公开(公告)号：EP1177179A1

公开(公告)日：2002-02-06

申请号：EP00929502.3

申请日：2000-05-05

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MAYER, Guido ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MISSLITZ, Ulf ,  NEIDLEIN, Ulf ,  WITSCHEL, Matthias ,  RACK, Michael ,  VOLK, Thorsten ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D249/18 ,  C07D271/12 ,  C07D285/14 ,  C07D263/54 ,  C07D277/62 ,  C07D235/04 ,  A01N43/647 ,  A01N43/78 ,  A01N43/828 ,  A01N43/76

CPC classification number: C07D263/56 ,  A01N43/74 ,  C07D249/18 ,  C07D263/58 ,  C07D277/62 ,  C07D277/64 ,  C07D277/66 ,  C07D277/68 ,  C07D277/74 ,  C07D285/14

Abstract: The invention relates to cyclohexenone derivatives of benzo-condensed, unsaturated 5-ring nitrogen heterocycles of general formula (I) wherein X represents N or a group C-R3, Y represents O, S, SO, SO¿2? or NR?4¿ or X-Y represent S=N and X represents sulfur, and the variables R1, R2 and Hex have the meanings given in claim 1. The invention also relates to a method for producing these compounds, to agents containing these compounds, and to their use as herbicides.

Abstract translation: 本发明涉及通式（I）的苯并稠合不饱和5-环氮杂环的环己烯酮衍生物，其中X代表N或基团C-R3，Y代表O，S，SO，SO2- 或NR 4'或XY代表S = N且X代表硫，变量R 1，R 2和Hex具有权利要求1中给出的含义。本发明还涉及制备这些化合物的方法，含有这些化合物的试剂， 并涉及它们作为除草剂的用途。

公开(公告)号：EP1131298A2

公开(公告)日：2001-09-12

申请号：EP99957286.0

申请日：1999-11-06

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MAYWALD, Volker ,  STEINMETZ, Adrian ,  RACK, Michael ,  GÖTZ, Norbert ,  GÖTZ, Roland ,  HENKELMANN, Jochem ,  BECKER, Heike ,  AISCAR BAYETO, Juan Jose

IPC: C07D231/20

CPC classification number: C07D231/20

Abstract: The invention relates to a method for the production of 1-substituted 5-hydroxypyrazoles of formula (I) wherein R1 is C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C6-cycloalkyl or C1-C4-alkoxy, whereby these groups can be substituted by halogen, C1-C4-alkoxy, phenoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthiocarbonyl or a cyclic ring system with 3-14 ring atoms, by reacting a) an alkylvinylether of general formula (III) wherein R2 is C1-C6-alkyl or C3-C6-cycloalkyl, with phosgene (IVa), 'diphosgene' (IVb) or 'triphosgene' (IVc) to form acid chlorides of formula (V), b) transforming said acid chlorides by eliminating hydrogen chloride into the corresponding 3-alkoxyacrylic acid chloride of formula (VI) and c) reacting said acid chloride with hydrazines of formula (VII) wherein R1 has the above cited meaning, to form 5-hydroxypyrazoles of formula (I).

公开(公告)号：EP1034166A1

公开(公告)日：2000-09-13

申请号：EP98945309.7

申请日：1998-09-05

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  MENGES, Markus ,  MENKE, Olaf ,  RACK, Michael ,  REINHARD, Robert ,  ZAGAR, Cyrill ,  MÜNSTER, Peter ,  WESTPHALEN, Karl-Otto ,  OTTEN, Martina ,  WALTER, Helmut

