公开(公告)号：EP2602261A1

公开(公告)日：2013-06-12

申请号：EP11814640.6

申请日：2011-08-02

Applicant: Stella Pharma Corporation ,  Osaka Prefecture University Public Corporation

Inventor： KIRIHATA,Mitsunori ,  HATTORI,Yoshihide ,  UEHARA,Kohki ,  TAKENAKA,Hiroshi

IPC: C07F5/02

CPC classification number: C07F5/05 ,  C07F5/02 ,  C07F5/027

Abstract: The purpose of the present invention is to provide a novel boron-containing compound utilizable in BNCT and so on and a process for preparing same. According to the process, a boron compounds having an amino acid skeleton containing cyclo-type rings or a pharmaceutically acceptable salt thereof is prepared, said boron compound being represented by general formula (I)[wherein l is an integer of 1 to 6; m is 0, 1, or 2; and n is 0, 1 or 2].

Abstract translation: 本发明的目的是提供一种可用于BNCT等的新型含硼化合物及其制备方法。 根据该方法，制备具有含有环型环的氨基酸骨架的硼化合物或其药学上可接受的盐，所述硼化合物由通式（I）表示[其中l为1至6的整数; m为0,1或2; 和n为0,1或2]。