公开(公告)号：EP1112256A1

公开(公告)日：2001-07-04

申请号：EP99944541.4

申请日：1999-08-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  LANGEMANN, Klaus ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  GÖTZ, Roland ,  GÖTZ, Norbert ,  RACK, Michael ,  ENGEL, Stefan ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D215/18 ,  A01N43/42 ,  C07D215/14 ,  C07D215/36 ,  C07D405/12 ,  C07D401/08 ,  C07D401/06 ,  C07F9/60

CPC classification number: C07D401/06 ,  A01N43/42 ,  C07D215/14 ,  C07D215/18 ,  C07D215/36 ,  C07D401/08 ,  C07D405/12 ,  C07F9/60

Abstract: The invention relates to cyclohexenonquinolinoyl derivatives of formula (I), wherein the variables have the following meanings: R1 means hydrogen, nitro, halogen, cyano, alkyl, halogenalkyl, alkoxyiminomethyl, alkoxy, halogenalkoxy, alkylthio, C1-C6-halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, optionally substituted aminosulfonyl, optionally substituted sulfonylamino, optionally substituted phenoxy, optionally substituted heterocyclyloxy, optionally substituted phenylthio or optionally substited heterocyclylthio; R2, R3 mean hydrogen, alkyl, halogenalkyl or halogen; and R4 means substituted (3-oxo-1-cyclohexen-2-yl)-carbonyl or substituted (1,3-dioxo-2-cyclohexyl)-methylidene. The invention also relates to the agriculturally useable salts of said derivatives, to a method for producing the derivatives, to agents containing them and to the use of the derivatives or agents containing them for combating undesirable plants.

公开(公告)号：EP1084116A1

公开(公告)日：2001-03-21

申请号：EP99923435.4

申请日：1999-04-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WITSCHEL, Matthias ,  LANGEMANN, Klaus ,  VON DEYN, Wolfgang ,  MISSLITZ, Ulf ,  BAUMANN, Ernst ,  ENGEL, Stefan ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WAGNER, Oliver ,  GÖTZ, Roland ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D335/06 ,  C07D339/08 ,  C07D409/08 ,  A01N43/18 ,  A01N43/32

CPC classification number: C07D335/06 ,  A01N43/08 ,  A01N43/18 ,  A01N43/36 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/80 ,  A01N43/84 ,  C07D339/08 ,  C07D409/08

Abstract: The invention relates to cyclohexenondioxothiochromanoyl derivatives of formula (I) wherein the variables have the following meanings: X is oxygen, sulphur, S=O, S(=O)2, CR4R5, C=O or C=NR6; R1 is hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, optionally substituted aminosulfonyl or optionally substituted sulfonylamino; R2 is alkyl, alkyl halide, alkoxy or halogenalkoxy; R3 is hydrogen, alkyl or halogen; and R4, R5 are hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkylthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl or substituted amino; or R?4 and R5¿ together form a chain which can be substituted and/or interrupted by oxygen or sulphur; or an optionally substituted methylide group; l is 0 to 4; R7 is substituted (3-oxo-1-cyclohexen-2-yl)-carbonyl or substituted (1,3-dioxo-2-cyclohexyl-methylides. The invention also relates to the agriculturally usable salts of said derivatives, to methods for producing the derivatives, to substances containing them, and to the use of the derivatives or substances containing them for combating undesirable plants.

Abstract translation: （I）的环己烯酮二氧代二氢苯并噻喃酰基衍生物，其中各变量具有以下含义： 卤素，烷基，烷基卤，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基，任选取代的氨基磺酰基或任选取代的磺酰基氨基; R2是烷基，烷基卤，烷氧基或卤代烷氧基; R3是氢，烷基或卤素; 硝基，卤素，氰基，烷基，烷基卤，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基或取代的氨基; 或R 4和R 5'一起形成可被氧或硫取代和/或插入的链; 或任选取代的甲基基团; l是0到4; R7是取代的（3-氧代-1-环己烯-2-基） - 羰基或取代的（1,3-二氧代-2-环己基 - 甲基化物）。本发明还涉及所述衍生物的农业上可使用的盐， 衍生物，含有它们的物质，以及使用衍生物或含有它们的物质来对付不需要的植物。

