C07D209/02 , C07D209/52 , C07D221/02
Abstract: Methods and compounds for production of cycloproyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV are provided.
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5.
公开(公告)号:CA2508619A1
公开(公告)日:2004-06-24
申请号:CA2508619
申请日:2003-12-04
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: MAGNIN DAVID R , GODFREY JOLLIE DUAINE JR , HANSON RONALD L , MAZZULLO JOHN A JR , HAMANN LAWRENCE G , AUGERI DAVID J , KOLOTUCHIN SERGEI V , VU TRUC CHI , ZHU JASON , YU JURONG , BRZOZOWSKI DAVID B , PATEL RAMESH N , WANG JIANJI , WONG KWOK , FOX RITA
IPC: A61K31/403 , A61K31/435 , C07C62/06 , C07C69/00 , C07C69/716 , C07C229/28 , C07C271/22 , C07D20060101 , C07D201/00 , C07D207/22 , C07D207/277 , C07D209/02 , C07D209/52 , C07D221/02
Abstract: Methods and compounds for production of cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV are provided.
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