IMINO OXYPHENYL ACETIC ACID DERIVATIVES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND USE THEREOF
    96.
    发明申请
    IMINO OXYPHENYL ACETIC ACID DERIVATIVES, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AND USE THEREOF 审中-公开
    IMINOOXYPHENYLESSIGSÄUREDERIVATE,工艺和中间产品和使用

    公开(公告)号:WO1997024317A1

    公开(公告)日:1997-07-10

    申请号:PCT/EP1996005642

    申请日:1996-12-16

    CPC classification number: C07C251/60 C07C2601/10 C07C2601/14

    Abstract: The invention relates to 2-imino oxyphenyl acetic acid derivatives of formula (I) in which the substituents and the index have the following meanings: R is C(CO2CH3)=NOCH3 (Ia), C(CONHCH3)=NOCH3 (Ib), C(CONH2)=NOCH3 (Ic), C(CO2CH3)=CHOCH3 (Id), or C(CO2CH3)=CHCH3 (Ie); R is cyano, nitro, halogen, alkyl, alkyl halide or alkoxy; m is 0,1 or 2; R is hydrogen, cyano, hydroxy, halogen, alkyl, alkyl halide, alkoxy alkyl, alkoxy, alkoxy halide, alkylthio, cyclopropyl, alkenyl, optionally substituted aryloxy alkyl, benzyl or benzyloxy; R is hydrogen, cyano, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, heterocyclyl, aryl and hetaryl, optionally substituted alkoxy, alkenyloxy, alkinyloxy, cycloalkoxy, heterocyclyloxy, aryloxy and hetaryloxy, optionally substituted arylthio and hetarylthio; -Q-C(R )=N-Y -R or -Q-O-N=CR R ; R and R together with the carbon atom to which they are bound, are an optionally substituted four to eight-membered ring which can contain in addition to carbon atoms one or two oxygen atoms and/or sulphur atoms and/or NH- and/or N(C1-C4-alkyl)groups; wherein R and R are not simultaneously bound via heteroatoms to the carbon atom. The invention also relates to the salts of said derivatives, methods and intermediates for their preparation and use thereof.

    Abstract translation: 式(I),2-Iminooxyphenylessigsäurederivate其中取代基和指数具有以下含义:R t <1> C(CO 2 CH 3)= NOCH 3(Ia)中,C(CONHCH 3)= NOCH 3(Ib)中,C(CONH 2)= NOCH 3(Ic)中,C(CO2CH3)= CHOCH 3(同上)或C(CO2CH3)= CHCH3(IE); [R <2>氰基,硝基,卤素,烷基,卤代烷基或烷氧基; m是0,1或2; [R <3>是氢,氰基,羟基,卤素,烷基,卤代烷基,烷氧基烷基,烷氧基,卤代烷氧基,烷硫基,环丙基,链烯基,未取代的或取代的。 芳氧基烷基,苄基或苄氧基; [R <4>是氢,氰基,未取代的或取代的。 烷基,烯基,炔基,环烷基,杂环基,芳基和杂芳基; 未取代的或取代的。 烷氧基,烯氧基,炔氧基,环烷氧基,杂环氧基,芳氧基和杂芳氧基; 未取代的或取代的。 芳和杂芳硫基; -Q-C(R <5>)= N-Y <1> -R <6>或-Q-O-N = CR <7> - [R <8>; [R <3>和R <4>的碳原子一起形成它们所连接的未取代或取代的。 四到八位元环,其除了碳原子,一个或两个氧和/或硫原子和/或NH和/或N(C1-C4烷基)可以含有基团; 其中R <3>和R <4>不同时经由键合至的碳原子键合的杂原子; 和它们的盐,过程和它们的制备方法和它们的使用的中间体。

    IMINOOXYBENZYLCROTONIC ACID ESTERS, PROCESS FOR THEIR PREPARATION AND USE THEREOF
    98.
    发明申请
    IMINOOXYBENZYLCROTONIC ACID ESTERS, PROCESS FOR THEIR PREPARATION AND USE THEREOF 审中-公开
    IMINOOXYBENZYLCROTONSÄUREESTER,其制造方法相同,它们的用途

    公开(公告)号:WO1996016943A1

    公开(公告)日:1996-06-06

    申请号:PCT/EP1995004555

    申请日:1995-11-20

    CPC classification number: C07D239/26 A01N43/54 C07D239/34

    Abstract: The invention concerns iminooxybenzylcrotonic acid esters of formula (I) in which the index and the substituents have the following meanings: n is 0, 1, 2, 3 or 4; R is nitro, cyano, halogen, optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy or, if n stands for 2, additionally an optionally substituted bridge bonded to two adjacent ring atoms; R is a C1 to C4 alkyl; R is hydrogen or alkyl; R is hydrogen, cyano, halogen, alkyl, alkylhalide, alkoxy, alkoxyhalide, alkylthio, alkylthiohalide or cycloalkyl; and R is a 5 to 10-member mono or bicyclic substituted heteroaromatic cyclic system. The invention further concerns a process for their preparation and the use thereof.

