公开(公告)号：WO2004041824A2

公开(公告)日：2004-05-21

申请号：PCT/EP0312276

申请日：2003-11-04

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 取代的式（I）的6-（2-卤代苯基） - 三唑并嘧啶，其中R1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或 芳族杂环，其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义地被取代，R 2表示氢，或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或N（R b）2，其中R b如说明书中所定义，其中至少一个L 1，L 2， 而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基，它们的制备方法，含有它们的组合物和它们用于防治植物病原性真菌的用途。

公开(公告)号：WO2007116011A3

公开(公告)日：2007-12-21

申请号：PCT/EP2007053355

申请日：2007-04-05

Applicant: BASF AG ,  DIETZ JOCHEN ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH

Inventor： DIETZ JOCHEN ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: Disclosed are compounds of formula (I), wherein X, Y, and Z are defined as indicated in the description, methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant pathogenic fungi.

Abstract translation: 其中X，Y和Z如所述定义的式（I）化合物，用于制备这些化合物的方法和中间体，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

公开(公告)号：WO2006079556A2

公开(公告)日：2006-08-03

申请号：PCT/EP2006000774

申请日：2006-01-30

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  NAVE BARBARA ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  JABS THORSTEN ,  BLETTNER CARSTEN

Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  NAVE BARBARA ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  JABS THORSTEN ,  BLETTNER CARSTEN

IPC: A61K31/506 ,  A61K31/505 ,  C07D239/42 ,  C07D239/48 ,  C07D401/04 ,  C07D403/04 ,  C07D417/04

CPC classification number: C07D239/48 ,  C07D239/42 ,  C07D401/04 ,  C07D403/04 ,  C07D417/04

Abstract: The present invention relates to substituted 5-phenyl pyrimidines I, which carry a radical X in the 4-position of the pyrimidine ring, a radical Y in the 6-position of the pyrimidine ring, the radical X denoting a group of the formula NR 1 R 2 , OR 1a or SR 1a , in which R 1 , R 2 , independently of each other, denote hydrogen, C 1 -C 10 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which radicals may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 ; or the radical NR 1 R 2 may also form a 5- or 6-membered optionally substituted heterocyclic ring, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which are non-adjacent to the nitrogen of NR 1 R 2 , in which two adjacent C atoms or one N atom and one adjacent C atom can be linked by a C 1 -C 4 -alkylene chain and wherein the heterocyclic ring may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 as defined in claim 1, R 1a has one of the meanings given for R 1 except for hydrogen; the radical Y being selected from the group consisting of halogen, cyano, C 1 -C 4 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 3 -C 4 -alkynyloxy, C 1 -C 6 -alkylthio, di-(C 1 -C 6 -alkyl)amino or C 1 -C 6 -alkylamino, where the alkyl, alkenyl and alkynyl radicals of Y may be substituted by halogen, cyano, nitro, C 1 -C 2 -alkoxy or C 1 -C 4 -alkoxycarbonyl; and wherein the pyrimidine radical may also carry a radical different from hydrogen in the 2-position and wherein the phenyl ring in the 5-position of the pyrimidine ring may be unsubstituted or carry 1, 2, 3, 4 or 5 radicals L which are different from hydrogen, and the pharmaceutically acceptable salts substituted 5-phenyl pyrimidines for use in therapy, in particular in therapy or treatment of cancerous diseases.

Abstract translation: 本发明涉及取代的5-苯基嘧啶I，其在嘧啶环的4-位上携带基团X，嘧啶环的6-位的基团Y，基团X表示式NR的基团 其中R 1，R 2，R 2，R 1，R 2， R 2彼此独立地表示氢，C 1 -C 10 - 烷基，C 2 - C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 10 - C 1 -C 3烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代烷基，C 3 -C 8 - 苯基或含有1,2,3或4个氮原子或1,2或3个氮原子和一个硫或氧原子作为环成员的5-或6-元杂芳基或5-或6-元杂环基，该基团可以 未被取代或可以携带1,2,3或4个基团R a1a; 或自由基NR 1 R 2还可以形成含有1,2,3或4个氮原子或1,2或2个氮原子的5或6元任选取代的杂环 或3个氮原子和一个硫或氧原子作为环成员，其与NR 1 R 2 O 2的氮不相邻，其中两个相邻的C原子或一个 N原子和一个相邻的C原子可以通过C 1 -C 4 - 亚烷基链连接，并且其中杂环可以是未取代的或可以携带1,2,3 或如权利要求1所定义的4个基团R a1，其中R 1a除了氢之外具有R 1给出的含义之一; 基团Y选自卤素，氰基，C 1 -C 4 - 亚烷基，C 2 -C 3 - 烷基， 4 - 烯基，C 2 -C 4 - 炔基，C 3 -C 6 - 环烷基，C 1 -C 4 - 烷氧基，C 3 -C 4 - 炔基氧基，C 1 -C 4 - 3-C 4 - 炔基氧基，C 1 -C 6 - 烷硫基，二 - （C 1 -C 6） C 1 -C 6 - 烷基）氨基或C 1 -C 6 - 烷基氨基，其中Y的烷基，烯基和炔基可以 被卤素，氰基，硝基取代，C 1 -C 2 - 烷氧基或C 1 -C 4 - - 烷氧基; 并且其中嘧啶基团还可以携带2-位上与氢不同的基团，其中嘧啶环的5-位上的苯环可以是未取代的或携带1,2,3,4或5个基团L，其为 不同于氢，以及用于治疗，特别是治疗或治疗癌性疾病的药学上可接受的盐取代的5-苯基嘧啶。

公开(公告)号：WO0238565A3

公开(公告)日：2003-10-09

申请号：PCT/EP0112977

申请日：2001-11-09

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.

