公开(公告)号：EP0830342B1

公开(公告)日：2002-10-09

申请号：EP96916055.5

申请日：1996-05-13

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  KIRSTGEN, Reinhard ,  KÖNIG, Hartmann ,  RACK, Michael ,  OBERDORF, Klaus ,  RÖHL, Franz ,  SAUTER, Hubert ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07D231/22 ,  A01N43/56 ,  A01N43/653 ,  C07D231/18 ,  C07D249/12 ,  C07D401/04 ,  C07D403/04

CPC classification number: C07D401/04 ,  A01N43/56 ,  A01N43/653 ,  C07D231/20 ,  C07D249/12

公开(公告)号：EP0958276B1

公开(公告)日：2002-03-13

申请号：EP97953895.6

申请日：1997-12-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HILL, Regina, Luise ,  KARDORFF, Uwe ,  RACK, Michael ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  MAYER, Guido ,  OTTEN, Martina ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07C251/60 ,  C07C251/86 ,  A01N33/24 ,  A01N33/26

CPC classification number: A01N41/10 ,  A01N35/10 ,  A01N37/52 ,  C07C251/48 ,  C07C259/10 ,  C07C317/32 ,  C07C317/44 ,  C07C2601/16

Abstract: The invention concerns 2-benzoyl-cyclohexan-1,3-diones of formula (I), in which R , R stand for hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkyl, alkoxyalkyl, alkenyl, alkinyl, -OR , -OCOR , -OSO2R , -SH, -S(O)nR , -SO2OR , -SO2NR R , -NR SO2R or -NR COR ; R stands for hydrogen, cyano, alkyl, halogen alkyl, -OR , -SR or -NR R ; R stands for hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkinyl, -COR , -CO2R , -COSR or -CONR R ; X stands for oxygen or NR ; n equals 0, 1 or 2; R stands for hydrogen, alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R stands for alkyl or halogen alkyl; R stands for alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R stands for hydrogen or alkyl; R stands for alkyl, alkenyl, alkinyl, phenyl or benzyl; R stands for alkyl, halogen alkyl, alkenyl or alkinyl; Q stands for an optionally substituted cyclohexan-1,3-dione ring linked in position 2. Also disclosed are the salts of these compounds useful in agriculture; processes and intermediate products for preparing the compounds of formula (I), agents containing the same and the use of these derivatives or agents containing the same for controlling undesirable plants.

公开(公告)号：EP1163232A1

公开(公告)日：2001-12-19

申请号：EP00906364.5

申请日：2000-02-21

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WITSCHEL, Matthias ,  GÖTZ, Roland ,  RACK, Michael ,  PLATH, Peter ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D275/06 ,  A01N43/80

CPC classification number: C07D275/06 ,  A01N43/80

Abstract: The invention relates to saccharin 5 carbonyl derivatives of formula (I), wherein the substituents have the following meaning: L represents C1-C6-alkyl, C1-C6-alkoxy; Z represents C1-C6-alkyl, C3-C8-cycloalkyl, C3-C6-alkenyl, C3-C5-alkinyl, phenyl-C1-C6-alkyl or phenyl, wherein the phenyl rings are optionally substituted once or several times by C1-C6-alkyl, C1-C6-alkoxy or halogen; M represents hydrogen, C1-C6-alkyl, C1-C6-alkoxy, halogen, cyano, nitro or halogen-C1-C6-alkyl; R?1, R2, R3, R4, R5, R6, R7, R8¿ represent hydrogen, C¿1?-C6-alkyl. The invention also relates to the agriculturally usable salts of compound (I).

