公开(公告)号：WO2005110080A2

公开(公告)日：2005-11-24

申请号：PCT/EP2005005070

申请日：2005-05-11

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N20060101 ,  A01N43/90 ,  A01N

CPC classification number: A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R is alkyl, halogenalkyl, alkenyl or cyclopentyl, R is hydrogen or alkyl, R and R together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L is fluorine or chlorine, L , L are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (I) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

Abstract translation: 一种杀真菌混合物，其包含作为活性组分：1）式（I）的5-甲基-7-氨基三唑并嘧啶，其中R <1>是烷基，卤代烷基，链烯基或环戊基; [R <2>是氢或烷基; [R <1>和R <2>也可以与氮原子一起与它们所连接的形式，其可以由甲基取代的哌啶环; →<1>是氟或氯; →<2>，L <3>独立地是氢，氟或氯; 和2）选自组A）唑类中的至少一种活性化合物; B）嗜球果伞素; C）酰基丙氨酸类; D）胺衍生物; E）苯胺基嘧啶; F）二甲酰亚胺; G）肉桂酸和类似物; 1H）抗生素; K）二硫代氨基甲酸酯; L）杂环化合物; M）硫和铜杀真菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）Sulfensäurederivate; Q）其他杀菌剂; R）Wachstumsretardantien; 根据描述; 在协同有效量; 新的三唑并嘧啶，用于控制使用I化合物的混合物与基团A），以R的活性成分）包含这些混合物的有害真菌及其制造这样的混合物使用I化合物与基团A）至R）的活性成分和组合物的方法 ，

公开(公告)号：WO2005113555A8

公开(公告)日：2006-12-14

申请号：PCT/EP2005005270

申请日：2005-05-13

Applicant: BASF AG ,  BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.

Abstract translation: 本发明涉及如下通式的新型三唑并嘧啶化合物I和它们在防治有害真菌中的用途，以及植物保护剂，这样的化合物作为活性成分enthalten.In式I，X，Y，L，M，Ar和A具有下列含义：X 卤素，氰基，C _{1 -C 4 烷基，C 1 -C 4 卤代烷基，C < SUB> 1 -C 4 - 烷氧基或C 1 -C 4 卤代烷氧基; Y是卤素，C 1 -C 4 烷基或C 1 -C 4 卤代烷基; 独立地为卤素，C 1 -C 6 烷基，C 2 -C 6 烯基，C 1 -C ç 6 卤代烷基，C 1 -C 6 烷氧基，C 1 -C 6 < / SUB>卤代烷氧基，硝基，氨基，NHR，NR 2 ，氰基，S（= O）名词 A“或C（= O）A ^{2 ; m是0，1，2，3或4; A是一个化学键或基团CR 4 - [R 5 是; Ar是苯基或5-或6-元杂芳基具有1个，选自O，S和N的杂原子作为环成员，其中苯基和杂芳基可以具有一个稠合的苯环和1，2，3 2或3 ，4或5个取代基R 一可以包括;. R“至R 3 具有权利要求1中给出的含义。}}

公开(公告)号：WO2006066818A3

公开(公告)日：2006-11-02

申请号：PCT/EP2005013577

申请日：2005-12-16

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D213/55 ,  C07D237/14 ,  C07D487/04

Abstract: The invention relates to novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds and the salts thereof that can be used in agriculture, the use of the same for controlling pathogenic fungi, and plant protection agents containing at least one such compound as an active constituent. Said novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds correspond to general formula (I) wherein the substituents R 1 , R 2 , Het, X and Y have the following designations: Het represents a six-membered heteroaromatic radical selected from pyridinyl, pyridazinyl, pyrazinyl, 1,2,4-triazinyl and 1,3,5-triazinyl, the six-membered heteroaromatic radical comprising 1, 2 or 3 substituents L which are the same or different, R 1 , R 2 independently represent hydrogen, C 1 -C 8 alkyl, C 1 -C 8 halogenalkyl, C 1 -C 8 alkoxy, C 3 -C 8 cycloalkyl, C 3 -C 8 cycloalkoxy, C 5 -C 10 bicycloalkyl, C 3 -C 8 halogencycloalkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkenyloxy, C 4 -C 10 alkadienyl, C 2 -C 8 halogenalkenyl, C 3 -C 8 cycloalkenyl, C 3 -C 8 halogencycloalkenyl, C 2 -C 8 alkinyl, C 2 -C 8 alkinyloxy, C 2 -C 8 halogenalkinyl, NH 2, C 1 -C 8 alkylamino, Di-C 1 -C 8 -alkylamino, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle, X represents hydrogen, halogen, OH, cyano, C 1 -C 4 alkyl and the like, and Y represents hydrogen, halogen, cyano, C 1 -C 4 alkyl, and the like.

