公开(公告)号：WO02074753A3

公开(公告)日：2002-12-27

申请号：PCT/EP0202739

申请日：2002-03-13

Applicant: BASF AG ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

CPC classification number: C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

Abstract: The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group 0, N or S, and which can be substituted as defined in the description; R represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R and R can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R and R represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, halogen, alkyl or halogenalkyl; and R represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi.

Abstract translation: 式（I）其中取代基具有以下Begende含义的5-苯基嘧啶，R <1> 5〜10元饱和，部分不饱和或芳族单环或双环杂环，选自下组0含有一至四个杂原子，N或 如说明书中所定义的可被取代的S，R <2>为氢，卤素，氰基，烷基，卤代烷基或烷氧基; [R <3>，R <4>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R <3>和R <4>可与氮原子一起他们 连接，形成可以被杂原子中断并且可以携带一个或多个取代基的五元或六元环; [R <5> - [R <6>是氢，卤素，烷基，卤代烷基或烷氧基; [R <7> - [R <8>是氢，卤素，烷基或卤代烷基; [R <9>是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰，卤代烷氧基或烷氧羰，涉及用于制备这些化合物和它们在防治有害真菌中的用途的方法和中间体。

公开(公告)号：WO0248146A2

公开(公告)日：2002-06-20

申请号：PCT/EP0114577

申请日：2001-12-12

Applicant: BASF AG ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D471/04 ,  C07D487/04

CPC classification number: C07D471/04 ,  A01N43/90 ,  C07D487/04

Abstract: The invention relates to the use of substituted imidazoazines of formula (I), in which the variables have the following meanings: R represents alkyl, phenyl, phenylalkyl, naphthyl, anthracenyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, or condensed 8-membered to 12-membered hetaryl or condensed 8-membered to 12-membered heterocyclyl, containing one to four N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, whereby R can be unsubstituted or can be substituted as cited in the description; R and R represent hydrogen, alkyl, alkenyl, alkynyl, alkyl halide, alkenyl halide, alkynyl halide, trialkyl silylalkyl, phenyl, phenylalkyl or R and R , together with the bridging N atom, form a 5-membered or 6-membered heterocyclic or heteroaromatic ring, which can be interrupted by one to three N atoms and/or one O atom or S atom or by one or two O atoms and/or S atoms, and which can be substituted; A and B represent N or CR ; R , R and R represent hydrogen, halogen, cyano, nitro, hydroxy, alkyl, alkyl halide, cycloalkyl, alkoxy, alkoxy halide, alkylthio, amino, alkyl amino, dialkylamino, alkenyl, alkenyloxy, alkynyl or alkynyloxy. The inventive compounds are used for controlling phytopathogenic harmful fungi. The invention further relates to agents containing the inventive compounds, to novel imidazoazines, and to methods for the production thereof.

Abstract translation: 使用式（I）的取代的Imidazoazinen的，其中各变量具有以下含义：R t <1>是烷基，苯基，苯基烷基，萘基，蒽基，环烷基，5-或6-员杂芳基或5-或6-元杂环基 含有1至3个N原子和/或一个O或S原子或一个或两个O和/或S原子，或稠合8-12 gliederiges杂芳基或稠合的8-12 gliederiges杂环基， 含有一至四个N原子和/或一个O或S原子或一个或两个O和/或O原子，其中R是未取代的<1>或作为可在本说明书中被取代; [R <2>，R <3>是氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，三烷基甲硅烷基，苯基，苯基烷基或R <2>，R <3>连同桥接氮原子的5-或6- 形成 - 元杂环基或可被一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子被中断杂芳族环; A，B，N或CR <4>; [R <4>，R <5> - [R <6>为氢，卤素，氰基，硝基，羟基，烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，烷硫基，氨基，烷基氨基，二烷基氨基，烯基，烯氧基，炔氧基或炔氧基; 防治植物病原性有害真菌的，含有它们，它们的制备新imidazoazines和方法的组合物。

公开(公告)号：WO0020399A3

公开(公告)日：2000-07-27

申请号：PCT/EP9907125

申请日：1999-09-24

Applicant: BASF AG ,  GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D231/08 ,  C07D401/04 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

