公开(公告)号：WO0125187A3

公开(公告)日：2001-11-01

申请号：PCT/EP0009744

申请日：2000-10-05

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

Inventor： RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A61P31/10 ,  A01N37/52 ,  A61K31/165 ,  C07C259/14 ,  A01N43/10 ,  A01N43/40 ,  C07D213/54 ,  C07D333/24

CPC classification number: C07C259/14 ,  A01N37/52 ,  C07C2601/02

Abstract: The invention relates to benzyl amidoxime derivatives of formula (I) as fungicides wherein: A represents an aryl or heteraryl radical; Y represents a straight-chained or branched C1-C4 alkylene group, whereby a carbon atom can be substituted by an oxygen, nitrogen or sulphur atom or by a cyclopropyl group; Rn represents one to five similar or different radicals from the group consisting of hydrogen, halogen, C1-C6 alkyl, C1-C6 alkoxy, C1-C4 halogen alkyl, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 alkoxyalkoxy; R represents optionally substituted phenyl C1-C6 alkyl, thienyl C1-C4 alkyl, or pyrazolyl C1-C4 alkyl, Rp represents one to five similar or different radicals from the group consisting of hydrogen, halogen, C1-C6 alkyl, C1-C6 alkoxy, C1-C4 halogen alkyl, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 alkoxyalkoxy, C1-C6 alkyl carbonyl; n represents 0-5; and p represents 0-4, according to the number of free valences.

Abstract translation: 本申请涉及式（I）作为杀真菌剂的Benzylamidoxim衍生物。 其中A为芳基或杂芳基; Y线性或支链的C1-C4亚烷基，其中一个碳原子可以被氧，氮或硫原子或由环丙基取代; RN <1>一至选自五个相同或不同的基团：氢，卤素，C1-C6烷基，C1-C6-烷氧基，C1-C4卤代烷基，C1-C4卤代烷氧基，C1-C4烷硫基，C1 -C4烷氧烷; [R <2>任选取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 4 - 烷基，或吡唑基-C 1 -C 4 - 烷基，卢比<3>一个从组五个相同或不同的基团：氢，卤素 ，C1-C6烷基，C1-C6-烷氧基，C1-C4卤代烷基，C1-C4卤代烷氧基，C1-C4烷硫基，C1-C4烷氧基烷氧基，C1-C6烷基羰基; n为0-5; p取决于自由价的0-4的数量。

公开(公告)号：WO2007113322A2

公开(公告)日：2007-10-11

申请号：PCT/EP2007053332

申请日：2007-04-04

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

CPC classification number: C07D401/04 ,  A01N43/54

Abstract: The invention relates to 5-hetaryl-4-pyrimidines of formula (I) and to their salts and plant protection agents which contain at least one compound of said type as an active component, wherein W represents oxygen, sulphur, a group S=O or S(=O) 2 ; R 1 represents optionally substituted C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl, or a C-bound five- or six-membered saturated, partially unsaturated or aromatic heterocycle containing one, two, three or four heteroatoms from the groups O, N or S as ring members; R 2 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 C 6 -halogenalkyl, C 1 C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 C 6 -halogenalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -halogenalkylthio, or a radical of formulae C(=Z)OR 21 , C(=Z)NR 22 R 23 , C(=Z)NR 24 -NR 22 R 23 , C(=Z)R 25 , CR 26 R 27 -OR 28 , CR 26 R 27 -NR 22 R 23 , ON(=CR 29 R 30 ), O-C(=Z)R 25 , NR 22 R 23a , NR 31 (C(=Z)R 25 ), NR 31 (C(=Z)OR 21 ), NR 31 (C(=Z)-NR 22 R 23 ), NR 32a (N=CR 29 R 30 ), NR 32 NR 22 R 23 , NR 32 OR 21 , or C(=N-Z'-R 25 )SR 21 ; or a cyclic radical; R3 represents hydrogen, OH, halogen, cyano, NR 37 R 38 , C 1 -C--alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulfinyl, C 1 -C--alkylsulfonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkinyl, whereby the seven latter radicals can be partially or totally halogenated and/or optionally can support one, two or three substitutes, selected among nitro, cyano, OH, C 1 -C 2 -alkoxy, C 1 -C 4 -alkoxycarbonyl, amino, C 1 -C 4 -alkylamino and Di-C 1 -C 4 -alkylamino, Het represents a substituted C- or N-bound, 5-or 6-membered aromatic heterocycle which comprises 1, 2, 3 or 4 heteroatoms as ring members selected among nitrogen, oxygen and sulphur. The invention also relates to the use of 5-hetaryl-4-pyrimidines of formula (I) and there salts for combating plant pathogenic fungi.

