公开(公告)号：WO0012465A3

公开(公告)日：2000-06-22

申请号：PCT/EP9906251

申请日：1999-08-26

Applicant: BASF AG ,  ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

Inventor： ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

IPC: C07C233/61 ,  A01N25/02 ,  A01N25/08 ,  A01N37/18 ,  A01N53/00 ,  A01N53/12 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24

CPC classification number: A01N53/00 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24 ,  C07C2601/02

Abstract: The invention relates to novel cycloalkylalkane carboxylic acid amides of the general formula (I), as well as salts thereof which are suitable for use in agriculture, in which the substituents have the following meanings: A is C3-C6 cycloalkyl which can carry one or more substituents; Alk is straight-chain or branched C1-C6-alkylene; R is C1-C6-alkyl or C2-C6-alkenyl, which can carry one or more substituents; R , R are hydrogen, C1-C6-alkyl or C2-C6-alkenyl, which rests can be partly or fully halogenated; and W is a fused bicyclic ring system with six ring atoms each. The invention also relates to fungicidal agents containing a compound of formula (I) as plant protectant.

Abstract translation: 本发明涉及新的cycloalkylalkanecarboxamides通式（I），其中取代基具有以下含义：A，C 3 -C 6环烷基，其可带有一个或多个取代基; ALK的直链或支链C1-C6亚烷基; [R <1>，C1-C6烷基或C2-C6链烯基，其可以带有一个或nehrere取代基; [R <2>，R <3>为氢，C1-C6烷基或C2-C6链烯基，其中这些基团可以部分或完全被卤代; 具有六个环原子W，稠合的双环环系; 及其可农用可用的盐。 此外，本发明涉及包含式（I）的化合物用作植物保护剂的杀真菌组合物。

公开(公告)号：WO0249438A3

公开(公告)日：2003-08-21

申请号：PCT/EP0114635

申请日：2001-12-13

Applicant: BASF AG ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  LEYENDECKER JOACHIM

Inventor： MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  LEYENDECKER JOACHIM

IPC: A01N43/653 ,  A01N43/50 ,  A01N43/56 ,  A01N43/80 ,  A01N47/24

CPC classification number: A01N47/24 ,  A01N43/90 ,  A01N43/50 ,  A01N2300/00

Abstract: The invention relates to a fungicidal mixture containing, A) carbamates of formula (I) wherein X, represents CH and N, n represents 0, 1 or 2 and R represents halogen, C1-C4-alkyl and C1-C4-halogenalkyl, wherein the radicals R can be different if n represents 2, a salt thereof or adduct, and B) imidazole derivatives of formula (II) wherein R and R represent halogen and phenyl which can be substituted by halogen or alkyl, or R and R together with the bridging C=C-double bond form a 3.4-difluoromethylene dioxy phenyl group; R represents cyano or halogen, and R represents dialkylamino or isoxazole-4-yl which can include two alkyl radicals in a synergistically active quantity. The invention also relates to a method for combating harmful fungi with mixtures of compounds I and II and the use thereof for producing said mixtures.

Abstract translation: 一种杀真菌混合物，包含：A）通式（I的氨基甲酸酯），其中X为CH和N，n是0，1或2，R是卤素，C1-C4烷基和C1-C4卤代烷基，其中所述基团 中，R是不同的，如果n为2，其盐或加合物的一个，和B）下式的咪唑衍生物（II），其中R <1>和R <2>是可被卤素或烷基取代的卤素和苯基， 或R <1>和R <2>与桥接C一起= C双键形成3,4- Difluormethylendioxyphenyl基; [R <4>二烷基氨基或异恶唑-4-基，其可带有两个烷基基团，意味着<3>是氰基或卤素，和R，以协同有效量，用于控制使用I和II和使用的化合物的混合物防治有害真菌的方法 化合物I和II在制备该类混合物。

公开(公告)号：WO0195721A3

公开(公告)日：2002-04-25

申请号：PCT/EP0106686

申请日：2001-06-13

Applicant: BASF AG ,  GRAMMENOS WASILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

Inventor： GRAMMENOS WASILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMAN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIGFRIED

IPC: A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22 ,  C07C233/69

CPC classification number: A01N37/36 ,  A01N37/18 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22

Abstract: The invention relates to the use of phenethyl acrylamides of formula (I) for controlling phytopathogenic fungi, wherein the substituents of said phenethyl acrylamides have the following significations: X signifies halogen, alkyl, halogenalkyl, alkoxy halogenalkoxy and -O-C(Ra, Rb)-C C-R?6; Ra, Rb and Rc¿ have the signification given in the description; m, n independently signify 1 to 4, the radicals X or Y being potentially different if m or n is higher than 1; Y signifies halogen, nitro, cyano, alkyl, CF¿3?, alkoxy and phenyl; R?1, R2¿ independently signify hydrogen, halogen, alkyl, alkoxy, halogenalkoxy and CF¿3?; R?3, R4, R5, and R6¿ independently signify hydrogen, alkyl and alkoxy, or R?3 and R4¿ together form a cyclopropyl ring, whereby the C-R5 and C-R6 bonds can be in position E or Z in relation to each other. The invention also relates to novel phenethyl acrylamides, a method for the production thereof, and agents containing the same.

