AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS
    21.
    发明申请
    AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    用于组合动物疫苗的咪唑烷化合物

    公开(公告)号:WO2006097279A1

    公开(公告)日:2006-09-21

    申请号:PCT/EP2006/002331

    申请日:2006-03-14

    CPC classification number: C07C259/20 A01N37/52 C07C2601/02

    Abstract: The present invention relates to new amidrazone compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids. The amidrazone compounds are of the general formula (I) including the tautomers of I and the salts thereof; wherein X and Y are hydrogen or together form a chemical bond; Ar is an aromatic radical selected from phenyl and a 5- or 6-membered heteroaryl having 1 , 2, 3 or 4 heteroatoms as ring members, which are selected, independently of one another, from O, N and S, and where the aromatic radical may have 1 , 2, 3, 4 or 5 substituents R a ; R 1 is selected from the group consisiting of C 1 -C 1O -alkyl, C 1 -C 4 -alkoxy-C 1 -C 4 -alkyl, cyano-C 1 -C 4 -alkyl, hydroxy-C 1- C 4 -alkyl, C 1 -C 10 -haloalkyl, tri-(C 1 -C 4 -alkyl)-silyl-C 1 - C 4 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 -haloalkynyl, C 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1 C 4 -alkyl, phenyl-C 1 -C 4 - alkyl and heteroaryl-C 1 C 4 alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above; R 2 is selected from the group consisiting of C 1- C 1 0-alkyl, c 1- c 4 -alkoxy- C 1- C 4 -alkyl, C 1- C 10 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 - haloalkynyl,c 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1- C 4 -alkyl, phenyl-C 1 -C 4 -alkyl and heteroaryI-C 1- C 4 -alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above.

    Abstract translation: 本发明涉及可用于对抗动物害虫,特别是昆虫,蜘蛛和线虫的新的氨基腙化合物。 本发明还涉及一种防治昆虫,线虫和蜘蛛的方法。 氨基腙化合物具有通式(I),其包括I的互变异构体及其盐; 其中X和Y是氢或一起形成化学键; Ar是选自苯基和具有1,2,3或4个杂原子作为环成员的5-或6-元杂芳基的芳族基团,其彼此独立地选自O,N和S,并且其中芳族 基团可以具有1,2,3,4或5个取代基R a, R 1选自C 1 -C 10 - 烷基,C 1 -C 1 - 烷基, C 1 -C 4烷基,C 1 -C 4烷基,C 1 -C 4烷基,氰基-C 1 -C 4烷基, C 1 -C 6烷基,羟基-C 1 -C 4 - 亚烷基,C 1 -C 10 - 烷基, 卤代烷基,三 - (C 1 -C 4 - 烷基) - 甲硅烷基-C 1 -C 4 - 烷基,C 2 -C 10 - 烯基,C 2 -C 10 - 卤代烯基,C 1 -C 10 - C 2 -C 10 - 炔基,C 2 -C 10 - 卤代炔基,C 3 - C 10 - 环烷基,苯基,杂芳基,C 3 -C 10 - 环烷基-C 1 -C C 1-4烷基,苯基-C 1 -C 4 - 烷基和杂芳基-C 1 -C 4烷基, 其中C 3 -C 10 - 环烷基,杂芳基和苯基在后面六个提及的基团中可以是未取代的或携带1,2,3,4或4个 5个取代基R b如上所定义; R 2选自C 1 -C 1-4烷基,C 1 -C 4烷基, C 1-4烷基,C 1 -C 10烷基,C 1 -C 4烷基,C 1〜 亚烷基,C 2 -C 10 - 烯基,C 2 -C 10 - 卤代烯基,C C 2 -C 10 - 炔基,C 2 -C 10 - 卤代炔基,C 3 - C 1 -C 10 - 环烷基,苯基,杂芳基,C 3 -C 10 - 环烷基-C 1 - C 1 -C 4 - 烷基,苯基-C 1 -C 4 - 烷基和杂芳基C 1 -C 其中C 3 -C 10 - 环烷基,最后六个所述基团中的杂芳基和苯基可以是未取代的或携带1, 2,3,4或5个如上定义的取代基R b。

    3-HETEROARYLSUBSTITUIERTE 5 METHYLOXYMETHYL-ISOXAZOLINE ALS HERBIZIDE
    25.
    发明申请
    3-HETEROARYLSUBSTITUIERTE 5 METHYLOXYMETHYL-ISOXAZOLINE ALS HERBIZIDE 审中-公开
    3 - 杂芳基 - 取代的异恶唑啉5甲氧基甲基-AS除草剂