CPC classification number: C07D401/04 ,  C07D231/08 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

Abstract: The invention relates to the use of substituted 5-hydroxypyrazoles of formula (I) in which the substituents have the following meanings: B represents aryl or heteroaryl; A represents C=O, C=S or SO2; R represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, cycloalkyl, C3-C10-cycloalkenyl, cycloalkynyl, or aryl, heterocyclyl or heteroaryl; R represents hydrogen; R represents hydrogen, nitro, cyano, N(R')2, alkyl, alkyl halide, alkoxy, alkoxy halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, whereby R', independent of one another, represents hydrogen or alkyl; or R and R , together, represent a group =O, =S or =N-O-R , whereby R represents hydrogen, alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide; R represents hydrogen, halogen, nitro, cyano N(R')2, alkyl, alkyl halide, COOR', heteroaryl or heterocyclyl. The invention also relates to the use of said compounds for combating harmful fungi, to agents containing the compounds, to novel 5-hydroxypyrazoles and to methods for the production thereof.

Abstract translation: 本发明涉及式（I）的5-羟基吡唑啉的用途，其中取代基具有以下含义：B芳基或杂芳基; A C = O，C = S或SO 2; R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，C 3 -C 10 - 环烯基，环炔基或芳基，杂环基或杂芳基; R 2氢; [R <3>为氢，硝基，氰基，N（R '）2，烷基，卤代烷基，烷氧基，卤代烷氧基，链烯基，卤代烯基，炔基或卤代炔基，其中R' 独立地为氢或烷基; 或R <2>和R <3>一起表示基团= O，= S或= N-O-R <5>，其中R <5>是氢，烷基，卤代烷基，链烯基，卤代烯基，炔基或卤代炔基; R 4是氢，卤素，硝基，氰基，N（R'）2，烷基，卤代烷基，COOR'，杂芳基或杂环基; 用于控制有害真菌，含有它们的试剂和新的5-羟基吡唑及其制备方法。

公开(公告)号：WO2008012234A2

公开(公告)日：2008-01-31

申请号：PCT/EP2007057353

申请日：2007-07-17

Applicant: BASF AG ,  DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

Inventor： DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

IPC: C07D405/14 ,  A01N43/707 ,  C07D409/14

CPC classification number: C07D405/14 ,  A01N43/653 ,  C07D409/14

Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.

Abstract translation: 本发明涉及通式（I），其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素，CN，NO _{2 ，氨基，C <五 SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4卤代烷，C 1 -C 4 烷基氨基， ç 1 -C 4 二烷基氨基，硫代，或C 1 -C 4 是烷硫基，被取代的，和 各其他取代基A或B为苯基或5元或6元杂芳基，所述取代基任选地被1-3个下列取代基取代：卤素，CN，NO 2 ，氨基，C < SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 二烷基氨基，巯基或C 1 -C 4 - 烷硫基，被取代的，和它们的植物耐受的酸加成盐或金属盐，使用式（I）的用于控制植物病原真菌包含它们的化合物和试剂。}

公开(公告)号：WO2005113555A8

公开(公告)日：2006-12-14

申请号：PCT/EP2005005270

申请日：2005-05-13

Applicant: BASF AG ,  BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.

Abstract translation: 本发明涉及如下通式的新型三唑并嘧啶化合物I和它们在防治有害真菌中的用途，以及植物保护剂，这样的化合物作为活性成分enthalten.In式I，X，Y，L，M，Ar和A具有下列含义：X 卤素，氰基，C _{1 -C 4 烷基，C 1 -C 4 卤代烷基，C < SUB> 1 -C 4 - 烷氧基或C 1 -C 4 卤代烷氧基; Y是卤素，C 1 -C 4 烷基或C 1 -C 4 卤代烷基; 独立地为卤素，C 1 -C 6 烷基，C 2 -C 6 烯基，C 1 -C ç 6 卤代烷基，C 1 -C 6 烷氧基，C 1 -C 6 < / SUB>卤代烷氧基，硝基，氨基，NHR，NR 2 ，氰基，S（= O）名词 A“或C（= O）A ^{2 ; m是0，1，2，3或4; A是一个化学键或基团CR 4 - [R 5 是; Ar是苯基或5-或6-元杂芳基具有1个，选自O，S和N的杂原子作为环成员，其中苯基和杂芳基可以具有一个稠合的苯环和1，2，3 2或3 ，4或5个取代基R 一可以包括;. R“至R 3 具有权利要求1中给出的含义。}}

