MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-kB ACTIVITY AND USE THEREOF
    31.
    发明申请
    MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-kB ACTIVITY AND USE THEREOF 有权
    GLUCOCORTICOID受体的调节剂,AP-1和/或NF-kB活性及其用途

    公开(公告)号:US20090075995A1

    公开(公告)日:2009-03-19

    申请号:US11835438

    申请日:2007-08-08

    Abstract: Novel non-steroidal compounds are provided which are useful in treating diseases associated with modulation of the glucocorticoid receptor, AP-1, and/or NF-κB activity, including inflammatory and immune diseases, having the structure of formula (I): an enantiomer, diastereomer, or tautomer thereof, or a prodrug ester thereof, or a pharmaceutically-acceptable salt thereof, in which: Z is heterocyclo or heteroaryl; A is a 5- to 8-membered carbocyclic ring or a 5- to 8-membered heterocyclic ring; B is a cycloalkyl, cycloalkenyl, aryl, heterocyclo, or heteroaryl ring, wherein each ring is fused to the A ring on adjacent atoms and optionally substituted by one to four groups which are the same or different and are independently selected from R5, R6, R7, and R8; J1, J2, and J3 are at each occurrence the same or different and are independently -A1QA2-; Q is a bond, O, S, S(O), or S(O)2; A1 and A2 are the same or different and are at each occurrence independently selected from a bond, C1-3alkylene, substituted C1-3alkylene, C2-4alkenylene, and substituted C2-4alkenylene, provided that A1 and A2 are chosen so that ring A is a 5- to 8-membered carbocyclic or heterocyclic ring; R1 to R11 are as defined herein. Also provided are pharmaceutical compositions and methods of treating inflammatory- or immune-associated diseases and obesity and diabetes employing said compounds.

    Abstract translation: 提供了新的非甾体化合物,其可用于治疗与式(I)结构的糖皮质激素受体,AP-1和/或NF-κB活性(包括炎症和免疫疾病)调节相关的疾病:对映异构体 ,非对映异构体或其互变异构体,或其前药酯或其药学上可接受的盐,其中:Z是杂环或杂芳基; A是5至8元碳环或5至8元杂环; B是环烷基,环烯基,芳基,杂环基或杂芳基环,其中每个环与相邻原子上的A环稠合并任选地被一至四个相同或不同的基团取代,并且独立地选自R5,R6, R7和R8; J1,J2和J3各自出现相同或不同,独立地为-A1QA2-; Q是键,O,S,S(O)或S(O)2; A1和A2相同或不同,并且在每次出现时独立地选自键,C1-3亚烷基,取代的C1-3亚烷基,C2-4亚烯基和取代的C2-4亚烯基,条件是选择A1和A2使得环A为 5-至8-元碳环或杂环; R1至R11如本文所定义。 还提供了使用所述化合物治疗炎性或免疫相关疾病和肥胖症和糖尿病的药物组合物和方法。

    Self-Adpting Transmission Scheme of the Channel Environment in the Multiantenna Wireless Transmission System
    32.
    发明申请
    Self-Adpting Transmission Scheme of the Channel Environment in the Multiantenna Wireless Transmission System 有权
    多天线无线传输系统中通道环境的自适应传输方案

    公开(公告)号:US20080310542A1

    公开(公告)日:2008-12-18

    申请号:US12095194

    申请日:2006-11-24

    Abstract: An adaptive transmission scheme of the channel environment in the multi-antenna wireless transmission system can raise the spectrum use rate and power efficiency of the communication system in fast. Comparing with the traditional single antenna input and single antenna output, the channel environment in MIMO wireless communication system is more complex. When the terminal is moving, the different types of channels between terminal and base station can be gone through and then its capacity can be changed more largely. It is characterized in: at first, obtaining the statistical channel information at the receiving end using the result of channel estimation; then, quantizing and encoding the obtained statistical channel information to get feedback bit information and send the feedback bit information to the transmitting end through a feedback channel; thereby using statistical information, the sending end calculates link self-adapting control parameters, which are used for controlling coding modulation and sending the pre-code; the sending end obtains the digital base band transmission signal using a characteristic mode transmission method and a random virtual space selection transmission method, and the receiving end carries out self-adapting receiving by the same parameters.