公开(公告)号：EP0973771A1

公开(公告)日：2000-01-26

申请号：EP98912471.4

申请日：1998-03-12

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MAYER, Guido ,  OTTEN, Martina ,  KARDORFF, Uwe ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  GÖTZ, Roland ,  RACK, Michael ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf ,  WALTER, Helmut

IPC: C07D417/04 ,  C07D417/14 ,  C07F9/6558 ,  A01N43/78 ,  A01N47/18 ,  A01N47/36

CPC classification number: C07D417/04 ,  A01N43/78 ,  A01N47/18 ,  A01N47/22 ,  A01N47/36 ,  A01N57/32 ,  C07D417/14 ,  C07F9/65586

Abstract: The invention relates to thiazolimines derivatives of formula (I), wherein the substituents have the following meanings: X, Y independently of each other stand for hydrogen, halogen, C1-C4-alkyl, C1-C4-haloalkyl, Z means hydrogen, C1-C8-alkyl, C2-C8-alkenyl, C2-C8-alkinyl, C1-C8-alkoxy, C1-C8-alkylthio, wherein these groups can be substituted by 1-5 halogen or C1-C4-alkoxy; aryl, hetaryl, benzyl, wherein these groups can be substituted with C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, halogen, nitro or cyano; or one of the following groups (a...); R1, R2 are hydrogen, halogen; C¿1?-C4-alkyl, C2-C4-alkenyl, C2-C4-alkinyl, wherein these groups can be substituted by 1-5 halogen or by C1-C4-alkoxy; n is 1 or 2; m is 0, 1 or 2, and R?3-R6¿ have the meaning cited in the application. The invention further relates to salts of compound I which can be used in agriculture.

公开(公告)号：EP0946514A1

公开(公告)日：1999-10-06

申请号：EP97953736.0

申请日：1997-12-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VOGELBACHER, Uwe, Josef ,  KEIL, Michael ,  KLINTZ, Ralf ,  WAHL, Joseph ,  WINGERT, Horst ,  KÖNIG, Hartmann ,  RACK, Michael ,  GÖTZ, Roland ,  TELES, Joaquim, Henrique

IPC: C07D231

CPC classification number: C07D231/22 ,  C07D231/20

Abstract: The invention relates to a method for producing n-substituted 3-hydroxypyrazoles of formula (I), wherein R1 stands for optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aryl or heteroaryl and R?2 and R3¿ mean hydrogen, cyano, halogen and optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, aryl or heteroaryl, by oxidizing a corresponding pyrazolidin-3-ons.

公开(公告)号：EP0812317B1

公开(公告)日：1999-09-08

申请号：EP96916056.3

申请日：1996-05-13

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  MÜLLER, Bernd ,  SAUTER, Hubert ,  OBERDORF, Klaus ,  KÖNIG, Hartmann ,  GÖTZ, Norbert ,  RACK, Michael ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried

IPC: C07D249/12 ,  C07D271/07 ,  C07D271/113 ,  C07D285/13 ,  C07D401/04 ,  C07D403/04 ,  C07D413/04 ,  C07D417/04 ,  A01N43/653 ,  A01N43/82

CPC classification number: C07D271/07 ,  A01N43/653 ,  A01N43/82 ,  C07D249/12 ,  C07D271/113 ,  C07D285/13 ,  C07D401/04

公开(公告)号：EP0934275A1

公开(公告)日：1999-08-11

申请号：EP97944808.0

申请日：1997-08-29

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HAMPRECHT, Gerhard ,  GEBHARDT, Joachim ,  ISAK, Heinz ,  RACK, Michael ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter

IPC: C07D213

CPC classification number: C07D213/71

Abstract: Substituted thiopyridines having general formula (I), wherein n means 1 or 2, R1 means chlorine, C¿1?-C3 fluoralkyl, nitro or methylsulfonyl; a non-substituted or halogen, C1-C4 - alkoxy, C1-C4 aloxycarbonyl, di- (C1-C4-alkylamino) carbonyl, cyano or nitro substituted C1-C10-Alkyl, C2-C10-alkenyl or C2-C10 alkinyl radical, a C3-C8-cycloalkyl radical or a non-substituted in the phenyl part or hydrogen, C1-C3-alkyl, C1-C3-alkoxy, trifluormethyl, cyano or nitro substituted C1-C4-alkylene phenyl, phenyl or naphthyl radical.

