公开(公告)号：EP1218350A1

公开(公告)日：2002-07-03

申请号：EP00967704.8

申请日：2000-09-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MENKE, Olaf ,  REINHARD, Robert ,  HAMPRECHT, Gerhard ,  PUHL, Michael ,  SAGASSER, Ingo ,  ZAGAR, Cyrill ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D233/86 ,  C07D233/70 ,  A01N43/50

CPC classification number: C07D401/04 ,  A01N43/50 ,  C07D233/70 ,  C07D233/86 ,  C07D413/04

Abstract: The invention relates to novel substituted 1-aryl-1,3-dihydro-imidazol-2-(thi)one of formula (I) and the salts of said compound whereby R1=NH2, C1-C6-alkyl, C1-C6-halogenalkyl; R2=OH, SH, C¿1?-C6-alkoxy, C1-C4-halogenalkoxy, C1-C6-alkylthio, C1-C4-halogenalkylthio, C1-C6-alkylsulfinyl, C1-C4-halogenalkylsulfonyl, C1-C4-halogenalkyl or C1-C6-alkyl; R?3¿=H, halogen, C¿1?-C6-alkyl, halogenmethyl; R?4¿=H, halogen; R5=CN, halogen, -CO-NH¿2?, -CS-NH2, -OC(R?8,R9¿)-CO-O(C¿1?-C6-alkyl); Y=N, CH or in conjunction with R?6¿ a bridge ⊃C-O-C(R10)=N-, ⊃C-S-C(R10)=N- or ⊃C-N=C(R?10)-O-; R6+R5¿= or a N(R7)-C(O/S)-C(R8',R9')-O- radical, bonded at the oxygen moiety to R5 or 1) OH, SH, CN, NO¿2?, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C1-C6-halogenalkylthio, C1-C6-alkylthio-(C1-C6-alkyl)carbonyl, (C1-C6-alkyl)iminooxycarbonyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-alkoxyamino-C1-C6-alkyl, C1-C6-alkoxy-C1-C6-alkoxyamino-C1-C6-alkyl, 2) optionally substit. C1-C6-alkoxy, C1-C6-alkylthio, C3-C6-cycloalkoxy, C3-C6-cycloalkylthio, C2-C6-alkenyloxy, C2-C6-alkenylthio, C2-C6-alkinyloxy, C2-C6-alkinylthio, (C1-C6-alkyl)carbonyloxy, (C1-C6-alkyl)carbonylthio, (C1-C6-alkoxy)carbonyloxy, (C2-C6-alkenyl)carbonyloxy, (C2-C6-alkenyl)carbonylthio, (C2-C6-alkinyl)carbonyloxy, (C2-C6-alkinyl)carbonylthio, C1-C6-alkylsulfonyloxy or C1-C6-alkylsulfonyl, 3) 28 other radicals; R?7¿=H, optionally subst. C¿1?-C6-alkyl, C3-C6-alkenyl, C3-C6-alkinyl, C1-C6-alkoxy, C3-C6-alkenyloxy, C3-C6-alkinyloxy, C3-C6-cycloalkyl or C3-C6-cycloalkyloxy; R?8, R9, R8', R9'¿ = H, CN, C¿1?-C6-alkyl; R?10¿=H, halogen, optionally subst. C¿1?-C6-alkyl, C3-C6-alkenyl, C3-C6-alkinyl, C1-C6-alkoxy, C3-C6-alkenyloxy, C3-C6-alkinyloxy, C3-C6-cycloalkyl or C3-C6-cycloalkyloxy. Use: as a herbicide or as a dessicating/defoliating agent for plants.

公开(公告)号：EP1200428A1

公开(公告)日：2002-05-02

申请号：EP00958421.0

申请日：2000-08-10

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： REINHARD, Robert ,  HAMPRECHT, Gerhard ,  MENKE, Olaf ,  PUHL, Michael ,  SAGASSER, Ingo ,  ZAGAR, Cyrill ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D413/04 ,  C07D263/56 ,  A01N43/653 ,  A01N43/836 ,  A01N43/76

CPC classification number: C07D263/56 ,  A01N43/76 ,  C07D413/04

Abstract: The present invention relates to substituted benzoxazoles of general formula (I) wherein R?1, R2 and R3¿ have the meanings cited in claim 1, and Het stands for a 5- or 6-membered heterocycle bonded by nitrogen and having general formulae (II-1) to (II-18). The invention also relates to agents containing such compounds as well as to a method for combating undesired plant growth; the compounds of general formulae (III), (IV) and (V) are used as intermediate products for the production of the formula (I) compoun ds.