Abstract translation: 本发明涉及新颖的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物及其农业上可接受的盐，以及它们在防治有害真菌中的用途，以及植物保护剂，这些化合物的至少一种作为 含有活性成分。 新的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物可通过通式（I）所示，其中取代基R ^{1 来表示 ，R 2 ，（I）的Het，X和Y在式具有以下含义：Het是其选自吡啶基，哒嗪基，吡嗪基的6元杂芳基，1,2,4- 三嗪基和1,3,5-三嗪基，其中所述6元杂芳基1，2或3个相同或不同的取代基L可以包括，R 1 ，R 2 独立地 另一个氢，C _{1 -C 8 烷基，C 1 -C 8 卤代烷基，C 1 -C 8 烷氧基，C 3 -C 8 环烷基，C 3 -C 8 环烷氧基，C 5 -C 10 双环，C 3 -C 8 卤代环烷基，C 2 -C 8 烯基，C 2 -C 8 烯 ，C 4 -C 10 链二烯基，C 2 -C 8 卤代，C 3 -C 8 环烯基，C 3 -C 8 卤代环，C 2 -C 8 炔基，C 2 -C 8 炔氧基，C 2 -C 8 卤代炔基，NH 2 C 1 -C 8 烷基氨基，二-C 1 -C 8 烷基氨基，苯基，萘基或五 - 或六元饱和，部分不饱和或芳族的杂环，X是氢，卤素，OH，氰基，C < SUB> 1 -C 4 烷基等，Y是氢，卤素，氰基，C 1 -C 4 烷基， 等等。}}

公开(公告)号：WO2005121146A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005006171

申请日：2005-06-08

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/647 ,  A01N43/90 ,  C07D487/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to triazolopyrimidines of formula (I), wherein the index n and the substituents R, R

Abstract translation: 本发明涉及下式的三唑并嘧啶I，其中索引n和取代基R，R

公开(公告)号：WO2005010000A3

公开(公告)日：2005-05-19

申请号：PCT/EP2004007924

申请日：2004-07-15

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  C07D471/04

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R ; n stands for 1, 2, 3, 4 or 5; R represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R , and R represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

Abstract translation: 本发明涉及通式I的双环化合物，其中X，Y彼此独立地是N或C-R 4; n是1,2,3,4或5; ř表示卤素，氰基，C1-C6烷基，C1-C6烷氧基，C1-C6卤代烷基，C1-C6卤代烷氧基，C2-C6链烯基，C2-C6链烯氧基或C （O）R 5代表; [R <1>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8-环烷基，其任选被烷基和/或卤素取代的或者 多取代，C5-C8环烯基，其任选与乘法烷基和/或卤素或单 - ，或<6>，SR <6>或NR <7> - [R <8>取代; [R <2>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8环烷基，任选地被烷基和/或卤素单取代的 或多取代的，C5-C8环烯基，其任选地被烷基和/或卤素取代基取代一次或多次，或<6>，SR <6>或NR <7> - [R <8>; R 3是任选被烷基和/或卤素单取代或多取代的氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; 和化合物（I），植物保护剂的农业上可接受的盐，其包含通式（I）和/或（I）的农业上可接受的盐和至少一种液体或固体载体和用于防治植物病原性有害真菌的方法中的至少一种化合物。