IPC: C07D237/20 ,  C07D405/10 ,  A01N43/58

CPC classification number: C07D405/10 ,  A01N43/58 ,  C07D237/22

Abstract: The invention concerns substituted 2-phenyl-3(2H)-pyridazinones of formula (I), and their salts. In said formula, n = 0, 1, 2; R1 = alkyl C¿1?-C4, alkyl halide C1-C4; R?2¿ = H, halogen; R3 = halogen, CN; R4 = H, NO¿2?, CN, CHO, NH-OH, alkyl C1-C4, alkyl halide C1-C4, -OR?5¿, -CH=N-OR6, -CH=C(R?7)-CO-OR8¿, -CO-OR9, alkyl C¿1?-C6 -SO2-NH, di(alkylsulphonyl C1-C6)amino or (a); R?5¿ = alkyl C¿1?-C6, alkenyl C3-C6, alkinyl C3-C6, (alkoxy C1-C6)carbonyl-alkyl C1-C4, (alkenyloxy C3-C6)carbonyl-alkyl C1-C4, (alkinyloxy C3-C6)carbonyl-alkyl C1-C4, alkoxy C1-C4-(alkoxy C1-C4) carbonyl-alkyl C1-C4; R?6¿ = H, alkyl C¿1?-C4, hydroxycarbonyl-alkyl C1-C4, (alkoxy C1-C4) carbonyl-alkyl C1-C4; R?7¿ = H, halogen, alkyl C¿1?-C4; R?8¿ = H, alkyl C¿1?-C6; R?9¿ = H, alkyl C¿1?-C6, alkenyl C3-C6, alkinyl C3-C6, alkoxy-C1-C4-alkoxy C1-C4, hydroxycarbonyl-alkyl C1-C4, (alkoxy C1-C6)carbonyl-alkyl C1-C4, (alkenyloxy C3-C6)carbonyl-alkyl C1-C4, (alkinyloxy C3-C6)carbonyl-alkyl C1-C4, alkoxy C1-C4-(alkoxy C1-C4)carbonyl-alkyl C1-C4; R?10¿ = H, alkyl C¿1?-C6, COOH, (alkoxy C1-C6)carbonyl. Said compounds are used as herbicides for desiccation/defoliation of plants.

公开(公告)号：EP1003725A1

公开(公告)日：2000-05-31

申请号：EP98942623.4

申请日：1998-07-25

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： EICKEN, Karl ,  RACK, Michael ,  WETTERICH, Frank ,  AMMERMANN, Eberhard ,  LORENZ, Gisela ,  STRATHMANN, Siegfried

IPC: C07D231/16 ,  A01N43/48

CPC classification number: C07D231/16 ,  A01N43/56

Abstract: The invention relates to biphenylamides having general formula (I), and their salts, in which R1 is H or F; R2 is H, halogen, alkyl, halogen methyl, alkoxy, alkylthio; R3 is CH¿3?, CHF2, CF3. The invention also relates to agents containing biphenylamides, the production of biphenylamides and their use in combating parasitic fungus.

公开(公告)号：EP0984914A1

公开(公告)日：2000-03-15

申请号：EP98924202.9

申请日：1998-04-24

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  MAYER, Guido ,  OTTEN, Martina ,  RACK, Michael ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf ,  WALTER, Helmut

IPC: C07C49/835 ,  C07C49/813 ,  C07C205/45 ,  C07C317/24 ,  C07C45/54 ,  A01N35/06

CPC classification number: C07D307/38 ,  A01N35/06 ,  A01N35/10 ,  A01N37/42 ,  A01N37/50 ,  A01N43/08 ,  A01N43/10 ,  A01N43/30 ,  C07C45/46 ,  C07C45/54 ,  C07C49/813 ,  C07C49/835 ,  C07C49/84 ,  C07C49/86 ,  C07C69/76 ,  C07C205/45 ,  C07C205/56 ,  C07C251/40 ,  C07C251/52 ,  C07C255/40 ,  C07C317/24 ,  C07C323/22 ,  C07C2601/16 ,  C07D319/06 ,  C07D333/12 ,  C07C49/807

Abstract: The invention relates to 2-(3-alkenyl-benzoyl)-cyclohexane-1,3-diones of formula (I), wherein the variables can have the following meanings: R1, R2 = hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkane, alkoxyalkyl, alkenyl, alkinyl, -OR?6, -OCOR7¿, -OSO¿2R?7, -SH, -S(O)nR8, -SO2OR6, -SO2NR?6R9, -NR9SO¿2R?7 or -NR9COR7; R3¿ = hydrogen, halogen, alkyl, halogen alkane, alkoxy, alkenyl, alkinyl; R4, R5 = hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkane, cycloalkyl, alkenyl, cycloalkenyl, alkinyl, alkythio, halogen alkoxy, -COR10, -CO2R?10, -COSR10, -C(R12)=NR13¿, -PO(OR?10) (OR11¿); optionally substituted alkyl, heterocyclyl, heterocyclylalkyl, phenyl, phenylalkyl, hetaryl or hetarylalkyl; or R?4 and R5¿ together form an alkandiyl chain which can be substituted and/or interrupted by a heteroatom; Q = an unsubstituted or substituted position 2 bonded cyclohexane-1,3-dione ring. The invention further relates to the salts thereof, which can be used in agriculture. The invention also relates to a method for the production of compounds of formula (I), to agents containing said compounds and to the use of said derivatives or agents containing said compounds to control undesired plants.

