USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME
    21.
    发明申请
    USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME 审中-公开
    使用5-烷基-6-苯基 - 7-氨基AZOLOPYRIMIDINEN,NEW azolopyrimidines,METHOD用于生产和AGENTS CONTAINING THE SAME

    公开(公告)号:WO2006114405A2

    公开(公告)日:2006-11-02

    申请号:PCT/EP2006061786

    申请日:2006-04-24

    CPC classification number: A01N43/90 C07D487/04

    Abstract: The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.

    Abstract translation: 式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I:其中各变量具有以下含义:Y是任选被烷基取代的亚烷基,亚烯基或亚炔基; [R 1 为卤素,氰基,硝基,羟基,巯基,烷基,卤代烷基,链烯基,环烷基,环烯基,烷氧基,卤代烷氧基,烯氧基,炔氧基,烷硫基,NR - [R < SUP>乙,烷基羰基,苯基,萘基或五 - 或六元饱和环,其包含选自一至四个杂原子的部分不饱和或罗马杂环O,N或S; [R ,R 是氢,烷基和烷基羰基; n是零,1,2,3或4; [R 2 烷基,烯基,环烷基,烷氧基烷基和烷硫基烷基; [R 3 为氢,卤素,氰基,NR - [R ,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基, 环烷硫基,羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O)米 - ; m是0,1或2; A N和C-R ; [R 氢和烷基; 其中Y中的碳原子,R 1 ,R 2 ,R 3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines,处理用于制备这些化合物和含有它们的组合物。

    USE OF SUBSTITUTED IMIDAZOAZINES, NOVEL IMIDAZOAZINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THESE COMPOUNDS
    26.
    发明申请
    USE OF SUBSTITUTED IMIDAZOAZINES, NOVEL IMIDAZOAZINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THESE COMPOUNDS 审中-公开
    USE取代IMIDAZOAZINEN,新imidazoazines,制造方法,和代理人含

    公开(公告)号:WO0248146A2

    公开(公告)日:2002-06-20

    申请号:PCT/EP0114577

    申请日:2001-12-12

    CPC classification number: C07D471/04 A01N43/90 C07D487/04

    Abstract: The invention relates to the use of substituted imidazoazines of formula (I), in which the variables have the following meanings: R represents alkyl, phenyl, phenylalkyl, naphthyl, anthracenyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, or condensed 8-membered to 12-membered hetaryl or condensed 8-membered to 12-membered heterocyclyl, containing one to four N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, whereby R can be unsubstituted or can be substituted as cited in the description; R and R represent hydrogen, alkyl, alkenyl, alkynyl, alkyl halide, alkenyl halide, alkynyl halide, trialkyl silylalkyl, phenyl, phenylalkyl or R and R , together with the bridging N atom, form a 5-membered or 6-membered heterocyclic or heteroaromatic ring, which can be interrupted by one to three N atoms and/or one O atom or S atom or by one or two O atoms and/or S atoms, and which can be substituted; A and B represent N or CR ; R , R and R represent hydrogen, halogen, cyano, nitro, hydroxy, alkyl, alkyl halide, cycloalkyl, alkoxy, alkoxy halide, alkylthio, amino, alkyl amino, dialkylamino, alkenyl, alkenyloxy, alkynyl or alkynyloxy. The inventive compounds are used for controlling phytopathogenic harmful fungi. The invention further relates to agents containing the inventive compounds, to novel imidazoazines, and to methods for the production thereof.

    Abstract translation: 使用式(I)的取代的Imidazoazinen的,其中各变量具有以下含义:R t <1>是烷基,苯基,苯基烷基,萘基,蒽基,环烷基,5-或6-员杂芳基或5-或6-元杂环基 含有1至3个N原子和/或一个O或S原子或一个或两个O和/或S原子,或稠合8-12 gliederiges杂芳基或稠合的8-12 gliederiges杂环基, 含有一至四个N原子和/或一个O或S原子或一个或两个O和/或O原子,其中R是未取代的<1>或作为可在本说明书中被取代; [R <2>,R <3>是氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代炔基,三烷基甲硅烷基,苯基,苯基烷基或R <2>,R <3>连同桥接氮原子的5-或6- 形成 - 元杂环基或可被一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子被中断杂芳族环; A,B,N或CR <4>; [R <4>,R <5> - [R <6>为氢,卤素,氰基,硝基,羟基,烷基,卤代烷基,环烷基,烷氧基,卤代烷氧基,烷硫基,氨基,烷基氨基,二烷基氨基,烯基,烯氧基,炔氧基或炔氧基; 防治植物病原性有害真菌的,含有它们,它们的制备新imidazoazines和方法的组合物。

    2-SUBSTITUTED 7-AMINO-AZOLOPYRIMIDINE, A METHOD FOR THE PRODUCTION AND USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUND
    29.
    发明申请
    2-SUBSTITUTED 7-AMINO-AZOLOPYRIMIDINE, A METHOD FOR THE PRODUCTION AND USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUND 审中-公开
    2-取代的7- aminoazolopyrimidines,METHOD用于生产和它们用于防治有害真菌和代理含

    公开(公告)号:WO2006092428A2

    公开(公告)日:2006-09-08

    申请号:PCT/EP2006060399

    申请日:2006-03-02

    CPC classification number: C07D487/04

    Abstract: The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.

    Abstract translation: 2-取代的式(I)其中取代基具有以下含义的7-氨基azolopyrimidines:R t 1 为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基, benzyloxyalkyl,烷氧基烯基或alkoxyalkynyl; [R 2 为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中在R中的碳链 1 和/或R 2 可以根据描述被取代; [R 3 为卤素,氰基,NR - [R ,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基, 羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯丙氨酸nylthio,苄氧基,苄硫基,烷基-S(O)米 - ; A N和CR X ; ,R 3 X 是氢或其中R 称作; 的方法和中间体制备这些化合物,含有它们和它们在防治植物病原性有害真菌的组合物。

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