公开(公告)号：EP0958276B1

公开(公告)日：2002-03-13

申请号：EP97953895.6

申请日：1997-12-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HILL, Regina, Luise ,  KARDORFF, Uwe ,  RACK, Michael ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  MAYER, Guido ,  OTTEN, Martina ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07C251/60 ,  C07C251/86 ,  A01N33/24 ,  A01N33/26

CPC classification number: A01N41/10 ,  A01N35/10 ,  A01N37/52 ,  C07C251/48 ,  C07C259/10 ,  C07C317/32 ,  C07C317/44 ,  C07C2601/16

Abstract: The invention concerns 2-benzoyl-cyclohexan-1,3-diones of formula (I), in which R , R stand for hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkyl, alkoxyalkyl, alkenyl, alkinyl, -OR , -OCOR , -OSO2R , -SH, -S(O)nR , -SO2OR , -SO2NR R , -NR SO2R or -NR COR ; R stands for hydrogen, cyano, alkyl, halogen alkyl, -OR , -SR or -NR R ; R stands for hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkinyl, -COR , -CO2R , -COSR or -CONR R ; X stands for oxygen or NR ; n equals 0, 1 or 2; R stands for hydrogen, alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R stands for alkyl or halogen alkyl; R stands for alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R stands for hydrogen or alkyl; R stands for alkyl, alkenyl, alkinyl, phenyl or benzyl; R stands for alkyl, halogen alkyl, alkenyl or alkinyl; Q stands for an optionally substituted cyclohexan-1,3-dione ring linked in position 2. Also disclosed are the salts of these compounds useful in agriculture; processes and intermediate products for preparing the compounds of formula (I), agents containing the same and the use of these derivatives or agents containing the same for controlling undesirable plants.

公开(公告)号：EP0695296B1

公开(公告)日：2002-03-06

申请号：EP94914369.7

申请日：1994-04-14

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAUMANN, Ernst ,  RHEINHEIMER, Joachim ,  VOGELBACHER, Uwe, Josef ,  BRATZ, Matthias ,  MEYER, Norbert ,  GERBER, Matthias ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  RADEMACHER, Wilhelm

IPC: C07D239/60 ,  C07D239/52 ,  C07D333/24 ,  C07D307/46 ,  C07C69/22 ,  A01N43/54 ,  C07D405/12 ,  C07D409/12

CPC classification number: C07C69/734 ,  A01N43/54 ,  C07C69/712 ,  C07D239/60 ,  C07D251/30

Abstract: The invention concerns 3-(hetero)aryloxy(thio) carboxylic acid derivatives of the formula (I) in which the substituents are defined as follows: R1 is hydrogen, a COOH group or a group which can be hydrolysed to give a COOH group; R?2 and R3¿ are halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; X is nitrogen or CR14, R14 being hydrogen or, together with R3, a 3-membered or 4-membered alkylene or a alkenylene chain in which each methylene group can be replaced by oxygen; R4 is optionally substituted alkyl, cycloalkyl, cycloalkenyl, alkenyl or alkinyl, an optionally substituted five-membered or six-membered heteroaromatic ring containing one to three nitrogen atoms and/or a sulphur or oxygen atom, or optionally substituted phenyl or naphthyl; R?4 and R5¿ together form, together with the neighbouring carbon atom, a 3-membered to 8-membered ring which may contain an oxygen or sulphur atom and may also be substituted; R5 is hydrogen or optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl or phenyl; R6 is optionally substituted phenyl or naphthyl or an optionally substituted five-membered or six-membered heteroaromatic ring containng one to three nitrogen atoms and/or a sulphur or oxygen atom; Y is sulphur or oxygen or a single bond; Z is sulphur or oxygen.

公开(公告)号：EP1163232A1

公开(公告)日：2001-12-19

申请号：EP00906364.5

申请日：2000-02-21

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WITSCHEL, Matthias ,  GÖTZ, Roland ,  RACK, Michael ,  PLATH, Peter ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D275/06 ,  A01N43/80

CPC classification number: C07D275/06 ,  A01N43/80

Abstract: The invention relates to saccharin 5 carbonyl derivatives of formula (I), wherein the substituents have the following meaning: L represents C1-C6-alkyl, C1-C6-alkoxy; Z represents C1-C6-alkyl, C3-C8-cycloalkyl, C3-C6-alkenyl, C3-C5-alkinyl, phenyl-C1-C6-alkyl or phenyl, wherein the phenyl rings are optionally substituted once or several times by C1-C6-alkyl, C1-C6-alkoxy or halogen; M represents hydrogen, C1-C6-alkyl, C1-C6-alkoxy, halogen, cyano, nitro or halogen-C1-C6-alkyl; R?1, R2, R3, R4, R5, R6, R7, R8¿ represent hydrogen, C¿1?-C6-alkyl. The invention also relates to the agriculturally usable salts of compound (I).