Abstract translation: 本发明涉及式（I）的包含至少一种这样的化合物作为有效成分的5-杂芳基-4-嘧啶和它们的盐和杀虫剂。 其中W = O或S（= O） _{2 表示氧，硫，基团S; [R ^{1 表示任选subsitituiert.esç 1 -C 8 烷基，C 3 -C 8 环烷基，C 5 -C 10 双环，C 2 -C 8 - 烯基，C 4 -C 10 链二烯基，C 3 -C 6 环烯基，C 2 -C 8 是炔基，苯基，萘基或C-连接的五元或六元饱和，部分不饱和或芳族的含有一个，两个，三个或四个杂原子的从杂环 包含基团的O，N或S作为环成员; [R 2 表示卤素，氰基，羟基，巯基，N 3 ，C 1 -C 6 烷基， ç 2 -C 8 烯基，C 2 -C 8 - 炔基，C 1 < / SUB> C 6 卤代烷基，C 1 C 6 烷氧基，C 3 -C 8 烯，C 3 -C 8 炔氧基，C 1 C 6 卤代烷氧基 ，C 1 -C 6 烷硫基，C 3 -C 8 烯，C 3 -C 8 炔硫基，C 1 -C 6 卤代烷硫基，或一个基团，式C（= Z） OR 21 ，C（= Z）NR 22 - [R 23 ，C（= Z）NR 24 -NR 22 - [R 23 ，C（= Z）R 25 ，CR 26 - [R 27 -OR 28 ，CR 26 - [R 27 -NR 22 - [R 23 ， ON（= CR 29 - [R 30 ），OC（= Z）R 25 ，NR 22 - [R 图23A ，NR 31 （C（= Z）R 25 ），NR 31 （C（= Z）OR < SUP> 21 ）NR 31 （ C（= Z）-NR 22 - [R 23 ），NR 32A （N = CR 29 - [R 30 ），NR 32 NR 22 - [R 23 ，NR 32 OR 21 ，或C（= N-Z'-R 25 ）SR 21 ; 或环状基团; R 3是氢，OH，卤素，氰基，NR 37 - [R 38 ，C 1 -C - 烷基，C 1 -C 8 烷氧基，C 1 -C 8 烷硫基，C 1 -C 8 烷基亚磺酰基，C 1 -C - 烷基磺酰基，C 2 -C 8 链烯基或C 2 -C 8 炔基，其中所述7最后提到的基团可以部分或完全卤化和/或选自硝基一个，两个或三个取代基，氰基，OH，C 1 -C 2 烷氧基，C 1 -C 4 烷氧基羰基，氨基，C 1 -C 4 烷基氨基和二C 1 -C 4可携带>烷基氨基，}}

公开(公告)号：WO2005087770A3

公开(公告)日：2005-12-08

申请号：PCT/EP2005002424

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 5,6-二烷基 - 7-氨基三唑并嘧啶，其中取代基具有式（I）的以下含义：R t <1>是烷基，烷氧基烷基，烯基或炔基; [R <2>是烷基，烷氧基烷基，烯基或炔基; 其中R <1>和/或R <2>取代根据描述; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。

公开(公告)号：WO2004041824A2

公开(公告)日：2004-05-21

申请号：PCT/EP0312276

申请日：2003-11-04

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 取代的式（I）的6-（2-卤代苯基） - 三唑并嘧啶，其中R1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或 芳族杂环，其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义地被取代，R 2表示氢，或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或N（R b）2，其中R b如说明书中所定义，其中至少一个L 1，L 2， 而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基，它们的制备方法，含有它们的组合物和它们用于防治植物病原性真菌的用途。

公开(公告)号：WO0162087A3

公开(公告)日：2002-02-14

申请号：PCT/EP0102059

申请日：2001-02-23

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

Inventor： RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  A01N43/36 ,  C07D207/50

CPC classification number: C07D207/50 ,  A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  A01N43/36

Abstract: The invention relates to agrochemical compositions with a fungicidal action, containing compounds of formula (I) as their active agents. The radicals of said formula have the following meanings: R means hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-halogenalkylcarbonyl; R means halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halogen-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halogen-C1-C6-alkylsulfonyl, cyano or a radical NR R ; R -R mean hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, halogen-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halogen-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which can optionally be substituted by halogen atoms, C1-C6-alkyl or halogen-C1-C6-alkyl groups; R means hydrogen, C1-C6-alkyl; and R means C1-C6-alkyl, C1-C8-cycloalkyl or together with R and the nitrogen atom to which they are bonded, a saturated or unsaturated heterocyclic five or six-membered ring which has one or two heteroatoms selected from a group consisting of nitrogen atoms and oxygen atoms. The invention also relates to salts of said compositions which are suitable for agricultural use.