    Abstract translation: 多天线无线传输系统中的信道环境的自适应传输方案可以快速提高通信系统的频谱利用率和功率效率。 与传统的单天线输入和单天线输出相比,MIMO无线通信系统中的信道环境更加复杂。 当终端移动时,终端和基站之间的不同类型的信道可以通过,其容量可以更大地改变。 其特征在于:首先,使用信道估计结果在接收端获取统计信道信息; 然后对获得的统计信道信息进行量化和编码以获得反馈比特信息,并通过反馈信道将反馈比特信息发送到发送端; 从而使用统计信息,发送端计算用于控制编码调制和发送预编码的链路自适应控制参数; 发送端使用特征模式发送方法和随机虚拟空间选择发送方法获得数字基带发送信号,接收端通过相同的参数进行自适应接收。

    LEVEL
    33.
    发明申请
    LEVEL 失效
    水平

    公开(公告)号:US20050145784A1

    公开(公告)日:2005-07-07

    申请号:US10899329

    申请日:2004-07-26

    CPC classification number: G01C15/004

    Abstract: A level. A projected plane is generated substantially parallel to a reference plane by a light source rotatably emitting light. A main shaft, having a rotary portion and a pair of protrusions and connecting to the light source, is perpendicular to the projected plane. A universal joint is disposed in a housing with the main shaft rotatably passing therethrough. A level sensor detects inclination of the projected plane deviated from the reference plane and outputs an adjustment signal. An adjustment mechanism has a first movable member and a second movable member crossing each other. The first movable member impels one protrusion along a first axis, and the second movable member impels one protrusion along a second axis perpendicular to the first axis according to the adjustment signal. The main shaft is rotated around the universal joint until perpendicular to the reference plane with the projected plane parallel thereto.

    Abstract translation: 一个等级。 通过可旋转地发光的光源基本上平行于参考平面生成投影平面。 具有旋转部分和一对突起并连接到光源的主轴垂直于投影平面。 万向接头设置在主轴可旋转地穿过其中的壳体中。 水平传感器检测投影平面偏离参考平面的倾斜度并输出调整信号。 调节机构具有彼此交叉的第一可动构件和第二可动构件。 第一可动构件沿着第一轴推动一个突起,并且第二可动构件根据调整信号沿垂直于第一轴的第二轴推动一个突起。 主轴绕万向节旋转,直到垂直于参考平面,其中投影平面与其平行。

    Level
    34.
    发明授权
    Level 失效
    水平

    公开(公告)号:US06906310B1

    公开(公告)日:2005-06-14

    申请号:US10899329

    申请日:2004-07-26

    CPC classification number: G01C15/004

    Abstract: A level. A projected plane is generated substantially parallel to a reference plane by a light source rotatably emitting light. A main shaft, having a rotary portion and a pair of protrusions and connecting to the light source, is perpendicular to the projected plane. A universal joint is disposed in a housing with the main shaft rotatably passing therethrough. A level sensor detects inclination of the projected plane deviated from the reference plane and outputs an adjustment signal. An adjustment mechanism has a first movable member and a second movable member crossing each other. The first movable member impels one protrusion along a first axis, and the second movable member impels one protrusion along a second axis perpendicular to the first axis according to the adjustment signal. The main shaft is rotated around the universal joint until perpendicular to the reference plane with the projected plane parallel thereto.