Abstract translation: 7-（R）式（I）的-aminotriazolopyrimidine其中取代基和指数具有以下含义：R t <1>是氢或甲基; [R <2>是甲基; [R <3> C2-C10烷基，C1-C4烷氧基，C3-C10环烷基; [R <4>为卤素，C1-C4烷基，C1-C4卤代烷基或C1-C4烷氧基; n是从1到5的数; Y是卤素，氰基，C1-C4烷基或C1-C4烷氧基; 其中*是R构型的手性中心。 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9940082A3

公开(公告)日：1999-10-21

申请号：PCT/EP9900470

申请日：1999-01-26

Applicant: BASF AG ,  PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

Inventor： PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D401/12 ,  C07D401/14 ,  A01N43/48

CPC classification number: C07D401/12 ,  A01N43/56

Abstract: The present invention relates to compounds of the general formula (I) and to the salts thereof, wherein the substituents and the n index have the following values: Q represents -C(=CHCH3)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-CONH(CH3); R represents hydrogen, halogen, C1-C4 alkyl, C1-C2 halogenalkyl, C1-C4 alkoxy or C1-C2 halogenalkoxy; R represents halogen, C1-C4 alkyl, C1-C2 halogenalkyl or C1-C4 alkoxy; n is 0, 1 or 2, wherein the R substituents can be different when n = 2; and R represents phenyl, pyridyle or pyrimidyle. This invention also relates to agents containing these compounds as well as to the use of said compounds (I) and agents against noxious fungi and animal parasites.

Abstract translation: 通式（I）和它们的盐，其中取代基和指数n具有以下含义的化合物：Q是-C（= CHCH 3）-COOCH 3，-C（= CHOCH 3）-COOCH 3，C（= NOCH 3） - COOCH 3或-C（= NOCH 3）-CONH（CH 3）; R 1是氢，卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基或C 1 -C 2卤代烷氧基; R 2是卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基; n是0,1或2，其中当n = 2时取代基R 2可以不同; R 3苯基，吡啶基或嘧啶基，含有它们的试剂以及化合物（I）和防治有害真菌和动物害虫的试剂的用途。

公开(公告)号：WO2007006806A3

公开(公告)日：2007-03-22

申请号：PCT/EP2006064199

申请日：2006-07-13

Applicant: BASF AG ,  GEWEHR MARKUS ,  STIERL REINHARD ,  DIETZ JOCHEN ,  MUELLER BERND ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  WERNER FRANK ,  VONEND MICHAEL

Inventor： GEWEHR MARKUS ,  STIERL REINHARD ,  DIETZ JOCHEN ,  MUELLER BERND ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  WERNER FRANK ,  VONEND MICHAEL

IPC: A01N43/56

CPC classification number: A01N43/56 ,  A01N47/14 ,  A01N37/34 ,  A01N43/653 ,  A01N37/50 ,  A01N47/24 ,  A01N43/54 ,  A01N35/04 ,  A01N47/38 ,  A01N37/38 ,  A01N2300/00

Abstract: The invention relates to fungicide mixtures containing, as active components in a synergistically active quantity: 1) 1-methyl-pyrazol-4-yl carboxylic acid anilides (I) wherein X represents oxygen or sulphur, R1 represents halogen, d-C4-alkyl or d-C4-halogenalkyl, R2 represents H or halogen, and R3 represents nitro, cyano, halogen, CrC4-alkyl, CrC4-halogenalkyl, CrC4-alkoxy, CrC4-halogenalkoxy or Ci -C4-alkylthio, and 2) at least one active ingredient II, selected from the active ingredient groups A) to F): A) azoles; B) strobilurine; C) carboxylic acid amides; D) heterocyclic compounds; E) carbamates; F) other fungicides. The invention also relates to a method for controlling pathogenic fungi using mixtures consisting of at least one compound I and at least one active ingredient II, to the use of the compound(s) I with active ingredients II for producing such mixtures, and to agents and seeds containing said mixtures.