公开(公告)号：EP0961774B1

公开(公告)日：2001-12-12

申请号：EP96930126.6

申请日：1996-08-29

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OTTEN, Martina ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  VOSSEN, Marcus ,  PLATH, Peter ,  GÖTZ, Norbert ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D409/06 ,  A01N43/56 ,  C07D411/06 ,  C07D417/06

CPC classification number: C07D335/06 ,  A01N43/56 ,  C07D333/64 ,  C07D409/06 ,  C07D417/06

Abstract: The invention concerns pyrazol-4-yl-benzoyl derivatives of formula (I) in which the substituents L, M, X, Y, and n have the meanings given in claim 1, and Q is a pyrazol ring which is bonded in position 4 and corresponds to formula (II), in which: R15 designates a C¿1? - C4 alkyl; R?16¿ designates hydrogen, C¿1? - C4 alkyl or C1 - C4 alkyl halide; and R?17¿ designates hydrogen, C¿1? - C4 alkylsulphonyl, phenylsulphonyl or alkylphenylsulphonyl; wherein if Y = C=O, X is not NR?23¿. The invention further concerns salts for agricultural purposes, a process for their preparation and their use as herbicides.

公开(公告)号：EP0759907B1

公开(公告)日：2001-10-10

申请号：EP95920017.1

申请日：1995-05-10

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEM BUSSCHE-HÜNNEFELD, Christoph-Sweder ,  KLINTZ, Ralf ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  SCHÄFER, Peter ,  MÜNSTER, Peter ,  DITRICH, Klaus ,  KÖNIG, Hartmann ,  WESTPHALEN, Karl-Otto ,  GERBER, Matthias ,  WALTER, Helmut

IPC: C07D231/20 ,  A01N43/50 ,  C07D401/12 ,  C07D403/12 ,  C07D405/10 ,  C07D405/12 ,  C07D409/10 ,  C07D413/12

CPC classification number: A01N53/00 ,  A01N43/56 ,  C07D231/18 ,  C07D231/20 ,  C07F9/65033

Abstract: Substituted 3-phenylpyrazoles of formula (I), where R1 is H, or a substituent; R2 is CN, CF¿3?, halogen; R?3¿ is H, alkyl, halogenalkyl; R4 is C1-C4 alkyl, C1-C4 halogenalkyl; R5 is H, NO¿2?, halogen, -COOR, optionally substituted aminocarbonyl (where R is H, a substituent); and Z is -O-, -S-, -SO-, -SO2-; and agriculturally usable salts thereof, for use as herbicides.

公开(公告)号：EP1135386A1

公开(公告)日：2001-09-26

申请号：EP99966912.0

申请日：1999-12-02

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： NEIDLEIN, Ulf ,  GÖTZ, Norbert ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MAYER, Guido ,  WITSCHEL, Matthias ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D409/06 ,  C07D401/06 ,  C07D417/06 ,  A01N43/56

CPC classification number: C07D409/06 ,  C07D409/14

Abstract: The invention relates to a method for producing pyrazolylbenzoyl derivatives of formula (I), wherein the substituents have the following meanings: R1 represents hydrogen, C¿1?-C4-alkyl or C1-C4 alkyl halide; R?2¿ represents hydrogen, C¿1?-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, benzyl, benzoyl, C1-C4-alkylcarbonyl, hydroxycarbonyl-C1-C4-alkyl, C1-C4-alkoxycarbonyl-C1-C4-alkyl, C1-C4-alkylsulfonyl or phenylsulfonyl, and these groups can be substituted by C1-C4-alkyl, C1-C4-alkoxy, C1-C4-alkylthio, halogen, hydroxy, amino, nitro or cyano; A,B represent, independently of each other, hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C1-C4-alkoxy and these groups can be substituted by halogen, hydroxy, C1-C4-alkoxy or cyano, halogen, hydroxy, cyano; nitro, a group-(Y)n-S(O)mR?3¿ or a group-(Y)¿n-CO-R?4; Z represents a 5- or 6-membered heterocyclic, saturated or unsaturated fused ring; Y represents O, NR5; n represents zero or one; m represents zero, one or two; R3 represents C¿1?-C4-alkyl, C1-C4-alkyl halide or NR?5R6; R4¿ represents C¿1?-C4-alkyl, C1-C4-alkyl halide, C1-C4-alkoxy, or NR?5R6; R5¿ represents hydrogen or C¿1?-C4-alkyl; and R?6¿ represents C¿1?-C4-alkyl. The invention also relates to novel pyrazolylbenzoyl derivatives, to herbicidal agents containing these derivatives and to a method for combating unwanted vegetation.

