公开(公告)号：WO0020399A3

公开(公告)日：2000-07-27

申请号：PCT/EP9907125

申请日：1999-09-24

Applicant: BASF AG ,  GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D231/08 ,  C07D401/04 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

CPC classification number: C07D401/04 ,  C07D231/08 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

Abstract: The invention relates to the use of substituted 5-hydroxypyrazoles of formula (I) in which the substituents have the following meanings: B represents aryl or heteroaryl; A represents C=O, C=S or SO2; R represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, cycloalkyl, C3-C10-cycloalkenyl, cycloalkynyl, or aryl, heterocyclyl or heteroaryl; R represents hydrogen; R represents hydrogen, nitro, cyano, N(R')2, alkyl, alkyl halide, alkoxy, alkoxy halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, whereby R', independent of one another, represents hydrogen or alkyl; or R and R , together, represent a group =O, =S or =N-O-R , whereby R represents hydrogen, alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide; R represents hydrogen, halogen, nitro, cyano N(R')2, alkyl, alkyl halide, COOR', heteroaryl or heterocyclyl. The invention also relates to the use of said compounds for combating harmful fungi, to agents containing the compounds, to novel 5-hydroxypyrazoles and to methods for the production thereof.

Abstract translation: 本发明涉及式（I）的5-羟基吡唑啉的用途，其中取代基具有以下含义：B芳基或杂芳基; A C = O，C = S或SO 2; R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，C 3 -C 10 - 环烯基，环炔基或芳基，杂环基或杂芳基; R 2氢; [R <3>为氢，硝基，氰基，N（R '）2，烷基，卤代烷基，烷氧基，卤代烷氧基，链烯基，卤代烯基，炔基或卤代炔基，其中R' 独立地为氢或烷基; 或R <2>和R <3>一起表示基团= O，= S或= N-O-R <5>，其中R <5>是氢，烷基，卤代烷基，链烯基，卤代烯基，炔基或卤代炔基; R 4是氢，卤素，硝基，氰基，N（R'）2，烷基，卤代烷基，COOR'，杂芳基或杂环基; 用于控制有害真菌，含有它们的试剂和新的5-羟基吡唑及其制备方法。

公开(公告)号：WO2008012234A2

公开(公告)日：2008-01-31

申请号：PCT/EP2007057353

申请日：2007-07-17

Applicant: BASF AG ,  DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

Inventor： DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

IPC: C07D405/14 ,  A01N43/707 ,  C07D409/14

CPC classification number: C07D405/14 ,  A01N43/653 ,  C07D409/14

Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.

Abstract translation: 本发明涉及通式（I），其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素，CN，NO _{2 ，氨基，C <五 SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4卤代烷，C 1 -C 4 烷基氨基， ç 1 -C 4 二烷基氨基，硫代，或C 1 -C 4 是烷硫基，被取代的，和 各其他取代基A或B为苯基或5元或6元杂芳基，所述取代基任选地被1-3个下列取代基取代：卤素，CN，NO 2 ，氨基，C < SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 二烷基氨基，巯基或C 1 -C 4 - 烷硫基，被取代的，和它们的植物耐受的酸加成盐或金属盐，使用式（I）的用于控制植物病原真菌包含它们的化合物和试剂。}

公开(公告)号：WO2005113555A8

公开(公告)日：2006-12-14

申请号：PCT/EP2005005270

申请日：2005-05-13

Applicant: BASF AG ,  BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.

Abstract translation: 本发明涉及如下通式的新型三唑并嘧啶化合物I和它们在防治有害真菌中的用途，以及植物保护剂，这样的化合物作为活性成分enthalten.In式I，X，Y，L，M，Ar和A具有下列含义：X 卤素，氰基，C _{1 -C 4 烷基，C 1 -C 4 卤代烷基，C < SUB> 1 -C 4 - 烷氧基或C 1 -C 4 卤代烷氧基; Y是卤素，C 1 -C 4 烷基或C 1 -C 4 卤代烷基; 独立地为卤素，C 1 -C 6 烷基，C 2 -C 6 烯基，C 1 -C ç 6 卤代烷基，C 1 -C 6 烷氧基，C 1 -C 6 < / SUB>卤代烷氧基，硝基，氨基，NHR，NR 2 ，氰基，S（= O）名词 A“或C（= O）A ^{2 ; m是0，1，2，3或4; A是一个化学键或基团CR 4 - [R 5 是; Ar是苯基或5-或6-元杂芳基具有1个，选自O，S和N的杂原子作为环成员，其中苯基和杂芳基可以具有一个稠合的苯环和1，2，3 2或3 ，4或5个取代基R 一可以包括;. R“至R 3 具有权利要求1中给出的含义。}}