Abstract translation: 其中n表示1或2，R1表示氯，C1-C3烷基，硝基或甲基磺酰基; 未取代或卤素，C 1 -C 4烷氧基，C 1 -C 4烷氧基，二（C 1 -C 4烷基氨基）羰基，氰基或硝基取代的C 1 -C 10烷基，C 2 -C 10链烯基或C 2 -C 10炔基 苯基部分中的未取代的C 3 -C 8环烷基或氢，C 1 -C 3烷基，C 1 -C 3烷氧基，三氟甲基，氰基或硝基取代的C 1 -C 4亚烷基苯基，苯基或萘基。

公开(公告)号：EP0882025A1

公开(公告)日：1998-12-09

申请号：EP97901621.0

申请日：1997-01-31

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  BAYER, Herbert ,  GROTE, Thomas ,  KIRSTGEN, Reinhard ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  OBERDORF, Klaus ,  PTOCK, Arne ,  SAUTER, Hubert ,  RÖHL, Franz ,  RACK, Michael ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07D239 ,  A01N43

CPC classification number: C07D239/47 ,  A01N43/54 ,  C07D239/34

Abstract: The invention concerns pyrimidine derivatives of formula (I) in which the substituents have the following meanings: X is C(CO2CH3)=NOCH3, C(CONHCH3)=NOCH3, C(CO2CH3)=CHOCH3, C(CO2CH3)=CHCH3, N(CO2CH3)-OCH3; R?1 and R2¿, independently of each other, are hydrogen, C¿1?-C4 alkyl, C1-C4 alkyl halide or C1-C4 alkoxy; A is (i), the bond designated * being bonded to Y; R?3¿ is hydrogen, C¿1?-C4 alkyl, C1-C4 alkyl halide, phenoxy C1-C4 alkyl, C3-C6 cycloalkyl, cyano, C1-C4 alkoxy, hydroxy, halogen; R?4¿ is hydrogen, C¿1?-C8 alkyl, C1-C4 alkyl halide, C1-C6 cyanoalkyl, C1-C4 alkoxy-C1-C4 alkyl, C2-C4 alkenyloxy-C1-C4 alkyl, C1-C4 alkoxy halide-C1-C4 alkyl, C1-C4 oxoalkyl, C2-C4 alkenyl, C2-C4 alkinyl, C2-C4 alkenyl halide, C2-C4 alkinyl halide, C3-C6 cycloalkyl, C3-C6 cycloalkyl-C1-C4 alkyl, C1-C4 alkoxy; Y is hydrogen, hydroxy, halogen, optionally substituted aryl, hetaryl, cycloalkyl, cycloalkenyl, heterocyclyl, alkyl, alkenyl, alkinyl, alkyl halide, alkoxy, aryloxy, arylthio, hetaryloxy, hetarylthio, alkylthio or cycloalkyloxy; A not meaning -O- when X stands for C(CO2CH3)=CHOCH3. The invention also concerns the salts of these derivatives, a process and intermediate products for their preparation, and pesticides and fungicides containing them.

公开(公告)号：EP0851858A1

公开(公告)日：1998-07-08

申请号：EP96932485.0

申请日：1996-09-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  MENKE, Olaf ,  ZAGAR, Cyrill ,  RACK, Michael ,  GÖTZ, Norbert ,  HARREUS, Albrecht ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  MISSLITZ, Ulf

