Abstract:
Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.
Abstract translation:取代的式(I)的6-(2-卤代苯基) - 三唑并嘧啶,其中R1表示烷基,烯基,炔基,链二烯基,卤代烷基,卤代烯基,环烷基,苯基,萘基或5-或6-元饱和,不饱和或 芳族杂环,其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子,其中R 1和R 2基团可以如说明书中所定义地被取代,R 2表示氢,或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环,该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1,L 3独立地表示氢,卤素或烷基; L 2是氢,卤素,卤代烷基或NH 2,NHR b或N(R b)2,其中R b如说明书中所定义,其中至少一个L 1,L 2, 而L 3不是氢; X是卤素,氰基,烷基,烷氧基,卤代烷氧基或烯氧基,它们的制备方法,含有它们的组合物和它们用于防治植物病原性真菌的用途。
Abstract:
Disclosed are compounds of formula (I), wherein X, Y, and Z are defined as indicated in the description, methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant pathogenic fungi.
Abstract:
The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.
Abstract:
The present invention relates to compounds of the general formula (I) and to the salts thereof, wherein the substituents and the n index have the following values: Q represents -C(=CHCH3)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-CONH(CH3); R represents hydrogen, halogen, C1-C4 alkyl, C1-C2 halogenalkyl, C1-C4 alkoxy or C1-C2 halogenalkoxy; R represents halogen, C1-C4 alkyl, C1-C2 halogenalkyl or C1-C4 alkoxy; n is 0, 1 or 2, wherein the R substituents can be different when n = 2; and R represents phenyl, pyridyle or pyrimidyle. This invention also relates to agents containing these compounds as well as to the use of said compounds (I) and agents against noxious fungi and animal parasites.
Abstract translation:通式(I)和它们的盐,其中取代基和指数n具有以下含义的化合物:Q是-C(= CHCH 3)-COOCH 3,-C(= CHOCH 3)-COOCH 3,C(= NOCH 3) - COOCH 3或-C(= NOCH 3)-CONH(CH 3); R 1是氢,卤素,C 1 -C 4烷基,C 1 -C 2卤代烷基,C 1 -C 4烷氧基或C 1 -C 2卤代烷氧基; R 2是卤素,C 1 -C 4烷基,C 1 -C 2卤代烷基,C 1 -C 4烷氧基; n是0,1或2,其中当n = 2时取代基R 2可以不同; R 3苯基,吡啶基或嘧啶基,含有它们的试剂以及化合物(I)和防治有害真菌和动物害虫的试剂的用途。
Abstract:
Phenyl acetic acid derivatives of formula (I) in which the substituents and index have the following meanings: X is oxygen or sulphur; R is hydrogen and alkyl; R is hydrogen and alkyl; R is cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m is 0, 1 ou 2, in which the radicals R may be different if m is 2; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, halogen alkyl, alkoxy, halogen alkoxy, alkylthio, alkylamino or dialkylamino; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, possibly substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino; optionally substituted cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocylcyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, n-aryl-n-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino, N-hetaryl-N-alkylamino; R is hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl or alkylsulfonyl; optionally substituted aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl or hetarylsulphonyl; and their salts, process and intermediate products for their production, and their use.
Abstract:
The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.
Abstract:
The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R ; n stands for 1, 2, 3, 4 or 5; R represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R , and R represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.
Abstract:
Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.
Abstract:
The invention relates to substituted phenyl carbamates of formula (I), wherein E represents a group A or B, # characterises the bond with the phenyl ring, and R , R , Y, n, T, and Z have the meanings given in the description.