    公开(公告)号:WO2003090539A1

    公开(公告)日:2003-11-06

    申请号:PCT/EP2003/004136

    申请日:2003-04-22

    Abstract: Die vorliegende Erfindung betrifft 3-heteroarylsubstituerte Isoxazoline der Formel (I): in der die Variablen die folgenden Bedeutungen haben: X substituiertes 5-gliedriges Heteroaryl mit ein bis vier Stickstoffatomen, oder mit ein bis drei Stickstoffatomen und einem Sauerstoff- oder Schwefelatom, oder mit einem Sauerstoff- oder Schwefelatom; oder substituiertes 6-gliedriges Heteroaryl mit ein bis vier Stickstoffatomen; wobei das oben genannte 5-gliedrige Heteroaryl nicht Pyrazolyl oder Thienyl ist; R 1 - R 7 Wasserstoff, Alkyl oder Halogenalkyl; Y gegebenenfalls substituiertes Aryl, oder Benzo[1,4]dioxonyl, Benzo[1,3]dioxolanyl, 2,3-Dihydrobenzofuranyl oder Benzimidazol; oder gegebenenfalls substituiertes 5- bis 6-gliedriges Heteroaryl; sowie deren landwirtschaftlich brauchbaren Salze,Verfahren und Zwischenprodukte zu ihrer Herstellung; sowie die Verwendung dieser Verbindungen oder diese Verbindungen enthaltende Mittel zur Bekämpfung unerwünschter Pflanzen.

    Abstract translation: 本发明涉及式(I)的3- heteroarylsubstituerte异恶唑啉:其中各变量具有以下含义:X为取代的具有一至四个氮原子或具有一至三个氮原子和一个氧或硫原子,或具有5元杂芳基 一个氧或硫原子; 的或取代的具有一至四个氮原子的6元杂芳基; 其中,上述的5元杂芳基未被吡唑基或噻吩基; [R <1> - R的<7>是氢,烷基或卤代烷基; Y是任选取代的芳基,或苯并[1,4] dioxonyl,苯并[1,3]二氧戊环基,2,3-二氢苯并呋喃基或苯并咪唑; 或任选取代的5-至6-元杂芳基; 及其可农用盐,它们的制备方法和中间体; 和使用这些化合物或包含用于控制不希望的植物的装置这些化合物。

    α-CYANOACRYLATES
    26.
    发明申请
    α-CYANOACRYLATES 审中-公开
    阿尔法 - 氰基丙烯酸酯

    公开(公告)号:WO2003051824A1

    公开(公告)日:2003-06-26

    申请号:PCT/EP2002/014353

    申请日:2002-12-17

    Abstract: α-Cyanoacrylates of the formula (I), where: R 1 is OR a wherein R a is hydrogen, substituted alkyl, branched alkyl, branched alkenyl, cycloloalkyl, heterocyclyl, aryl, phenylalkyl or alkyl­imino; is NR b R c wherein R b is hydrogen, alkyl which may be substituted, alkenyl, alkynyl; R c is hydrogen, alkyl which may be substituted alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, phenylalkyl or alkylimino; or R b and R c form an alkandiyl-chain which may be substituted; or is SR d wherein R d is hydrogen, alkyl which may be substituted, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, phenylalkyl or alkylimino; R 2 is alkyl which may be substituted; is alkenyl or alkynyl; R 3 is alkyl may be substituted; is alkenyl or alkynyl; R 4 is hydrogen, halogen, cyano or alkyl; and their agriculturally useful salts, processes and intermediates for their preparation; and the use of these compounds or of compositions comprising these compounds for controlling undesirable plants are described.

    Abstract translation: 式(I)的烷基丙烯酸酯,其中:R 1是其中R a a是氢的取代的烷基,支链烷基 ,支链烯基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基; 其中R b是氢,可以被取代的烷基,烯基,炔基; 烯基,炔基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基; 或者R c和R c形成可以被取代的烷撑二链; 或者是其中R d为氢的烷基,可被取代的烷基,烯基,炔基,环烷基,杂环基,芳基,苯基烷基或烷基亚氨基; R 2是可被取代的烷基; 是烯基或炔基; R 3是烷基可以被取代; 是烯基或炔基; R 4是氢,卤素,氰基或烷基; 及其农业上有用的盐,其制备方法和中间体; 并且描述了这些化合物或包含这些化合物的组合物用于防治不期望的植物的用途。