公开(公告)号：EP1135385A1

公开(公告)日：2001-09-26

申请号：EP99962201.2

申请日：1999-12-02

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： LANGEMANN, Klaus ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  MAYER, Guido ,  MISSLITZ, Ulf ,  NEIDLEIN, Ulf ,  WITSCHEL, Matthias ,  GÖTZ, Norbert ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D409/06 ,  C07D409/14 ,  A01N43/56

CPC classification number: C07D409/06 ,  C07D409/14

Abstract: The invention relates to thiochromanoylpyrazolone derivatives of formula (I), wherein the variables have the following meanings: A is an optionally substituted, saturated or unsaturated alkyl chain; R1 is cyano, rhodano, nitro, OR?4, SR5, SOR6, SO¿2R?6, ONR6NR7, ON=CR6R8, NR9R10, P(O)R11R12, P(S)R11R12, COR6, CO¿2R6, optionally substituted phenyl or heterocyclyl; R2 is alkyl, alkyl halide, alkoxy or halogenalkoxy; R3 is hydrogen, alkyl or halogen; X is oxygen, sulphur, S=O, S(=O)¿2?, CR?13R14¿, C=O or C=NR15, m is 0, 1 or 2; n is 0, 1, 2, 3 or 4; and R16 is substituted pyrazol-4-yl-carbonyl or substituted (4,5-dihydro-5-oxo-pyrazol-4-yl)-methylidene; and to their agriculturally useable salts. The invention also relates to a method for producing thiochromanoylpyrazolone derivatives, to products containing them and to the use of these derivatives and products containing them for combating undesirable plants.

Abstract translation: 本发明涉及式（I）的二氢苯并噻喃酰基吡唑啉酮衍生物，其中各变量具有以下含义：A为任选取代的饱和或不饱和的烷基链; R1是氰基，氰基，硝基，OR4，SR5，SOR6，SO2R6，ONR6NR7，ON = CR6R8，NR9R10，P（O）R11R12，P（S）R11R12，COR6，CO2R6， 苯基或杂环基; R2是烷基，烷基卤，烷氧基或卤代烷氧基; R3是氢，烷基或卤素; X是氧，硫，S = O，S（= O）2 2，CR 13 R 14，C = O或C = NR 15，m是0,1或2; n是0,1,2,3或4; 和R 16是取代的吡唑-4-基 - 羰基或取代的（4,5-二氢-5-氧代 - 吡唑-4-基） - 亚甲基; 和它们的农用盐。 本发明还涉及一种生产二氢苯并噻喃酰基吡唑啉酮衍生物的方法，含有它们的产品以及这些衍生物和含有它们的产品用于防治不希望的植物的用途。

公开(公告)号：EP0836594B1

公开(公告)日：2001-03-07

申请号：EP96922038.3

申请日：1996-06-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： KLINTZ, Ralf ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  SCHÄFER, Peter ,  ZAGAR, Cyrill ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  MISSLITZ, Ulf ,  MENKE, Olaf ,  MENGES, Markus

IPC: C07D239/54 ,  C07C265/12 ,  C07C239/20 ,  A01N43/54

CPC classification number: C07D239/54 ,  A01N43/54 ,  A01N47/12 ,  A01N47/24 ,  A01N47/30 ,  A01N53/00 ,  C07C239/08 ,  C07C239/10 ,  C07C265/12 ,  C07C271/22 ,  C07C271/28 ,  C07C271/54 ,  C07C271/58 ,  C07C275/40

Abstract: The invention pertains to benzylhydroxylamines of formula (I), wherein X is -N(R7)-O-; Y is O, S; R1 is halogen, CN, NO¿2?, CF3; R?2¿ is H, halogen; R3 is H, NH¿2?, CH3; R?4¿ is H, halogen, C¿1?-C6 alkyl, C1-C6 alkyl halide, C1-C6 alkyl thio, C1-C6 alkyl sulfinyl or C1-C6 alkyl sulfonyl; R?5¿ is H, halogen, C¿1?-C6 alkyl; R?6¿ is H, C¿1?-C6 alkyl, C1-C6 alkyl halide, C3-C6 cycloalkyl, C2-C6 alkenyl; R?8¿ is H, C¿1?-C6 alkyl, C3-C8 cycloalkyl, C1-C6 alkyl halide, C3-C6 alkenyl or C3-C6 alkinyl, where each of the last five radicals indicated can carry 1-3 substituents. The invention also pertains to the salts of (I), with R?3, R7¿ and/or R8 being hydrogen. These compounds are useful as herbicides and for desiccation/defoliation of plants.