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9926930A2

公开(公告)日：1999-06-03

申请号：PCT/EP9807099

申请日：1998-11-06

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT

Inventor： RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D413/06 ,  C07D413/10 ,  C07D417/10 ,  C07D231/18

CPC classification number: C07D413/06 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20

Abstract: The invention relates to benzylidene pyrazolones of formula (I), wherein the substituents and index n have the following meanings: R = optionally substituted C1-C6 alkyl; R = optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, halogen, nitro, cyano; R = hydrogen, halogen, nitro, cyano, a group NR R , OCOR , NR COR ,CO2R , -COSR , -CONR R , C1-C4-alkoxyiminoalkyl, C1-C6 alkoxycarbonyl, optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, optionally substituted C1-C6 alkylthio, optionally substituted C2-C6 alkenyl, optionally substituted phenyl, optionally substituted phenoxy, an optionally substituted 5- or 6-membered saturated or unsaturated heterocycle which can contain up to 4 nitrogen atoms and/or up to 2 oxygen or sulphur atoms as ring members; R = C1-C6 alkyl, C1-C4 halogen alkyl; or R and R = an optionally substituted saturated or unsaturated 2- or 3-membered bridge which can contain one sulphur atom which can be oxidized into sulfoxide or sulfone, R = hydrogen or optionally substituted C1-C6 alkyl; R = hydrogen, C1-C6 alkyl or C1-C4 halogenalkyl; n = 0, 1 or 2; X = hydrogen, chlorine or bromine. The compounds to which claim is laid are available in both a trans and a cis form or can be a mixture of these isomers.

Abstract translation: 式（I）的Benzylidenpyrazolone其中取代基和指数n具有以下含义：R t <1>是未取代的或取代的。 C1-C6烷基; [R <2>是未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，卤素，硝基，氰基; [R <3>是氢，卤素，硝基，氰基，基团NR <5> - [R <6>，OCOR <5>，NR <5> COR <6>，CO 2 <5>，-COSR <5>，-CONR <5> - [R <6>，C1-C4-alkoxyiminoalkyl，C1-C6烷基羰基，未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，未取代的或取代的。 C1-C6烷硫基，未取代或取代的。 C2-C6链烯基，未取代的或取代的。 C2-C6炔基，未取代的或取代的。 苯基，未取代的或取代的。 苯氧基，未取代的或取代的。 5-或6-元饱和或可含有至多4个氮原子和/或至多2个氧或硫原子作为环成员的不饱和的杂环; [R <4> C1-C6-烷基，C1-C4卤代烷基; 或R <3>，R <4>为可以含有可被氧化为亚砜或砜硫原子的任选取代的饱和或不饱和2-或3-元桥; [R <5>为氢或未取代或取代的。 C1-C6烷基; [R <6>是未取代的或取代的。 C1-C6烷基; [R <7>是氢，C1-C6烷基或C1-C4卤代烷基; n为0.1或2; X是氢，氯或溴; 其中要求保护的化合物在跨及在所述顺式 - 形式两者呈现，或者可以是这些异构体的混合物。

公开(公告)号：WO2006114405A2

公开(公告)日：2006-11-02

申请号：PCT/EP2006061786

申请日：2006-04-24

Applicant: BASF AG ,  DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA

Inventor： DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  LOHMANN JAN KLAAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA

IPC: A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.

Abstract translation: 式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I：其中各变量具有以下含义：Y是任选被烷基取代的亚烷基，亚烯基或亚炔基; [R ^{1 为卤素，氰基，硝基，羟基，巯基，烷基，卤代烷基，链烯基，环烷基，环烯基，烷氧基，卤代烷氧基，烯氧基，炔氧基，烷硫基，NR 一 - [R < SUP>乙，烷基羰基，苯基，萘基或五 - 或六元饱和环，其包含选自一至四个杂原子的部分不饱和或罗马杂环O，N或S; [R 一，R 乙是氢，烷基和烷基羰基; n是零，1，2，3或4; [R 2 烷基，烯基，环烷基，烷氧基烷基和烷硫基烷基; [R 3 为氢，卤素，氰基，NR 一 - [R 乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基， 环烷硫基，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O）_{米 - ; m是0，1或2; A N和C-R 一; [R 一氢和烷基; 其中Y中的碳原子，R 1 ，R 2 ，R 3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines，处理用于制备这些化合物和含有它们的组合物。}}

