公开(公告)号：EP1080089B1

公开(公告)日：2003-11-05

申请号：EP99924925.3

申请日：1999-05-10

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  LANGEMANN, Klaus ,  VON DEYN, Wolfgang ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  ENGEL, Stefan ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WAGNER, Oliver ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D409/06 ,  C07D409/14 ,  A01N43/56

CPC classification number: C07D409/06 ,  A01N43/56 ,  C07D409/14 ,  C07F9/65586

Abstract: The invention relates to pyrazolyldioxothiochromanoyl derivatives of formula (I) in which the variables have the following meanings: X represents oxygen, sulfur, S=O, S(=O)2, CR4R5, C=O or C=NR6; R1 hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl thio, alkyl thio halide, alkyl sulfinyl, alkyl sulfinyl halide, alkyl sulfonyl, alkyl sulfonyl halide, optionally substituted amino sulfonyl or optionally substituted sulfonyl amino; R2 represents alkyl, alkyl halide, alkoxy or alkoxy halide; R3 represents hydrogen, alkyl or halogen; R4, R5 represent hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl thio, alkyl thio halide, alkyl sulfinyl, alkyl sulfinyl halide, alkyl sulfonyl, alkyl sulfonyl halide or optionally substituted amino; or R?4 and R5¿ jointly construct a chain which can be substituted and/or discontinued by oxygen or sulfur; or an optionally substituted methylidene group; l represents 0 to 4; and R7 represents substituted pyrazole-4-yl-carbonyl or substituted pyrazole-4-yl-methylidene. The invention also relates to the salts of said derivatives which can be used for agricultural purposes, to a method for producing the pyrazolyldioxothiochromanoyl derivatives, to agents containing the same, and to the use of these derivatives or agents containing the same for controlling undesirable plants.

Abstract translation: 本发明涉及式（I）的吡唑基二氧代二氢苯并噻喃酰基衍生物，其中变量具有以下含义：X代表氧，硫，S = O，S（= O）2，CR4R5，C = O或C = NR6; 卤素，氰基，烷基，烷基卤，烷氧基，烷氧基卤化物，烷基硫基，烷基硫代卤化物，烷基亚磺酰基，烷基亚磺酰卤，烷基磺酰基，烷基磺酰卤，任选取代的氨基磺酰基或任选取代的磺酰基氨基; R2表示烷基，烷基卤，烷氧基或烷氧基卤化物; R3代表氢，烷基或卤素; 硝基，卤素，氰基，烷基，烷基卤，烷氧基，烷氧基卤，烷基硫基，烷基硫代卤化物，烷基亚磺酰基，烷基亚磺酰卤，烷基磺酰基，烷基磺酰卤或任选取代的氨基; 或R 4和R 5'共同构成可被氧或硫取代和/或中断的链; 或任选取代的亚甲基; l表示0至4; 并且R 7代表取代的吡唑-4-基 - 羰基或取代的吡唑-4-基 - 亚甲基。 本发明还涉及可用于农业目的的所述衍生物的盐，制备吡唑基二氧代二氢苯并噻喃酰基衍生物的方法，含有它们的试剂，以及这些衍生物或含有它们的试剂用于防治不希望的植物的用途。

公开(公告)号：EP1240163A1

公开(公告)日：2002-09-18

申请号：EP00991216.3

申请日：2000-12-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MAYER, Guido ,  MI LITZ, Ulf ,  NEIDLEIN, Ulf ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  WITSCHEL, Matthias