Abstract translation: 本发明的目的是具有包含（I），其中各基团具有以下含义的式作为活性成分的化合物的杀真菌作用的农药组合物，R <1>是氢，C1-C6烷基，C1-C6烷基羰基，甲酰基或C1-C6 卤代; [R <2>为卤素，C1-C6-烷硫基，C1-C6烷氧基，C3-C6环烷基-C1-C6-烷氧基，C1-C6烷氧基C1-C6烷基，卤代C1-C6烷氧基， C1-C6烷基磺酰基，C1-C6-烷基亚磺酰基，卤代C1-C6烷基磺酰基，氰基或基团NR <13> - [R <14>; [R <3> -R <12>为氢，卤素，C1-C8环烷基，C1-C6-烷基，卤代C1-C6烷基，C1-C6-烷氧基，卤代C1-C6烷氧基，C1-C6 烷基磺酰基，卤代C1-C6烷基磺酰基，甲酰基，C1-C6烷基羰基，氰基，C1-C6烷硫基或苯基，其是任选地被卤素原子，C1-C6烷基或烷基 - 卤素-C 1 -C 6 - 取代的 基团可被取代，R <13>为氢，C1-C6烷基，R <14> C1-C6-烷基，C1-C8环烷基，或一起为R <13>和的氮原子它们所连接形成其 意味着饱和或ungesätttigten杂环五元或含有从包含氮原子或氧原子，和它们的可农用可用的盐的组中选择的一个或两个杂原子的六元环。

公开(公告)号：WO0012465A3

公开(公告)日：2000-06-22

申请号：PCT/EP9906251

申请日：1999-08-26

Applicant: BASF AG ,  ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

Inventor： ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

IPC: C07C233/61 ,  A01N25/02 ,  A01N25/08 ,  A01N37/18 ,  A01N53/00 ,  A01N53/12 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24

CPC classification number: A01N53/00 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24 ,  C07C2601/02

Abstract: The invention relates to novel cycloalkylalkane carboxylic acid amides of the general formula (I), as well as salts thereof which are suitable for use in agriculture, in which the substituents have the following meanings: A is C3-C6 cycloalkyl which can carry one or more substituents; Alk is straight-chain or branched C1-C6-alkylene; R is C1-C6-alkyl or C2-C6-alkenyl, which can carry one or more substituents; R , R are hydrogen, C1-C6-alkyl or C2-C6-alkenyl, which rests can be partly or fully halogenated; and W is a fused bicyclic ring system with six ring atoms each. The invention also relates to fungicidal agents containing a compound of formula (I) as plant protectant.

Abstract translation: 本发明涉及新的cycloalkylalkanecarboxamides通式（I），其中取代基具有以下含义：A，C 3 -C 6环烷基，其可带有一个或多个取代基; ALK的直链或支链C1-C6亚烷基; [R <1>，C1-C6烷基或C2-C6链烯基，其可以带有一个或nehrere取代基; [R <2>，R <3>为氢，C1-C6烷基或C2-C6链烯基，其中这些基团可以部分或完全被卤代; 具有六个环原子W，稠合的双环环系; 及其可农用可用的盐。 此外，本发明涉及包含式（I）的化合物用作植物保护剂的杀真菌组合物。

公开(公告)号：WO2006097489A8

公开(公告)日：2007-03-08

申请号：PCT/EP2006060753

申请日：2006-03-15

Applicant: BASF AG ,  GRAMMENOS WASSILIOS ,  RHEINHEIMER JOACHIM ,  LOHMANN JAN KLAAS ,  GROTE THOMAS ,  PUHL MICHAEL ,  KORADIN CHRISTOPHER ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  LANGEWALD JUERGEN ,  GOETZ NORBERT ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS D ,  OLOUMI-SADEGHI HASSAN ,  COTTER HENRY VAN TUYL ,  KUHN DAVID G

Inventor： GRAMMENOS WASSILIOS ,  RHEINHEIMER JOACHIM ,  LOHMANN JAN KLAAS ,  GROTE THOMAS ,  PUHL MICHAEL ,  KORADIN CHRISTOPHER ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  LANGEWALD JUERGEN ,  GOETZ NORBERT ,  CULBERTSON DEBORAH L ,  ANSPAUGH DOUGLAS D ,  OLOUMI-SADEGHI HASSAN ,  COTTER HENRY VAN TUYL ,  KUHN DAVID G