    Abstract translation: 一个等级。 通过可旋转地发光的光源基本上平行于参考平面生成投影平面。 具有旋转部分和一对突起并连接到光源的主轴垂直于投影平面。 万向接头设置在主轴可旋转地穿过其中的壳体中。 水平传感器检测投影平面偏离参考平面的倾斜度并输出调整信号。 调节机构具有彼此交叉的第一可动构件和第二可动构件。 第一可动构件沿着第一轴推动一个突起,并且第二可动构件根据调整信号沿垂直于第一轴的第二轴推动一个突起。 主轴绕万向节旋转,直到垂直于参考平面,其中投影平面与其平行。

    Method for power sharing and controlling the status of a display wall
    36.
    发明授权
    Method for power sharing and controlling the status of a display wall 有权
    功率共享和控制显示墙状态的方法

    公开(公告)号:US08902127B2

    公开(公告)日:2014-12-02

    申请号:US12213041

    申请日:2008-06-13

    Abstract: Described is a method for power sharing of a display wall, in particular of a LED display wall having a plurality of display modules, and a plurality of N power supply units, each for driving a number of display modules, whereby during a failure of a first power supply unit of the plurality of N power supply units, the outputs of other power supply units are linked together such that the module or modules driven by the first and failed power supply continue(s) to operate, by redistribution of power from the other power supply units. Power sharing is also described in the context of a method for controlling the status of a display wall, in particular of a LED display wall, controlled by a central unit. The method includes collecting status and/or diagnostic information of the display wall inputted to the central unit; converting the status and/or diagnostic information to a picture; and displaying the picture on the display wall.

    Abstract translation: 描述了一种用于显示墙的功率共享的方法,特别是具有多个显示模块的LED显示墙和多个N个电源单元的功率共享的方法,每个用于驱动多个显示模块,由此在一个 多个N个电源单元的第一电源单元,其他电源单元的输出被连接在一起,使得由第一和故障电源驱动的模块或模块继续运行,通过从 其他电源单元。 在用于控制由中央单元控制的显示墙,特别是LED显示墙的状态的方法的上下文中也描述了功率共享。 该方法包括收集输入到中央单元的显示墙的状态和/或诊断信息; 将状态和/或诊断信息转换成图片; 并在显示墙上显示图像。

    Multi-antenna channel estimation method based on polyphase decomposition
    37.
    发明授权
    Multi-antenna channel estimation method based on polyphase decomposition 有权
    基于多相分解的多天线信道估计方法

    公开(公告)号:US08654879B2

    公开(公告)日:2014-02-18

    申请号:US13387308

    申请日:2010-11-02

    CPC classification number: H04L25/0204 H04B7/0413 H04L25/0232 H04L27/2647

    Abstract: A multi-antenna channel estimation method based on polyphase decomposition includes: receiving frequency domain received signals transformed using discrete fourier transformation (DFT) in pilot symbols; performing phase correction on the frequency domain received signals; performing polyphase decomposition on the frequency domain received signals which are corrected using phase correction and acquiring polyphase signals; performing interpolation on the polyphase signals and acquiring the estimation values of the multi-antenna channel parameters with various linear combinations on each frequency; acquiring decorrelation array based on the pilot structure of the transmission antenna and decorrelating the estimation values of the multi-antenna channel parameters with various linear combination on each frequency using the decorrelation array and acquiring channel parameters of the pilot symbols on each frequency; acquiring channel parameters of data symbols based on the channel parameters of the pilot symbols. With the present invention, the inversion problem in multi-antenna channel estimation is avoided with lower complexity, and results of the multi-antenna channel estimation method become more accurate since the DFT and filtering are performed in the interpolation after polyphase decomposition.