公开(公告)号：WO2006097488A8

公开(公告)日：2006-11-02

申请号：PCT/EP2006060752

申请日：2006-03-15

Applicant: BASF AG ,  PUHL MICHAEL ,  KORADIN CHRISTOPHER ,  RHEINHEIMER JOACHIM ,  GRAMMENOS WASSILIOS ,  LOHMANN JAN KLAAS ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  LANGEWALD JUERGEN ,  GOETZ NORBERT ,  ANSPAUGH DOUGLAS D ,  CULBERTSON DEBORAH L ,  COTTER HENRY VAN TUYL ,  OLOUMI-SADEGHI HASSAN

Inventor： PUHL MICHAEL ,  KORADIN CHRISTOPHER ,  RHEINHEIMER JOACHIM ,  GRAMMENOS WASSILIOS ,  LOHMANN JAN KLAAS ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  LANGEWALD JUERGEN ,  GOETZ NORBERT ,  ANSPAUGH DOUGLAS D ,  CULBERTSON DEBORAH L ,  COTTER HENRY VAN TUYL ,  OLOUMI-SADEGHI HASSAN

IPC: A01N43/40 ,  A01N43/42 ,  A01P7/00 ,  C07D213/36 ,  C07D215/12 ,  C07D333/34

CPC classification number: C07D213/42 ,  A01N43/40 ,  A01N43/42 ,  C07D215/12 ,  C07D409/12

Abstract: N-(4-Pyridyl)methylsulfonamides for combating arthropodal pests The present invention relates to the use of N-(4-pyridyl)methylsulfonamides of the formula for combating arthropodal pests (harmful arthropodes) and for protecting materials against infestation and/or destruction by said pests: (I) where the substituents are as follows: R 1 is hydrogen, C 1 -C 4 -alkyl, C 1- C 4 -alkoxy, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl or benzyl; R 2 , R 3 , R 4 , R 5 independently of one another are hydrogen, halogen, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkoxy or C 1 -C 4 -haloalkyl; R 2 and R 3 or R 4 and R 5 together with the carbon atoms to which they are attached may also form a condensed 5- or 6-membered hydro- carbon ring, it being possible for the hydrocarbon ring to carry one or two groups R 2' , R 3' , R 2' , R 3' independently of one another are halogen, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, halomethoxy or halomethyl; X is a cyclic radical selected from phenyl, naphthyl and five- or six-membered saturated, partially unsaturated or aromatic heterocycles, the heterocycle being attached to the sulfur atom via a carbon atom and containing 1 , 2 or 4 heteroatoms selected from the group consisting of O, N and S, where the cyclic radical X may carry 1 , 2, 3 or 4 substituents R a .

Abstract translation: 用于对抗节肢动物害虫的N-（4-吡啶基）甲基磺酰胺本发明涉及下式的N-（4-吡啶基）甲基磺酰胺用于防治节肢动物害虫（有害的节肢动物）和用于保护物质免受感染和/或破坏的物质 所述害虫：（I）其中取代基如下：R 1是氢，C 1 -C 4 - 烷基，C

公开(公告)号：WO2005110088A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005005068

申请日：2005-05-11

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  RHEINHEIMER JOACHIM

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  RHEINHEIMER JOACHIM

IPC: A01N43/90 ,  A01N43

CPC classification number: A01N43/90 ,  A01N43/86 ,  A01N43/54 ,  A01N43/16 ,  A01N43/42 ,  A01N2300/00

Abstract: The inventive fungicide mixtures contain as active components 1) a of formula (I) and 2) at least one component of formula (II), wherein variables have the following meanings: A is O or N, B is N or a direct bond, G is C or N, R

Abstract translation: 一种杀真菌混合物，其包含作为活性组分1）式（I）的三唑并嘧啶衍生物，以及2）式的至少一种化合物（II），其中各变量具有以下含义：A是O或N; B是N或直接键; G是C或N; [R