IPC: C07D413/00 ,  C07D413/14 ,  A01N43/80

CPC classification number: C07D409/14 ,  A01N43/80 ,  C07D413/10

Abstract: The invention relates to 3-(4,5-dihydroisoxazole-5-yl)benzoylpyrazole of the formula (I), wherein the variables have the following meanings: R1, R2 represent hydrogen, nitro, halogen, cyano, alkyl, halogenalkyl, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl or halogenalkylsulfonyl; hydrogen, R¿3? represents halogen or alkyl; R?4¿ represents hydrogen or alkyl; R5, R6 represent hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, wherein the latter six groups can be substituted; R7 represents halogen, cyano, hydroxy, alkyl, halogenalkyl, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, amino, alkylamino, dialkylamino, dialkoxymethyl, hydroxyiminoalkyl, alkoxyiminoalkyl or optionally substituted carbonyl; R11 represents optionally substituted pyrazole that is bound in the 4 position and that carries a hydroxy group or a derivative thereof in the 5 position. The invention also relates to the agriculturally useful salts thereof, to methods and to intermediate products for preparing the 3-(4,5-dihydroisoxazole-5-yl)benzoylpyrazole, to agents containing them and to the use of said derivatives or the agents containing them for combatting undesired plants.

公开(公告)号：EP1194407A2

公开(公告)日：2002-04-10

申请号：EP00945814.2

申请日：2000-06-23

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： NEIDLEIN, Ulf ,  GÖTZ, Norbert ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  GÖTZ, Roland ,  LANGEMANN, Klaus ,  MAYER, Guido ,  MISSLITZ, Ulf ,  WITSCHEL, Matthias ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D231/20 ,  A01N43/56

CPC classification number: A01N43/56 ,  C07D231/20

Abstract: The invention relates to cycloalkyl-substituted benzoyl pyrazoles of formula (I) wherein said variables can, for example, have the following meanings: R1 = hydrogen, nitro, halogen, cyano, rhodano or an optionally substituted aliphatic radical; R2 = an optionally substituted aliphatic radical, halogen, nitro, in addition to substituted sulfonyl or amino groups; R3 = hydrogen, halogen, C¿1-C?6-alkyl, C¿1?-C6-halogenalkyl, C1-C6-alkoxy, C2-C6-alkenyl or C2-C?6¿-alkinyl; R4, R5 = hydrogen, nitro, halogen, cyano, rhodano, an optionally substituted aliphatic radical or substituted sulfonyl or amino groups; R6 = hydrogen, halogen, C¿1?-c6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkyl; R?7¿ = a cyclic ring system with 3 - 14 ring atoms; R16 = hydroxy or a substituted hydroxy group; in addition to tautomers or agriculturally useful salts thereof. The invention also relates to methods for the production of compounds of formula (I), agents containing said compounds, the use of compounds of formula (I) and agents containing said compounds as herbicides.

公开(公告)号：EP1181295A2

公开(公告)日：2002-02-27

申请号：EP00940273.6

申请日：2000-05-26

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  BAUMANN, Ernst ,  DEYN, Wolfgang von ,  MAYER, Guido ,  MISSLITZ, Ulf ,  NEIDLEIN, Ulf ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D495/04 ,  C07D498/04 ,  A01N43/90

CPC classification number: C07D495/04

Abstract: The invention relates to tricyclic benzoylcyclohexanedione derivatives of formula (I), wherein the variables have the following meanings: X is oxygen, sulphur, S=O, S(=O)2, CR?6R7, NR8¿ or a bond; y forms a saturated, partially saturated or unsaturated 5- or 6-membered heterocycle with the two carbons to which it is bonded; R?1, R2, R6, R7¿ is hydrogen, alkyl, alkyl halide, alkoxy or alkoxy halide; R3 is halogen, alkyl, alkyl halide, alkoxy or alkoxy halide; R4 is hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, C¿1?-C6- alkylthio halide, alkylsulfinyl, alkylsulfinyl halide, alkylsulfonyl, alkylsulfonyl halide, optionally substituted aminosulfonyl, or optionally substituted sulfonylamino; R?5¿ is hydrogen, alkyl or halogen; m is 0, 1 or 2; R8 is hydrogen, alkyl, alkyl halide, alkylcarbonyl, formyl, alkoxycarbonyl, alkoxycarbonyl halide, alkylsulfonyl or alkylsulfonyl halide; and R9 is substituted (3-oxo-1-cyclohexen-2-yl)-carbonyl or substituted (1,3-dioxo-2-cyclohexyl)-methylidene; and to agriculturally useable salts thereof. The invention also relates to a method for producing the tricyclic benzoylcyclohexanedione derivatives, to products containing them and to the use of said derivatives or said products containing them for combating unwanted vegetation.