公开(公告)号：EP0873313B1

公开(公告)日：2000-03-15

申请号：EP96934777.2

申请日：1996-10-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  SAUTER, Hubert ,  BAYER, Herbert ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  RÖHL, Franz ,  GÖTZ, Norbert ,  RACK, Michael ,  MÜLLER, Ruth ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07D213/54 ,  A01N43/40

CPC classification number: C07D213/56 ,  A01N43/40 ,  C07D213/55

Abstract: The invention concerns pyridylacetic acid derivatives of formula (I) in which the substituents and the index have the following meanings: X is NOCH3, CHOCH3 and CHCH3; Y is oxygen or NRa; Ra is hydrogen or alkyl; R is cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m is 0, 1 or 2; R1 is hydrogen or alkyl; R?2 and R3¿, independently of each other, stand for hydrogen, cyano, nitro, hydroxy, amino, halogen, optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino, cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino or N-hetaryl-N-alkylamino; R4 is one of the groups mentioned under R2 or a CRd =NORe group. The invention further concerns their salts, a process and intermediate products for their preparation and their use.

公开(公告)号：EP0929546A1

公开(公告)日：1999-07-21

申请号：EP97943851.0

申请日：1997-09-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OTTEN, Martina ,  GÖTZ, Norbert ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  KARDORFF, Uwe ,  RACK, Michael ,  HILL, Regina, Luise ,  PLATH, Peter ,  WITSCHEL, Matthias ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  MISSLITZ, Ulf

IPC: A01N43 ,  C07D401

CPC classification number: C07D401/06 ,  A01N43/56

Abstract: Hetaroyl derivatives having the formula (I) are disclosed, as well as their salts useful in agriculture. In the formula, the variables have the following meanings: R1, R2 are hydrogen, nitro, halogen, cyano, rhodano, hydroxy, mercapto, optionally substituted and/or functionalised C¿1?-C6 alkyl, C1-C6 alkoxy, C1-C6 alkylthio, C1-C6 alkylsulfinyl, C1-C6 alkylsulfonyl, C1-C6 alkoxysulfonyl, or optionally substituted phenyl, phenoxy, phenylthio, phenylsulfinyl or phenylsulfonyl; Z is an optionally substituted, 4-membered, unsaturated, partially or completely saturated chain with three carbon atoms and one nitrogen atom; and Q is optionally substituted hydroxypyrazol of Formula (II) linked at position 4 in addition to the salts thereof which can be used in agriculture. Also disclosed is a process for preparing the hetaroyl derivatives, agents containing the same, as well as the use of these derivatives or the agents containing the same for controlling undesirable plants.

公开(公告)号：EP0876351A1

公开(公告)日：1998-11-11

申请号：EP96943127.0

申请日：1996-12-16

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： KIRSTGEN, Reinhard ,  BAYER, Herbert ,  GÖTZ, Norbert ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  MÜLLER, Bernd ,  MÜLLER, Ruth ,  OBERDORF, Klaus ,  RACK, Michael ,  RÖHL, Franz ,  SAUTER, Hubert ,  AMMERMANN, Eberhard ,  HARRIES, Volker ,  LORENZ, Gisela ,  STRATHMANN, Siegfried

IPC: A01N43 ,  C07D231

CPC classification number: C07D231/12 ,  A01N43/56 ,  C07D231/22

Abstract: Compounds of the general formula (I) and their salts, in which the variables mean: n is 0, 1, 2, 3 or 4, where the radical R1 may be different if n is greater than 1; Q is -C(=CHCH¿3?)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-NH(CH3); Het is a possibly substituted pyrazol ring; R?1¿ is nitro, cyano, halogen, C¿1?-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkylthio or possibly substituted phenyl, phenoxy or, if n is greater than 1, a possible substituted 1,3 butadiene-1,4-diyl group bonded to two adjacent carbon atoms of the phenyl radical; R?2¿ is hydrogen or a possible substituted one or two-nuclear carbo or heterocyclic aromatic ring which is bonded to the radical Het directly or via a (-CR?3R4-) [R3, R4¿ = H or alkyl or -CR3R4- = (-C(=O)-) or (-C(=NOR?5)-); R5¿ = alkyl or alkinyl], agents containing them and the use of the compounds (I) and the agents to combat damaging fungi and animal pests.