    Abstract translation: 基于多相分解的多天线信道估计方法包括:在导频符号中接收使用离散傅立叶变换(DFT)变换的频域接收信号; 对频域接收信号进行相位校正; 对使用相位校正和获取多相信号校正的频域接收信号执行多相分解; 对所述多相信号执行插值,并且在每个频率上以各种线性组合获取所述多天线信道参数的估计值; 基于发射天线的导频结构获取解相关阵列,并使用解相关阵列在每个频率上用各种线性组合去除多个天线信道参数的估计值,并获取每个频率上的导频符号的信道参数; 基于导频符号的信道参数获取数据符号的信道参数。 利用本发明,以更低的复杂度避免了多天线信道估计中的反转问题,并且由于在多相分解之后的内插中执行DFT和滤波,所以多天线信道估计方法的结果变得更加精确。

    TRANSFORMER CONTROL DEVICE AND METHOD BASED ON THREE-DIMENSIONAL ZONE DIAGRAM POLICY
    39.
    发明申请
    TRANSFORMER CONTROL DEVICE AND METHOD BASED ON THREE-DIMENSIONAL ZONE DIAGRAM POLICY 有权
    基于三维图形图的变压器控制装置和方法

    公开(公告)号:US20130076130A1

    公开(公告)日:2013-03-28

    申请号:US13414279

    申请日:2012-03-07

    CPC classification number: H02J3/16 H02J3/1878 H02P13/06 Y02E40/34 Y10T307/297

    Abstract: Disclosed is a transformer control device and method based on a three-dimensional zone diagram policy. The method includes: setting transformers, including a transformer A and a transformer B; collecting three-phase voltage data and three-phase current data in a power system; rectifying the collected three-phase voltage data and the three-phase current data; transferring the data to the latches in a time-transfer method; transferring the data to an A/D converter of a processor to convert analog signals to digital signals; constructing a three-dimensional zone diagram in the processor; determining transformer operating conditions according to positions of points formed by voltage, reactive power factor and substation load; and adjusting the transformers. This invention adopts a simple, easy and clear three-parameter control policy including voltage, power factors and substation loads, so as to simplify analysis of transformer operating conditions, realize optimal substation operation, reduce transformer loss, and increase economic benefits.

    Abstract translation: 公开了一种基于三维区域图策略的变压器控制装置和方法。 该方法包括:设置变压器,包括变压器A和变压器B; 在电力系统中收集三相电压数据和三相电流数据; 整流收集的三相电压数据和三相电流数据; 以时间传送方式将数据传送到锁存器; 将数据传送到处理器的A / D转换器,以将模拟信号转换为数字信号; 在处理器中构建三维区域图; 根据由电压,无功功率因数和变电站负载形成的点的位置确定变压器工作条件; 并调整变压器。 本发明采用简单,简单,明确的三参数控制策略,包括电压,功率因数和变电站负载,简化变压器运行状况分析,实现最佳变电站运行,减少变压器损耗,增加经济效益。

    Loudspeaker module
    40.
    发明授权
    Loudspeaker module 失效
    扬声器模块

    公开(公告)号:US08340337B2

    公开(公告)日:2012-12-25

    申请号:US12817194

    申请日:2010-06-17

    CPC classification number: H04R1/345 H04R1/403

    Abstract: A loudspeaker module includes a hollow main body, two rotatable connecting portions, and two loudspeakers. The hollow main body includes two opposite sidewalls. Each of the opposite sidewall defines a first opening, an inner sidewall of the first opening defines an annular rotating slot. One end of the connecting portion extends an annular flange shaped corresponding to the rotating slot. The two rotatable connecting portions are respectively rotatably connected to the main body via the flange rotating about the rotating slot. Two loudspeakers are disposed in an end of the corresponding rotatable connecting portion away from the main body.

    Abstract translation: 扬声器模块包括中空主体,两个可旋转连接部分和两个扬声器。 中空主体包括两个相对的侧壁。 每个相对的侧壁限定第一开口,第一开口的内侧壁限定环形旋转槽。 连接部分的一端延伸成对应于旋转槽形成的环形凸缘。 两个可旋转连接部分分别经由围绕旋转槽旋转的凸缘可旋转地连接到主体。 两个扬声器设置在远离主体的相应的可旋转连接部分的端部。

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