IPC: C07D213 ,  A01N43

CPC classification number: C07D213/61 ,  A01N43/40

Abstract: The invention concerns 2-phenylpyridines (I) and their salts, in which, n = 0, 1; R1 = halogen, C¿1?-C4 alkylhalide; R?2, R3¿ = H, halogen; R4 = CN, halogen; R5 = -CO-O-( C¿1?-C4 alkylene)-CO-OR?6¿, -CO-O-(C¿1?-C4 alkylene)-CO-N(R?7)R8¿, -O-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-OR?6¿, -O-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-N(R?7)R8¿, -S-(C¿1?-C4 alkylen)-CO-O-(C1-C4 alkylene)-CO-OR?6¿ or -S-(C¿1?-C4 alkylene)-CO-O-(C1-C4 alkylene)-CO-N(R?7)R8; R6¿ = H, C¿1?-C4 alkyl,(C1-C4 alkoxy)(C1-C4 alkyl), C2-C4 alkenyle, C3-C4 alkinyl; R?7¿ = H, C¿1?-C4 alkyl, carboxyl(C1-C4 alkyl), (C1-C4 alcoxycarbonyl)(C1-C4 alkyl); R?8¿ = H or C¿1?-C4 alkyl. Such compounds are suitable for use as herbicides and as plant desiccants/defoliants.

Abstract translation: 本发明涉及2-苯基吡啶（I）及其盐，其中n = 0,1; R1 =卤素，C1-C4烷基卤化物; R 2，R 3'= H，卤素; R4 = CN，卤素; R 5 = -CO-O-（C 1 -C 4亚烷基）-CO-OR 6，-CO-O-（C 1 -C 4亚烷基）-CO-N（R 7）R 8， （C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-OR 6'， - O-（C 1 -C 4亚烷基）-CO-O-（C1 （亚烷基）-CO-N（R 7）R 8，-S-（C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-OR 6或-S- （C 1 -C 4亚烷基）-CO-O-（C 1 -C 4亚烷基）-CO-N（R 7）R 8; （C 1 -C 4烷氧基）（C 1 -C 4烷基），C 2 -C 4烯烯基，C 3 -C 4炔基; R 6是H，C 1 -C 4烷基， （C 1 -C 4烷基），（C 1 -C 4烷氧基羰基）（C 1 -C 4烷基）; R 4为H，C 1 -C 4烷基。 R 8 = H或C 1 -C 4烷基。 这样的化合物适合用作除草剂和植物干燥剂/脱叶剂。

公开(公告)号：EP1863752A1

公开(公告)日：2007-12-12

申请号：EP06725104.1

申请日：2006-03-16

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： RACK, Michael ,  SMIDT, Sebastian, Peer ,  BUDICH, Manuel ,  MAYWALD, Volker ,  KEIL, Michael ,  WOLF, Bernd

IPC: C07C51/08 ,  C07C63/70 ,  C07C17/23 ,  C07C17/363 ,  C07C25/13

CPC classification number: C07C25/13 ,  C07C17/23 ,  C07C17/363 ,  C07C51/08 ,  C07C63/68

Abstract: The invention relates to a method for producing 5-halo-2,4,6-trifluoroisophthalic acid of formula (I), wherein X represents F, Cl, Br, or I, by hydrolysis of 5-halo-2,4,6-trifluoroisophthalodinitrile of formula (II). Said invention is characterised in that in a first step, isophthalodinitrile (II) or a solution containing isophthalodinitrile (II) is reacted with a concentrated sulphuric acid at room temperature in order to form a 5-haIo-2,4,6-trifluoroisophthalodiamide of general formula (III), and is, subsequently, heated and in a second step, isophthalic acid (I) is produced after additional heating and addition of water.

Abstract translation: 本发明涉及通过5-卤代-2,4,6,6-四氢吡啶的水解制备式（I）的5-卤代-2,4,6-三氟间苯二甲酸的方法，其中X代表F，Cl，Br或I （II）的三氟间苯二甲腈。 所述发明的特征在于，在第一步中，异佛尔酮二腈（II）或含有间苯二甲腈（II）的溶液在室温下与浓硫酸反应，以形成5-卤-2,4,6-三氟间苯二甲酰二胺 通式（III），随后加热，并且在第二步中，间苯二甲酸（I）在额外加热和加入水之后生成。