公开(公告)号：WO2005121146A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005006171

申请日：2005-06-08

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/647 ,  A01N43/90 ,  C07D487/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to triazolopyrimidines of formula (I), wherein the index n and the substituents R, R

Abstract translation: 本发明涉及下式的三唑并嘧啶I，其中索引n和取代基R，R

公开(公告)号：WO2005010000A3

公开(公告)日：2005-05-19

申请号：PCT/EP2004007924

申请日：2004-07-15

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  C07D471/04

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R ; n stands for 1, 2, 3, 4 or 5; R represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R , and R represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

Abstract translation: 本发明涉及通式I的双环化合物，其中X，Y彼此独立地是N或C-R 4; n是1,2,3,4或5; ř表示卤素，氰基，C1-C6烷基，C1-C6烷氧基，C1-C6卤代烷基，C1-C6卤代烷氧基，C2-C6链烯基，C2-C6链烯氧基或C （O）R 5代表; [R <1>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8-环烷基，其任选被烷基和/或卤素取代的或者 多取代，C5-C8环烯基，其任选与乘法烷基和/或卤素或单 - ，或<6>，SR <6>或NR <7> - [R <8>取代; [R <2>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8环烷基，任选地被烷基和/或卤素单取代的 或多取代的，C5-C8环烯基，其任选地被烷基和/或卤素取代基取代一次或多次，或<6>，SR <6>或NR <7> - [R <8>; R 3是任选被烷基和/或卤素单取代或多取代的氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; 和化合物（I），植物保护剂的农业上可接受的盐，其包含通式（I）和/或（I）的农业上可接受的盐和至少一种液体或固体载体和用于防治植物病原性有害真菌的方法中的至少一种化合物。

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9920615A3

公开(公告)日：1999-06-24

申请号：PCT/EP9806299

申请日：1998-10-05

Applicant: BASF AG ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/82 ,  A01N43/836 ,  C07C259/14 ,  C07C265/12 ,  C07D271/06 ,  C07D271/07 ,  C07D413/12 ,  C07C239/12 ,  C07C251/38 ,  C07D413/14

CPC classification number: C07D271/07 ,  A01N43/82 ,  C07C259/14 ,  C07C265/12 ,  C07D413/12

Abstract: The invention relates to substituted phenyl carbamates of formula (I), wherein E represents a group A or B, # characterises the bond with the phenyl ring, and R , R , Y, n, T, and Z have the meanings given in the description.

Abstract translation: 本发明涉及式（I），其中E是基团A或B，其中＃为键合到苯基环的特征的取代的苯基氨基甲酸酯，且R <阿尔法>，R <克（B）>，Y，N，T 和Z具有描述中给出的含义。

公开(公告)号：WO2006092428A2

公开(公告)日：2006-09-08

申请号：PCT/EP2006060399

申请日：2006-03-02

Applicant: BASF AG ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  RACK MICHAEL

Inventor： GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  RACK MICHAEL

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04

Abstract: The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.

Abstract translation: 2-取代的式（I）其中取代基具有以下含义的7-氨基azolopyrimidines：R t ^{1 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基， benzyloxyalkyl，烷氧基烯基或alkoxyalkynyl; [R 2 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基和烷硫基烷基，其中在R中的碳链 1 和/或R 2 可以根据描述被取代; [R 3 为卤素，氰基，NR 一 - [R 乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基， 羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯丙氨酸nylthio，苄氧基，苄硫基，烷基-S（O）_{米 - ; A N和CR X ; ，R 3 基 X 是氢或其中R 称作; 的方法和中间体制备这些化合物，含有它们和它们在防治植物病原性有害真菌的组合物。}}