公开(公告)号：WO9959982A3

公开(公告)日：2000-03-16

申请号：PCT/EP9903003

申请日：1999-05-04

Applicant: BASF AG ,  BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

Inventor： BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

IPC: C07C251/38 ,  A01N37/40 ,  C07C49/303 ,  C07C251/42 ,  C07C251/50 ,  C07C251/52 ,  C07C251/60 ,  A01N37/50 ,  C07C49/35

CPC classification number: C07C251/60 ,  C07C2601/14

Abstract: The invention relates to bisoximether derivatives of formula (I) in which the variables have the following meanings: R represents halogen, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or C1-C4 alkoxy halide; n is 1 to 5, whereby the radicals R can be different if n is not equal to 1; R represents C1-C4 alkyl, C3-C6 alkenyl or C3-C6 alkynyl, whereby these groups can be partially or completely halogenated; Q represents C(=CHOCH3)-COOCH3, C(=CHCH3)-COOCH3, C(=NOCH3)-COOCH3 or C(=NOCH3)-CONHCH3. The invention also relates to the salts of the bisoximether derivatives, to methods and intermediate products for the production of these compounds and to their use for combating animal pests and fungicidal pests.

Abstract translation: 式（I），其中各变量具有以下含义的双肟醚衍生物，R <1>为卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基; n为1至5，其中基团可以是与R <1>不同的，当n不为1; [R <2> C1-C4烷基，C3-C6链烯基或C3-C6炔基，其中这些基团可以部分或完全被卤代; Q为C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3）-COOCH 3或C（= NOCH 3）-CONHCH 3; 和它们的盐，方法和中间体制备这些化合物和它们用于控制动物害虫和有害真菌中的用途。

公开(公告)号：WO03073852A2

公开(公告)日：2003-09-12

申请号：PCT/EP0301929

申请日：2003-02-26

Applicant: BASF AG ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHELBERGER KLAUS ,  SPADAFORA V JAMES ,  CHRISTEN THOMAS

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHELBERGER KLAUS ,  SPADAFORA V JAMES ,  CHRISTEN THOMAS

IPC: A01N25/04 ,  A01N37/06 ,  A01N37/18 ,  A01N43/40 ,  A01N43/653 ,  A01N47/24 ,  A01N37/50

CPC classification number: A01N43/653 ,  A01N37/18 ,  A01N37/50 ,  A01N43/40 ,  A01N43/56 ,  A01N47/24 ,  C07D249/12 ,  A01N37/52 ,  A01N2300/00

Abstract: Disclosed is a fungicidal mixture containing (1) 2-[2-(1-chlorocyclopropyl)-3-(2-chlorophenyl)-2-hydroxypropyl]-2,4-dihydro-[1,2,4]-triazole-3-thion of formula (I) or the salts or adducts thereof, and at least one additional fungicidal compound or the salts or adducts thereof, selected among (2) trifloxystrobin of formula (II), (3) picoxystrobin of formula (III), (4) pyraclostrobin of formula (IV), (5) dimoxystrobin of formula (V), and (6) a strobilurin derivative of formula (VI), in a synergistically active quantity.

Abstract translation: 含有1 2- [2-1-氯环-3-2氯苯基-2-羟基丙基] -2,4-二氢 - [1,2,4]式三唑-3-硫酮的杀真菌混合物Ⅰ或它们的盐 或加合物，以及与至少一个另外的杀真菌化合物或它的盐或加合物，从2肟菌酯式II的，和式III的3啶氧菌酯，和4唑菌胺酯的式IV，和5醚菌胺式V的选择，6嗜球果伞素 衍生物的式VI，协同有效量的。

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO02054870A2

公开(公告)日：2002-07-18

申请号：PCT/EP0200237

申请日：2002-01-12

Applicant: BASF AG ,  GROTE THOMAS ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HADEN EGON

Inventor： GROTE THOMAS ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HADEN EGON