Abstract translation: 本发明涉及式（I）的三环苯甲酰基环己二酮衍生物，其中各变量具有以下含义：X是氧，硫，S = O，S（= O）2，CR 6 R 7，NR 8或键; y与其所键合的两个碳形成饱和的，部分饱和或不饱和的5-或6-元杂环; R 1，R 2，R 6，R 7是氢，烷​​基，烷基卤，烷氧基或烷氧基卤化物; R3是卤素，烷基，烷基卤，烷氧基或烷氧基卤化物; 卤素，氰基，烷基，烷基卤，烷氧基，烷氧基卤，烷硫基，C1-C6烷硫基卤，烷基亚磺酰基，烷基亚磺酰卤，烷基磺酰基，烷基磺酰卤，任选取代的氨基磺酰基或任选取代的磺酰氨基 ; R 5是氢，烷基或卤素; m是0,1或2; R8为氢，烷基，烷基卤，烷基羰基，甲酰基，烷氧基羰基，烷氧基羰基卤，烷基磺酰基或烷基磺酰卤; （3-氧代-1-环己烯-2-基） - 羰基或取代的（1,3-二氧代-2-环己基） - 亚甲基; R 9为取代的（3-氧代-1-环己烯-2-基） 并涉及其可农用盐。 本发明还涉及生产三环苯甲酰基环己二酮衍生物的方法，含有它们的产品以及所述衍生物或含有它们的所述产品用于防治不想要的植物的用途。

公开(公告)号：EP1163240A1

公开(公告)日：2001-12-19

申请号：EP00915171.3

申请日：2000-03-08

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  MAYER, Guido ,  MISSLITZ, Ulf ,  NEIDLEIN, Ulf ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D413/06 ,  C07D498/04 ,  C07D495/04 ,  C07D491/04 ,  A01N43/90 ,  A01N43/80 ,  C07D261/20

CPC classification number: C07D413/06 ,  A01N43/80 ,  A01N43/90 ,  C07D491/04 ,  C07D495/04

Abstract: The invention relates to tricyclic benzoylpyrazole derivatives of formula (I), wherein the variables have the following meanings: X is oxygen or sulphur, S=O, S(=O)2, CR?6R7, NR8¿ or a bond; Y, together with the two other carbons to which it is bonded, forms a saturated, partially saturated or unsaturated 5 or 6-membered heterocycle; R?1, R2, R6, R7¿ are hydrogen, alkyl, alkyl halide, alkoxy or halogenalkoxy; R3 is halogen, alkyl, alkyl halide, alkoxy or halogenalkoxy; R4 is hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogen alkylthio, alkylsulfinyl, alkylsulfinyl halide, alkylsulfonyl, alkylsulfonyl halide, optionally substituted aminosulfonyl or optionally substituted sulfonylamino; R5 is hydrogen, alkyl or halogen; l is 0, 1 or 2; R8 is hydrogen, alkyl, alkyl halide, alkylcarbonyl, formyl, alkoxycarbonyl, alkoxycarbonyl halide, alkylsulfonyl or alkylsulfonyl halide and R9 is substituted pyrazole-4-yl-carbonyl or substituted 5-oxo-pyrazolin-4-yl-methylides; and the agriculturally useable salts thereof. The invention also relates to a method and intermediate products for producing tricyclic benzoylpyrazole derivatives, to products which contain the same and to the use of said derivatives or said products for combating undesirable plants.