Abstract translation: 一种杀真菌混合物，包含：1）1-甲基 - 吡唑-4-ylcarbonsäureanilide（I），其中X =氧或硫，R ^{1 为卤素，C作为活性组分 _{1 -C 4 烷基或C 1 -C 4 - 卤代烷基，R 2 = H或卤素，R 3 =硝基，氰基，卤素，C 1 -C 4 烷基，C 1 -C 4 卤代烷基，C 1 -C 4 烷氧基，C 1 -C 4 卤代烷氧基或C 1 -C 4 代表烷硫基和2）至少一种选自活性化合物组a）至f）中选择的活性化合物II：A）唑类; B）嗜球果伞素; C）羧酸酰胺; D）杂环化合物; E）氨基甲酸酯; F）其他杀菌剂; 在协同有效量，用于控制使用至少一种化合物I和至少一种活性化合物II，使用了化合物（S）1与活性化合物II在制备该类混合物和组合物和种子，其包含这些混合物的混合物防治有害真菌的方法。}}

公开(公告)号：WO2006114405A2

公开(公告)日：2006-11-02

申请号：PCT/EP2006061786

申请日：2006-04-24

Applicant: BASF AG ,  DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA

Inventor： DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA

IPC: A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.

Abstract translation: 式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I：其中各变量具有以下含义：Y是任选被烷基取代的亚烷基，亚烯基或亚炔基; [R ^{1 为卤素，氰基，硝基，羟基，巯基，烷基，卤代烷基，链烯基，环烷基，环烯基，烷氧基，卤代烷氧基，烯氧基，炔氧基，烷硫基，NR 一 - [R < SUP>乙，烷基羰基，苯基，萘基或五 - 或六元饱和环，其包含选自一至四个杂原子的部分不饱和或罗马杂环O，N或S; [R 一，R 乙是氢，烷基和烷基羰基; n是零，1，2，3或4; [R 2 烷基，烯基，环烷基，烷氧基烷基和烷硫基烷基; [R 3 为氢，卤素，氰基，NR 一 - [R 乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基， 环烷硫基，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O）_{米 - ; m是0，1或2; A N和C-R 一; [R 一氢和烷基; 其中Y中的碳原子，R 1 ，R 2 ，R 3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines，处理用于制备这些化合物和含有它们的组合物。}}

公开(公告)号：WO2005087771A3

公开(公告)日：2005-12-01

申请号：PCT/EP2005002425

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl or alkoxyalkyl; R represents alkyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 式（I）的5,6-二烷基 - 7-氨基 - 三唑并嘧啶，其中取代基具有以下含义：R t <1>是烷基或烷氧基烷基，R <2>是烷基，其中R <1>和/或R <2> 可以如上所述被替换; 这些化合物的制备方法，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

公开(公告)号：WO2005080396A2

公开(公告)日：2005-09-01

申请号：PCT/EP2005001965

申请日：2005-02-24

Applicant: BASF AG ,  SCHWOEGLER ANJA ,  GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

Inventor： SCHWOEGLER ANJA ,  GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA

IPC: A01N43/90 ,  C07D487/04 ,  C07D487/00

CPC classification number: C07D487/04

Abstract: The invention relates to azolopyrimidine compounds of general formula (I), wherein A represents N or C-R ; X and Y, independent of one another, represent a chemical compound or oxygen, sulphur or a group N-R ; the variables R , R , R , R , R , R and R have the meanings cited in the claims and the description. The invention also relates to tautomers of compounds of formula (I) and to the agriculturally compatible salts of compounds (I) and of the tautomers thereof. The invention further relates to the use of azolopyrimidine compounds of general formula (I), to the tautomers thereof and to the agriculturally compatible salts thereof which are used to combat phytopathogenic fungi, and to a method for combating phytopathogenic fungi and means for combating fungi, said means containing at least one compound of general formula (I), a tautomer of formula (I) and/or an agriculturally compatible salt thereof or the tautomer thereof and at least one liquid or solid carrier medium.

Abstract translation: 本发明涉及通式（I）的唑基嘧啶化合物，其中A是N或C-R 6; X，Y彼此独立地代表化学键或氧，硫或基团N-R 7; 其中变量R <1>，R <2>，R <3>，R <4>，R <5> - [R <6>和R <7>具有权利要求书所给出的含义和描述中，互变异构体 式（I）化合物和化合物I及其互变异构体的农业上可接受的盐。 本发明还涉及使用通式（I）的唑并嘧啶化合物，它们的互变异构体以及它们用于防治植物致病真菌（=有害真菌），以及用于防治植物病原性有害真菌的方法和用于防治有害真菌的手段农业上可接受的盐，含 至少一种通式（I）的化合物，（I）的互变异构体和/或其农业上可接受的盐或其互变异构体以及至少一种液体或固体载体。

公开(公告)号：WO03008417A9

公开(公告)日：2003-10-30

申请号：PCT/EP0207578

申请日：2002-07-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 式（I）的取代的6-（2-甲苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5-或6-元杂环基，或者含有1-4个氮原子或1-3个氮原子的5-或6-元杂芳基， 硫或氧原子，或者其中R 1和R 2基团可以如说明书中所定义的那样未被取代或被取代，或者R 1和R 2与中间的氮原子一起表示5或6 - 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的可被取代的 - 元杂环; R 3是卤素，氰基，烷基，烷氧基，卤代烷基或C（= O）A，其中A是氢，羟基，烷基，氨基或单或二烷基氨基; n是1至4的整数; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 它们的制备方法，含有它们的组合物以及它们用于防治植物病原性真菌的用途。