    Abstract translation: 式(I),其中,所述索引和所述取代基具有以下含义的Iminooxybenzylcrotonsäureester:n为0,1,2,3或4; R是硝基,氰基,卤素,未取代或取代的。 烷基,烯基,炔基,烷氧基,链烯氧基,炔氧基或在n为2,另外一组键合至两个相邻的环原子未取代或取代的情况。 桥; [R <1> C1-C4烷基; [R <2>是氢或烷基; [R <3>为氢,氰基,卤素,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基或环烷基; [R <4>是一个5-10元单环或双环,取代的杂芳环体系,其制备方法和它们的使用方法。

    PHENYL ACETIC ACID DERIVATIVES, PROCESS AND INTERMEDIATE PRODUCTS FOR THEIR PRODUCTION AND AGENTS CONTAINING THEM
    99.
    发明申请
    PHENYL ACETIC ACID DERIVATIVES, PROCESS AND INTERMEDIATE PRODUCTS FOR THEIR PRODUCTION AND AGENTS CONTAINING THEM 审中-公开
    苯乙酸衍生物,PROCESS和中间产品FOR THEIR和代理CONTAINING THE SAME

    公开(公告)号:WO1995021153A1

    公开(公告)日:1995-08-10

    申请号:PCT/EP1995000013

    申请日:1995-01-03

    Abstract: Phenyl acetic acid derivatives of formula (I) in which the components and index have the following meanings: X is NOCH3, CHOCH3 CHCH3 and CHCH2CH3; R is hydrogen and alkyl; R is cyano, nitro, trifluoro methyl, halogen, alkyl and alkoxy; m is 0, 1 or 2, in which the radicals R may be different if m is 2; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, halogen alkyl, alkoxy, halogen alkoxy, alkylthio, alkylamino or dialkylamino; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, possibly substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, possibly substituted cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino, N-hetaryl-N-alkylamino; R is hydrogen, possibly substituted alkyl, cycloalkyl, alkenyl, alkinyl, alkyl carbonyl, alkenyl carbonyl, alkinyl carbonyl or alkyl sulphonyl; possibly substituted aryl, aryl carbonyl, aryl sulphonyl, hetaryl, hetaryl carbonyl or hetaryl sulphonyl; and their salts, process and intermediate products for their production and their use.

    Abstract translation: 式(I),其中取代基和指数具有以下含义的苯乙酸衍生物:X是NOCH 3,CHOCH 3,CHCH 3和CHCH 2; [R <1>是氢和烷基; [R <2>氰基,硝基,三氟甲基,卤素,烷基和烷氧基; m是0,1或2,其中基团可以是与R <2>中,当m是2不同; [R <3>是氢,氰基,硝基,羟基,氨基,卤素,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,烷基氨基或二烷基氨基; [R <4>为氢,氰基,硝基,羟基,氨基,卤素,未取代或取代的。 烷基,烷氧基,烷硫基,烷基氨基,二烷基氨基,烯基,烯氧基,烯硫基,链烯基,N-链烯基 - N-烷基氨基,炔基,炔氧基,炔硫基,炔基氨基,N-炔基 - N-烷基氨基; 未取代的或取代的。 环烷基,环烷氧基,环烷硫基,环烷基氨基,N-环烷基-N-烷基氨基,环烯基,环烯氧基,环烯硫基,cycloalkenylamino,N-环烯基-N-烷基氨基,杂环基,杂环氧基,杂环硫基,杂环基氨基,N-杂环基 - N-烷基氨基,芳基, 芳氧基,芳硫基,芳基氨基,N-芳基-N-烷基氨基,杂芳基,杂芳氧基,杂芳硫基,Hetarylamino,N-杂芳基的N-烷基氨基; [R <5>氢,未取代或取代的。 烷基,环烷基,烯基,炔基,烷基羰基,烯基羰基,炔基羰基或烷基磺酰基; 未取代的或取代的。 芳基,芳基羰基,芳基磺酰基,杂芳基,或hetarylcarbonyl hetarylsulfonyl; 和它们的盐,过程和它们的制备方法和它们的使用的中间体。

Patent Agency Ranking