公开(公告)号：EP1112256A1

公开(公告)日：2001-07-04

申请号：EP99944541.4

申请日：1999-08-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  LANGEMANN, Klaus ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  GÖTZ, Roland ,  GÖTZ, Norbert ,  RACK, Michael ,  ENGEL, Stefan ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D215/18 ,  A01N43/42 ,  C07D215/14 ,  C07D215/36 ,  C07D405/12 ,  C07D401/08 ,  C07D401/06 ,  C07F9/60

CPC classification number: C07D401/06 ,  A01N43/42 ,  C07D215/14 ,  C07D215/18 ,  C07D215/36 ,  C07D401/08 ,  C07D405/12 ,  C07F9/60

Abstract: The invention relates to cyclohexenonquinolinoyl derivatives of formula (I), wherein the variables have the following meanings: R1 means hydrogen, nitro, halogen, cyano, alkyl, halogenalkyl, alkoxyiminomethyl, alkoxy, halogenalkoxy, alkylthio, C1-C6-halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, optionally substituted aminosulfonyl, optionally substituted sulfonylamino, optionally substituted phenoxy, optionally substituted heterocyclyloxy, optionally substituted phenylthio or optionally substited heterocyclylthio; R2, R3 mean hydrogen, alkyl, halogenalkyl or halogen; and R4 means substituted (3-oxo-1-cyclohexen-2-yl)-carbonyl or substituted (1,3-dioxo-2-cyclohexyl)-methylidene. The invention also relates to the agriculturally useable salts of said derivatives, to a method for producing the derivatives, to agents containing them and to the use of the derivatives or agents containing them for combating undesirable plants.

公开(公告)号：EP1084116A1

公开(公告)日：2001-03-21

申请号：EP99923435.4

申请日：1999-04-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  LANGEMANN, Klaus ,  VON DEYN, Wolfgang ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  ENGEL, Stefan ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WAGNER, Oliver ,  GÖTZ, Roland ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D335/06 ,  C07D339/08 ,  C07D409/08 ,  A01N43/18 ,  A01N43/32

CPC classification number: C07D335/06 ,  A01N43/08 ,  A01N43/18 ,  A01N43/36 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/80 ,  A01N43/84 ,  C07D339/08 ,  C07D409/08

Abstract: The invention relates to cyclohexenondioxothiochromanoyl derivatives of formula (I) wherein the variables have the following meanings: X is oxygen, sulphur, S=O, S(=O)2, CR4R5, C=O or C=NR6; R1 is hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, optionally substituted aminosulfonyl or optionally substituted sulfonylamino; R2 is alkyl, alkyl halide, alkoxy or halogenalkoxy; R3 is hydrogen, alkyl or halogen; and R4, R5 are hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl or substituted amino; or R?4 and R5¿ together form a chain which can be substituted and/or interrupted by oxygen or sulphur; or an optionally substituted methylide group; l is 0 to 4; R7 is substituted (3-oxo-1-cyclohexen-2-yl)-carbonyl or substituted (1,3-dioxo-2-cyclohexyl-methylides. The invention also relates to the agriculturally usable salts of said derivatives, to methods for producing the derivatives, to substances containing them, and to the use of the derivatives or substances containing them for combating undesirable plants.

Abstract translation: （I）的环己烯酮二氧代二氢苯并噻喃酰基衍生物，其中各变量具有以下含义： 卤素，烷基，烷基卤，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基，任选取代的氨基磺酰基或任选取代的磺酰基氨基; R2是烷基，烷基卤，烷氧基或卤代烷氧基; R3是氢，烷基或卤素; 硝基，卤素，氰基，烷基，烷基卤，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基或取代的氨基; 或R 4和R 5'一起形成可被氧或硫取代和/或插入的链; 或任选取代的甲基基团; l是0到4; R7是取代的（3-氧代-1-环己烯-2-基） - 羰基或取代的（1,3-二氧代-2-环己基 - 甲基化物）。本发明还涉及所述衍生物的农业上可使用的盐， 衍生物，含有它们的物质，以及使用衍生物或含有它们的物质来对付不需要的植物。