公开(公告)号：WO2006066818A3

公开(公告)日：2006-11-02

申请号：PCT/EP2005013577

申请日：2005-12-16

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D213/55 ,  C07D237/14 ,  C07D487/04

Abstract: The invention relates to novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds and the salts thereof that can be used in agriculture, the use of the same for controlling pathogenic fungi, and plant protection agents containing at least one such compound as an active constituent. Said novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds correspond to general formula (I) wherein the substituents R 1 , R 2 , Het, X and Y have the following designations: Het represents a six-membered heteroaromatic radical selected from pyridinyl, pyridazinyl, pyrazinyl, 1,2,4-triazinyl and 1,3,5-triazinyl, the six-membered heteroaromatic radical comprising 1, 2 or 3 substituents L which are the same or different, R 1 , R 2 independently represent hydrogen, C 1 -C 8 alkyl, C 1 -C 8 halogenalkyl, C 1 -C 8 alkoxy, C 3 -C 8 cycloalkyl, C 3 -C 8 cycloalkoxy, C 5 -C 10 bicycloalkyl, C 3 -C 8 halogencycloalkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkenyloxy, C 4 -C 10 alkadienyl, C 2 -C 8 halogenalkenyl, C 3 -C 8 cycloalkenyl, C 3 -C 8 halogencycloalkenyl, C 2 -C 8 alkinyl, C 2 -C 8 alkinyloxy, C 2 -C 8 halogenalkinyl, NH 2, C 1 -C 8 alkylamino, Di-C 1 -C 8 -alkylamino, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle, X represents hydrogen, halogen, OH, cyano, C 1 -C 4 alkyl and the like, and Y represents hydrogen, halogen, cyano, C 1 -C 4 alkyl, and the like.

Abstract translation: 本发明涉及新颖的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物及其农业上可接受的盐，以及它们在防治有害真菌中的用途，以及植物保护剂，这些化合物的至少一种作为 含有活性成分。 新的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物可通过通式（I）所示，其中取代基R ^{1 来表示 ，R 2 ，（I）的Het，X和Y在式具有以下含义：Het是其选自吡啶基，哒嗪基，吡嗪基的6元杂芳基，1,2,4- 三嗪基和1,3,5-三嗪基，其中所述6元杂芳基1，2或3个相同或不同的取代基L可以包括，R 1 ，R 2 独立地 另一个氢，C _{1 -C 8 烷基，C 1 -C 8 卤代烷基，C 1 -C 8 烷氧基，C 3 -C 8 环烷基，C 3 -C 8 环烷氧基，C 5 -C 10 双环，C 3 -C 8 卤代环烷基，C 2 -C 8 烯基，C 2 -C 8 烯 ，C 4 -C 10 链二烯基，C 2 -C 8 卤代，C 3 -C 8 环烯基，C 3 -C 8 卤代环，C 2 -C 8 炔基，C 2 -C 8 炔氧基，C 2 -C 8 卤代炔基，NH 2 C 1 -C 8 烷基氨基，二-C 1 -C 8 烷基氨基，苯基，萘基或五 - 或六元饱和，部分不饱和或芳族的杂环，X是氢，卤素，OH，氰基，C < SUB> 1 -C 4 烷基等，Y是氢，卤素，氰基，C 1 -C 4 烷基， 等等。}}

公开(公告)号：WO2005121146A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005006171

申请日：2005-06-08

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/647 ,  A01N43/90 ,  C07D487/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to triazolopyrimidines of formula (I), wherein the index n and the substituents R, R

Abstract translation: 本发明涉及下式的三唑并嘧啶I，其中索引n和取代基R，R

公开(公告)号：WO2005110089A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005005069

申请日：2005-05-11

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  GEWEHR MARKUS

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  GEWEHR MARKUS

IPC: A01N43/90 ,  A01N43

CPC classification number: A01N43/90 ,  A01N43/78 ,  A01N43/56 ,  A01N43/32 ,  A01N43/08 ,  A01N2300/00

Abstract: The inventive fungicide mixtures contain as active components 1) a triazolopyrimidine derivative of formula (I) and at least on type of biphenyl amide of formula (II) wherein variables have the following designations: A is oxathiin- or 5-membered heteroaryl containing one or four nitrogen atoms and/or three nitrogen atoms and/or one sulphur or oxygen atom, wherein A is substitutable according to the description, R1 is hydrogen, alkyl, alkylcarbonyl or a carbonyl bonded group A, Ra and Rb are halogen, cyano, alkyl, halogenalkyl, alkoxycarbonyl, alkoxy, halogenalkoxy, alkylthio, alkylcarbonyl, formyl, alkylene- or alkenylene which connects two adjacent carbon atoms, m is 0, 1, 2, 3, 4 or 5, n is 0, 1 or 2, wherein the fungicide mixtures contain said components in the synergistically effective amount. A method for controlling pathogenic fungi using the mixtures of the compounds (I) and (II), the use of the compounds (I) and (II) for producing such mixtures and mixture-containing agents are also disclosed.