    1-(IMIDAZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS
    29.
    发明申请
    1-(IMIDAZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-(咪唑烷-2-基)氨基-1,2-二苯醚化合物,用于组合动物乳剂

    公开(公告)号:WO2006125748A1

    公开(公告)日:2006-11-30

    申请号:PCT/EP2006/062419

    申请日:2006-05-18

    CPC classification number: A01N43/50 C07D233/48

    Abstract: The present invention relates to 1-(imidazolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and their agriculturally acceptable salts, wherein A is a radical of the formula A 1 or A 2 . The invention relates also to agricultural compositions and to seed comprising at least one compound I and/or a salt thereof, as well as a method of combating animal pests, a method for protecting crops from attack or infestation by animal pests and a method for protecting non-living materials from attack or infestation by animal pests, a method for the protection of seeds from animal pests and of the seedlings' roots and shoots from animal pests by applying a pesticidally effective amount of at least one 1-(imidazolin-2-yl)amino-1 ,2- diphenylethane compound I and/or a salt thereof.

    Abstract translation: 本发明涉及式I的1-(咪唑啉-2-基)氨基-1,2-二苯基乙烷化合物及其农业上可接受的盐,其中A是式A 1或 A 2 。 本发明还涉及农业组合物和包含至少一种化合物I和/或其盐的种子,以及防治动物害虫的方法,用于保护作物免受动物害虫侵袭或侵染的方法和保护方法 通过施用杀虫有效量的至少一种1-(咪唑啉-2-酮)的动物害虫的攻击或感染的非生物材料,动物害虫的种子保护方法和来自动物害虫的幼苗的根和芽, 吡啶-2-基)氨基-1,2-二苯基乙烷化合物I和/或其盐。

    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS
    30.
    发明申请
    1-(1,2-DIPHENYL-ETHYL)-3-(2-HYDROXYETHYL)-THIOUREA COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    1-(1,2-二苯基乙基)-3-(2-羟基乙基) - 硫脲化合物,用于组合动物饲料

    公开(公告)号:WO2006125745A2

    公开(公告)日:2006-11-30

    申请号:PCT/EP2006/062413

    申请日:2006-05-18

    CPC classification number: C07C335/12 A01N47/28

    Abstract: The present invention relates to a method of combating animal pests which comprises contacting the animal pest, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal at- tack or infestation, with a pesticidally effective amount of at least one 1-(1 ,2-diphenyl- ethyl)-3-(2-hydroxyethyl)-thiourea compound I or an agriculturally acceptable salt thereof, wherein m is 0 to 5, n is 0 to 5, R 3 and R 4 are H or optionally substituted alkyl, haloalkyl, cycloalkyl, phenyl or benzyl, R 7 , R 8 , R 9 and R 10 are H or optionally substituted C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 - alkylamino, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, phenyl or benzyl and the variables R 1 , R 2 , R 5 and R 6 are as defined in the claims. The invention relates also to a method for protecting crops from attack or infestation by animal pests, a method for protecting non-living materials from attack or infestation by animal pests, novel 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compounds I and their agriculturally acceptable salts as well as to an agricultural composition comprising a 1-(1 ,2-diphenyl-ethyl)-3-(2-hydroxyethyl)-thiourea compound I or a salt thereof.

    Abstract translation: 本发明涉及一种防治动物害虫的方法,包括使动物害虫,其习惯,繁殖地,食物供应,植物,种子,土壤,区域,动物害虫生长或可能生长的物质或环境接触,或 防止动物死亡或侵染的材料,植物,种子,土壤,表面或空间,具有杀虫有效量的至少一种1-(1,2-二苯基 - 乙基)-3-(2-羟乙基 ) - 硫脲化合物I或其农业上可接受的盐,其中m为0至5,n为0至5,R 3和R 4为H或任选取代的烷基 ,卤代烷基,环烷基,苯基或苄基,R 7,R 8,R 9和R 10是H 或任选取代的C 1 -C 6 - 烷基,C 1 -C 6 - 卤代烷基,C 1,R 2,R 5和R 6如权利要求中所定义。 本发明还涉及一种保护作物免受动物害虫侵袭或侵袭的方法,一种保护非生物材料免受动物害虫侵袭或侵染的方法,新的1-(1,2-二苯基 - 乙基)-3-( 2-羟乙基) - 硫脲化合物I及其农业上可接受的盐,以及包含1-(1,2-二苯基 - 乙基)-3-(2-羟乙基) - 硫脲化合物I或其盐的农业组合物。

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