IPC: A01N37/50 ,  A01N43/40 ,  A01N43/50 ,  A01N43/80 ,  A01N43/90

CPC classification number: A01N43/50 ,  A01N43/90 ,  A01N43/40 ,  A01N37/50 ,  A01N2300/00

Abstract: The invention relates to fungicide mixtures containing A) imidazole derivatives of formula (I) wherein R and R represent halogen and phenyl which can be substituted by halogen or alkyl, or R and R together with the bridging C=C double bond form a 3,4-difluoromethylene dioxyphenyl group, R represents cyano or halogen, and R represents di-(C1-C4-alkyl) amino or isoxazol-4-yl which can carry two C1-C4 alkyl radicals; and B) at least one phenylacetic acid derivative (II) selected from the group of formulae (IIa) to (IIe), in a synergistically active quantity. The invention also relates to methods for controlling pathogenic fungi using mixtures of compounds (I) and (II) (IIa to IIe), in addition to agents containing the same.

Abstract translation: 本发明涉及含有在R杀真菌混合物<1>和R <2>是可被卤素或烷基A取代卤素和苯基）（式I的咪唑衍生物），或R <1>和R <2 >一起与桥接C = C双键形成3,4- Difluormethylendioxyphenyl基; [R <3>是氰基或卤素，且R <4>二 - （C1-C4烷基）氨基或异恶唑-4-基，其可带有两个C1-C4烷基基团; 和B）至少一种以协同有效量选自下组的式（IIA）至（IIE）的选择的苯乙酸衍生物II中，用于控制使用的化合物的混合物防治有害真菌的I和II（IIA至IIE）和包含它们的组合物的方法。

公开(公告)号：WO9920615A3

公开(公告)日：1999-06-24

申请号：PCT/EP9806299

申请日：1998-10-05

Applicant: BASF AG ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/82 ,  A01N43/836 ,  C07C259/14 ,  C07C265/12 ,  C07D271/06 ,  C07D271/07 ,  C07D413/12 ,  C07C239/12 ,  C07C251/38 ,  C07D413/14

CPC classification number: C07D271/07 ,  A01N43/82 ,  C07C259/14 ,  C07C265/12 ,  C07D413/12

Abstract: The invention relates to substituted phenyl carbamates of formula (I), wherein E represents a group A or B, # characterises the bond with the phenyl ring, and R , R , Y, n, T, and Z have the meanings given in the description.

Abstract translation: 本发明涉及式（I），其中E是基团A或B，其中＃为键合到苯基环的特征的取代的苯基氨基甲酸酯，且R <阿尔法>，R <克（B）>，Y，N，T 和Z具有描述中给出的含义。

公开(公告)号：WO03008417A9

公开(公告)日：2003-10-30

申请号：PCT/EP0207578

申请日：2002-07-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 式（I）的取代的6-（2-甲苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5-或6-元杂环基，或者含有1-4个氮原子或1-3个氮原子的5-或6-元杂芳基， 硫或氧原子，或者其中R 1和R 2基团可以如说明书中所定义的那样未被取代或被取代，或者R 1和R 2与中间的氮原子一起表示5或6 - 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的可被取代的 - 元杂环; R 3是卤素，氰基，烷基，烷氧基，卤代烷基或C（= O）A，其中A是氢，羟基，烷基，氨基或单或二烷基氨基; n是1至4的整数; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 它们的制备方法，含有它们的组合物以及它们用于防治植物病原性真菌的用途。

公开(公告)号：WO02074753A3

公开(公告)日：2002-12-27

申请号：PCT/EP0202739

申请日：2002-03-13

Applicant: BASF AG ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

CPC classification number: C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

Abstract: The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group 0, N or S, and which can be substituted as defined in the description; R represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R and R can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R and R represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, halogen, alkyl or halogenalkyl; and R represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi.

Abstract translation: 式（I）其中取代基具有以下Begende含义的5-苯基嘧啶，R <1> 5〜10元饱和，部分不饱和或芳族单环或双环杂环，选自下组0含有一至四个杂原子，N或 如说明书中所定义的可被取代的S，R <2>为氢，卤素，氰基，烷基，卤代烷基或烷氧基; [R <3>，R <4>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R <3>和R <4>可与氮原子一起他们 连接，形成可以被杂原子中断并且可以携带一个或多个取代基的五元或六元环; [R <5> - [R <6>是氢，卤素，烷基，卤代烷基或烷氧基; [R <7> - [R <8>是氢，卤素，烷基或卤代烷基; [R <9>是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰，卤代烷氧基或烷氧羰，涉及用于制备这些化合物和它们在防治有害真菌中的用途的方法和中间体。