NOVEL ANTIMICROBIALS
    61.
    发明申请
    NOVEL ANTIMICROBIALS 审中-公开
    新的抗微生物剂

    公开(公告)号:WO2010058423A2

    公开(公告)日:2010-05-27

    申请号:PCT/IN2009000658

    申请日:2009-11-18

    Abstract: The present invention relates to novel phenyl oxazolidinone compounds of formula I, their pharmaceutically acceptable analogs, tautomeric forms, stereoisomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The invention also relates to the processes for the synthesis of novel compounds of formula I or their pharmaceutically acceptable analogs, tautomeric forms, stereoisomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The present invention also provides pharmaceutical compositions comprising novel compounds of formula I and methods of using them. The compounds of the present invention are useful as antimicrobial agents, effective against a number of aerobic and/or anaerobic Gram positive and/or Gram negative pathogens such as multi drug resistant species of Staphylococcus, Streptococcus, Enterococcus, Bacterioides, Clostridia, H. influenza, Moraxella, acid-fast organisms such as Mycobacterium tuberculosis as well as Linezolid resistant species of Staphylococcus and Enterococcus.

    Abstract translation: 本发明涉及式I的新型苯基恶唑烷酮化合物,其药学上可接受的类似物,互变异构形式,立体异构体,多晶型物,前药,代谢物,盐或溶剂化物。 本发明还涉及合成式I的新化合物或其药学上可接受的类似物,互变异构形式,立体异构体,多晶型物,前药,代谢物,盐或溶剂合物的方法。 本发明还提供了包含新型式I化合物和使用它们的方法的药物组合物。 本发明化合物可用作抗微生物剂,有效对抗许多需氧和/或厌氧革兰氏阳性和/或革兰氏阴性病原体,例如葡萄球菌,链球菌,肠球菌,细菌,梭菌,流感嗜血菌 ,莫拉菌属(Moraxella),耐酸生物体如结核分枝杆菌(Mycobacterium tuberculosis)以及耐利奈唑胺菌(Staphylococcus and Enterococcus)。

    VARIABLE-SPEED-DRIVE SYSTEM FOR A GRID BLOWER
    62.
    发明申请
    VARIABLE-SPEED-DRIVE SYSTEM FOR A GRID BLOWER 审中-公开
    变速驱动系统

    公开(公告)号:WO2009148766A2

    公开(公告)日:2009-12-10

    申请号:PCT/US2009/043421

    申请日:2009-05-11

    CPC classification number: B61C5/02 B60L1/003 B60L7/02 B60L7/10 B60L2200/26

    Abstract: A drive system for a grid blower of a vehicle is provided. The system includes: an electrical bus, a grid of resistive elements connected to the electrical bus, the grid of resistive elements configured to thermally dissipate electrical power generated from braking of the vehicle, the electrical power being transmitted on the electrical bus to the grid of resistive elements, an electrical power modulation device configured to modify electrical power received from at least one of the electrical bus and the grid of resistive elements, and a grid blower motor coupled to an output of the electrical power modulation device, wherein a speed of the grid blower motor varies based on the electrical power that has been modified by the electrical power modulation device.

    Abstract translation: 提供了一种用于车辆的电网鼓风机的驱动系统。 该系统包括:电气总线,连接到电气总线的电阻元件格栅,电阻元件格栅被配置为热散发由车辆制动产生的电力,电力在电气总线上传输到电网 电力元件,被配置为修改从电气总线和电阻元件网格中的至少一个接收的电力的电力调制装置,以及耦合到电力调制装置的输出的电网鼓风电动机,其中, 电网鼓风电机根据电力调制装置修改的电功率而变化。

    NOVEL HETEROCYCLIC COMPOUNDS
    64.
    发明申请
    NOVEL HETEROCYCLIC COMPOUNDS 审中-公开
    新型杂环化合物

    公开(公告)号:WO2009093269A1

    公开(公告)日:2009-07-30

    申请号:PCT/IN2009000061

    申请日:2009-01-23

    CPC classification number: C07D243/14 C07D403/06 C07D413/12 C07D487/04

    Abstract: The present invention relates to novel compounds of Formula I, their pharmaceutically acceptable derivatives, tautomeric forms, stereoisomers including R and S isomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The invention also relates to the processes for the synthesis of novel compounds of Formula I, their pharmaceutically acceptable derivatives, tautomeric forms, stereoisomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The present invention also provides pharmaceutical compositions comprising compounds of Formula I and methods of treating or preventing one or more conditions that may be regulated or normalized via inhibition of dipeptidyl peptidase IV (DPP-IV). Formula I

    Abstract translation: 本发明涉及式I的新化合物,其药学上可接受的衍生物,互变异构形式,包括R和S异构体在内的立体异构体,多晶型物,前药,代谢物,盐或溶剂化物。 本发明还涉及用于合成式I的新化合物,其药学上可接受的衍生物,互变异构形式,立体异构体,多晶型物,前药,代谢物,盐或溶剂合物的方法。 本发明还提供了包含式I化合物的药物组合物以及治疗或预防一种或多种可通过抑制二肽基肽酶IV(DPP-IV)而调节或正常化的条件的方法。 公式I

    RECEIVER SIDE PROTECTION WITH RESOURCE FORWARDING IN SIDELINK

    公开(公告)号:WO2021208021A1

    公开(公告)日:2021-10-21

    申请号:PCT/CN2020/085145

    申请日:2020-04-16

    Abstract: Certain aspects of the present disclosure provide techniques for receiver side protection in sidelink communications. In certain aspects, a method performed by an apparatus generally includes obtaining, from a first user equipment (UE), first control information, which includes a first resource allocation information of one or more resources allocated for transmission by the first UE to the apparatus and an indication of a first cell associated with the first UE. The method generally includes obtaining, from a second UE, second control information, which generally includes a second resource allocation information of resources allocated for transmission by the second UE to the apparatus and an indication of a second cell associated with the second UE. The method generally includes determining, based on the first and second control information, potential interference from transmissions by the first UE and the second UE and taking one or more actions to mitigate the potential interference.

    NOVEL SGLT INHIBITORS
    70.
    发明申请
    NOVEL SGLT INHIBITORS 审中-公开
    新型SGLT抑制剂

    公开(公告)号:WO2013038429A2

    公开(公告)日:2013-03-21

    申请号:PCT/IN2012/000612

    申请日:2012-09-12

    CPC classification number: C07D309/10 C07D493/08 C07H7/04

    Abstract: The present invention relates to novel compounds of Formula (I), their pharmaceutically acceptable derivatives, tautomeric forms, isomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The invention also relates to the processes for the synthesis of novel compounds of Formula (I), their pharmaceutically acceptable derivatives, tautomeric forms, isomers, polymorphs, prodrugs, metabolites, salts or solvates thereof. The present invention also provides pharmaceutical compositions comprising novel compounds of Formula (I) and methods of treating or preventing one or more conditions or diseases that may be regulated or normalized via inhibition of Sodium Glucose Cotransporter-2 (SGLT-2).

    Abstract translation: 本发明涉及式(I)的新化合物,其药学上可接受的衍生物,互变异构形式,异构体,多晶型物,前药,代谢物,盐或溶剂合物。 本发明还涉及合成式(I)的新化合物,其药学上可接受的衍生物,互变异构形式,异构体,多晶型物,前药,代谢物,盐或溶剂合物的方法。 本发明还提供包含式(I)的新型化合物和治疗或预防可通过抑制葡萄糖转运蛋白-2(SGLT-2)调节或归一化的一种或多种病症或疾病的药物组合物。

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