公开(公告)号：EP0873316A1

公开(公告)日：1998-10-28

申请号：EP96943079.0

申请日：1996-12-11

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OBERDORF, Klaus ,  GRAMMENOS, Wassilios ,  SAUTER, Hubert ,  GROTE, Thomas ,  KIRSTGEN, Reinhard ,  MÜLLER, Ruth ,  MÜLLER, Bernd ,  RÖHL, Franz ,  RACK, Michael ,  BAYER, Herbert ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried ,  HARRIES, Volker

IPC: C07D239 ,  A01N43 ,  A01N47 ,  A01P3

CPC classification number: C07D239/34 ,  A01N43/54

Abstract: 2-(O-[pyrimidin-4-yl]methylenoxy)phenyl acetic acid derivatives are disclosed having the general formula (I), as well as their salts and N-oxides. In the formula, the radicals R1 to R4 and Q have the following meanings: R1 stands for hydrogen or alkyl; R2 stands for halogen, alkyl or alkyl halide; R3 stands for hydrogen, amino, hydroxy, mercapto, halogen, optionally phenyl-substituted alkyl, alkyl halide, alkoxyalkyl, alkoxy, monoalkylamino, dialkylamino, alkylthio, alkylsulphoxyl, alkylsulphonyl, cycloalkyl, trialkylsilyloxy or in the aromatic ring optionally substituted phenyl, phenoxy, phenoxymethyl, benzyloxy or heteroaryl; R4 stands for hydrogen, cyano, halogen, alkyl, alkyl halide or alkoxy; Q stands for C(=NOCH¿3?)-CONHCH3, C(=NOCH3)-COOCH3 or N(OCH3)-COOCH3. Also disclosed are their salts and N-oxides and their use for controlling harmful fungi and animal pests.

公开(公告)号：EP0851863A1

公开(公告)日：1998-07-08

申请号：EP96931781.0

申请日：1996-09-09

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAYER, Herbert ,  MÜLLER, Ruth ,  SAUTER, Hubert ,  RACK, Michael ,  HARREUS, Albrecht ,  AMMERMANN, Eberhard ,  HARRIES, Volker ,  LORENZ, Gisela ,  STRATHMANN, Siegfried

IPC: C07D295 ,  A01N37 ,  A01N43 ,  C07D207 ,  C07D209 ,  C07D231 ,  C07D233 ,  C07D235 ,  C07D249 ,  C07D257 ,  C07D261 ,  C07D263 ,  C07D271 ,  C07D521

CPC classification number: C07D249/08 ,  A01N37/50 ,  A01N43/50 ,  A01N43/56 ,  C07D209/08 ,  C07D209/30 ,  C07D209/42 ,  C07D231/12 ,  C07D231/14 ,  C07D231/56 ,  C07D233/56 ,  C07D233/82 ,  C07D233/90 ,  C07D233/91 ,  C07D235/24 ,  C07D249/04 ,  C07D249/10 ,  C07D249/18 ,  C07D257/04 ,  C07D295/195

Abstract: The invention concerns phenylacetic acids of formula (I) in which the substituents and the index have the following meanings: X is NOCH3, CHOCH3, CHCH3 and CHCH2CH3; Y = O and NR (R = hydrogen and alkyl); Z is an optionally substituted nitrogen atom-bonded heterocyclyl or heteroaryl; R1 = hydrogen and alkyl; R2 = cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m = 0, 1 or 2; R3 = hydrogen, cyano, nitro, hydroxy, amino, cyclopropyl, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylamino and dialkylamino; R4 = hydrogen, optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, alkylsulphonyl, cycloalkyl, aryl, arylcarbonyl, arylsulphonyl, hetaryl, hetarylcarbonyl and hetarylsulphonyl. The invention further concerns salts thereof, processes for their preparation and agents containing them.