IPC: A01N43/40 ,  C07D213/42

CPC classification number: A01N43/40 ,  C07D213/42

Abstract: Biphenylsulfonamides of the formula (I) and the N-oxides and the agriculturally acceptable salts and the veterinarily acceptable salts of the compounds I, a process for preparing these compounds, compositions comprising them, their use for controlling phytopathogenic harmful fungi and harmful arthropodes, a method for combating arthropodal pests, a method for protecting crops from attack or infestation of arthropodal pests, a method for protecting seed and non-living materials from infestation by arthropodal pests, a method for protecting non-living materials from attack or infestation by arthropodal pests and seed comprising the compounds I.

Abstract translation: 式（I）的联苯磺酰胺和化合物I的N-氧化物和农业上可接受的盐和兽医学上可接受的盐，制备这些化合物的方法，包含它们的组合物，其用于控制​​植物病原性有害真菌和有害的节肢动物的用途 防治节肢动物害虫的方法，保护作物免受节肢动物害虫侵袭或侵扰的方法，保护种子和非生物材料免受节肢动物害虫侵扰的方法，保护非生物材料免受节肢动物害虫侵袭或侵袭的方法 和包含化合物I的种子。

公开(公告)号：WO2006092428A2

公开(公告)日：2006-09-08

申请号：PCT/EP2006060399

申请日：2006-03-02

Applicant: BASF AG ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  RACK MICHAEL

Inventor： GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  RACK MICHAEL

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.

Abstract translation: 2-取代的式（I）其中取代基具有以下含义的7-氨基azolopyrimidines：R t ^{1 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基， benzyloxyalkyl，烷氧基烯基或alkoxyalkynyl; [R 2 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基和烷硫基烷基，其中在R中的碳链 1 和/或R 2 可以根据描述被取代; [R 3 为卤素，氰基，NR 一 - [R 乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基， 羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯丙氨酸nylthio，苄氧基，苄硫基，烷基-S（O）_{米 - ; A N和CR X ; ，R 3 基 X 是氢或其中R 称作; 的方法和中间体制备这些化合物，含有它们和它们在防治植物病原性有害真菌的组合物。}}

公开(公告)号：WO2005095404A3

公开(公告)日：2006-04-06

申请号：PCT/EP2005003208

申请日：2005-03-26

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to the 6-(2-fluorophenyl)-triazolopyrimidines of formula (I), wherein the substituents are defined as follows: R

Abstract translation: 本申请公开了式-6-（2-氟苯基） - 三唑并嘧啶予其中的取代基具有下列含义：R t

公开(公告)号：WO2005095405A3

公开(公告)日：2005-12-22

申请号：PCT/EP2005004187

申请日：2005-03-29

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 6-(2,6-dichlorophenyl)-triazolopyrimidines of formula (I) wherein the substituents have the following designations: R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, halogencycloalkenyl, alkinyl, halogenalkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group containing O, N or S; R and R can also form, together with the nitrogen atom to which they are bound, a five-membered or six-membered heterocycle or heteroaryl which is bound by N and contains between one and three other heteroatoms from the group containing O, N and S as a cyclic member and is substituted according to the description; and X represents alkyl, cyano, alkoxy, halogenalkoxy, alkenyloxy or halogenalkenyloxy, but does not represent C1-C4 alkyl when R and R together represent piperidin-1-yl or 4-methylpiperidin-1-yl. The invention also relates to a method for producing said compounds, agents containing the same, and the use thereof for controlling plant pathogenic fungi.

Abstract translation: 6-（2,6-二氯苯基） - 三唑并嘧啶的式（I）的其中取代基具有以下含义：R t <1>，R <2>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基 基，炔基，卤代炔基，或苯基，萘基，或含有选自O，N，或S，R <1>和R <2>也可以，一起一至四个杂原子的五元或六元饱和，部分不饱和或芳族杂环 形成一个五元或六元杂环基或杂芳基的氮原子与它们所连接，这是经N个附接和选自O，N和S的一至三个另外的杂原子作为环成员，并且可以根据该描述被取代; X为烷基，氰基，烷氧基，卤代烷氧基，烯氧基或卤代链烯氧基，其中X不为C1-C4烷基，当R <1>和R <2>是常见的哌啶-1-基或4-甲基 - 哌啶-1-基; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。