Abstract translation: 一种杀真菌混合物，其包含作为活性组分1）式I的三唑并嘧啶衍生物，以及2）至少将式II的一个biphenylamide：其中各变量具有以下含义：甲Oxathiin-或5元杂芳基，含有一至四个氮原子或1至 三个氮原子和/或一个硫或氧原子，其中一个可根据描述被取代; R1是氢，烷基，烷基羰基或基团A通过羰基连接; RA，RB是卤素，氰基，烷基，卤代烷基，烷氧基羰基，烷氧基，卤代烷氧基，烷硫基，烷基羰基，甲酰基，亚烷基或亚烯基，其连接两个相邻碳原子; 米0，1，2，3，4或5; n为0，1或2; 在协同有效量，用于控制使用I化合物的混合物与化合物II和使用I化合物与用于制备这样的混合物和包含这些混合物的组合物的化合物（II）的有害真菌的方法。

公开(公告)号：WO2004045283A8

公开(公告)日：2005-06-02

申请号：PCT/EP0312776

申请日：2003-11-14

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90

CPC classification number: A01N43/90 ,  A01N37/50 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures for controlling rice pathogens, said mixtures containing 1) the compound of formula (I), and 2) the compound of formula (II), as active constituents in a synergistically effective quantity. The invention also relates to methods for controlling pathogenic fungi using mixtures containing compound (I) and compound (II), to the use of compounds (I) and (II) for producing such mixtures, and to agents containing said mixtures.

Abstract translation: 用于控制水稻病原体，其包含作为活性成分的杀真菌混合物：1）式（I的化合物），和2）式的化合物（II），协同有效量，用于控制使用化合物的混合物防治有害真菌的方法（I ）与化合物（II），使用的化合物的（I）和（II）一种制造这样的混合物和包含这些混合物的组合物。

公开(公告)号：WO2005010000A3

公开(公告)日：2005-05-19

申请号：PCT/EP2004007924

申请日：2004-07-15

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  C07D471/04

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R ; n stands for 1, 2, 3, 4 or 5; R represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R , and R represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

Abstract translation: 本发明涉及通式I的双环化合物，其中X，Y彼此独立地是N或C-R 4; n是1,2,3,4或5; ř表示卤素，氰基，C1-C6烷基，C1-C6烷氧基，C1-C6卤代烷基，C1-C6卤代烷氧基，C2-C6链烯基，C2-C6链烯氧基或C （O）R 5代表; [R <1>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8-环烷基，其任选被烷基和/或卤素取代的或者 多取代，C5-C8环烯基，其任选与乘法烷基和/或卤素或单 - ，或<6>，SR <6>或NR <7> - [R <8>取代; [R <2>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8环烷基，任选地被烷基和/或卤素单取代的 或多取代的，C5-C8环烯基，其任选地被烷基和/或卤素取代基取代一次或多次，或<6>，SR <6>或NR <7> - [R <8>; R 3是任选被烷基和/或卤素单取代或多取代的氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; 和化合物（I），植物保护剂的农业上可接受的盐，其包含通式（I）和/或（I）的农业上可接受的盐和至少一种液体或固体载体和用于防治植物病原性有害真菌的方法中的至少一种化合物。

公开(公告)号：WO2004045283A3

公开(公告)日：2004-07-29

申请号：PCT/EP0312776

申请日：2003-11-14

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90

CPC classification number: A01N43/90 ,  A01N37/50 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures for controlling rice pathogens, said mixtures containing 1) the compound of formula (I), and 2) the compound of formula (II), as active constituents in a synergistically effective quantity. The invention also relates to methods for controlling pathogenic fungi using mixtures containing compound (I) and compound (II), to the use of compounds (I) and (II) for producing such mixtures, and to agents containing said mixtures.

Abstract translation: 用于控制水稻病原体，其包含作为活性成分的杀真菌混合物：1）式（I的化合物），和2）式的化合物（II），协同有效量，用于控制使用化合物的混合物防治有害真菌的方法（I ）与化合物（II），使用的化合物的（I）和（II）一种制造这样的混合物和包含这些混合物的组合物。

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。