公开(公告)号：EP1077955A1

公开(公告)日：2001-02-28

申请号：EP99922160.9

申请日：1999-05-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： RHEINHEIMER, Joachim ,  VON DEYN, Wolfgang ,  GEBHARDT, Joachim ,  RACK, Michael ,  LOCHTMAN, Rene ,  GÖTZ, Norbert ,  KEIL, Michael ,  WITSCHEL, Matthias ,  HAGEN, Helmut ,  MISSLITZ, Ulf ,  BAUMANN, Ernst

IPC: C07D261/04 ,  C07D413/10 ,  C07C251/40 ,  C07C319/14

CPC classification number: C07C249/06 ,  C07C201/10 ,  C07C201/12 ,  C07C205/44 ,  C07C209/62 ,  C07C251/48 ,  C07C253/00 ,  C07C255/50 ,  C07C315/04 ,  C07C319/14 ,  C07D261/04 ,  C07D413/10 ,  C07C323/09 ,  C07C317/24 ,  C07C317/32 ,  C07C205/06 ,  C07C211/52

Abstract: The invention relates to a method for producing isoxazolene of the formula (I), where the substituents have the following meanings: R1 is hydrogen, C¿1?-C6 alkyl, R?2 is C¿1-C6 alkyl, R?3, R4, R5¿ are hydrogen, C¿1?-C6 alkyl or R?4 and R5¿ together form a linkage, R6 is a heterocyclic ring, and n is 0, 1 or 2. Said method comprises the production of an intermediate compound of the formula (VI) where R?1, R3, R4 and R5¿ have the meanings given above. This step is followed by halogenation, thiomethylation, oxidation and acylation to yield compounds of formula (I). The invention also relates to new intermediate products for producing compounds of formula (I) and new methods for producing the intermediate products.

公开(公告)号：EP1003730A1

公开(公告)日：2000-05-31

申请号：EP98943774.4

申请日：1998-07-23

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： ENGEL, Stefan ,  RHEINHEIMER, Joachim ,  BAUMANN, Ernst ,  von DEYN, Wolfgang ,  HILL, Regina, Luise ,  MAYER, Guido ,  MISSLITZ, Ulf ,  WAGNER, Oliver ,  WITSCHEL, Matthias ,  OTTEN, Martina ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07D261/04 ,  C07D307/58 ,  A01N43/80 ,  A01N43/08

CPC classification number: C07D307/58 ,  A01N43/80 ,  C07D261/04

Abstract: The invention relates to substituted 2-benzoyl-cyclohexane-1,3-diones of formula (I), wherein the substituents have the following meaning: R1, R2 stand for hydrogen, mercapto, nitro, halogen, cyano, rhodanine, C¿1?-C6-alkyl, C1-C6 halogen alkyl, C1-C6-alkoxy, C2-C6-alkenyl, C2-C6-alkinyl, -OR?3, -OCOR3¿, -OSO¿2R?3, -S(O)¿nR?3, SO2OR?3, -NR3SO¿2R?3 or -NR3COR3¿, wherein R3 can have different meanings; n represents 0, 1 or 2; Q stands for an optionally substituted two-position bonded chyclohexane-1,3-dion ring; X1 stands for a straight-chain or branched C¿1?-C6-alkylene, a C2-C6-alkenylene or a C2-C6-alkinylene chain, wherein the above-mentioned alkylene, alkenylene or alkinylene radicals can be partially halogenated and/or carry one to three of the following groups: -OR?4, -OCOR4¿, -OCONHR4 or -OSO¿2R?4; wherein R4 can have different meanings and the above-mentioned alkenylene radicals in which the double bond is located in the alpha, beta position with respect to the phenyle ring are excluded and in which Het is linked to the double bond in the beta position; Het represents a three to six-membered, partially or fully saturated heterocyclic group or a three to six-membered heteroaromatic group with up to three heteroatoms selected form the nitrogen, oxygen or sulfur group, wherein the above-mentioned heterocyclic or heteroaromatic group can be partially or totally halogenated and/or R5 can be substituted; wherein R5 can have different meanings. The invention further relates to the agricultural use of the salts of said compounds, to a method and to the intermediate products for the production of compounds of formula (I), to the agents contained in said compounds, to the use of the compounds of formula (I) and to the agents containing said compounds used in the control of harmful plants.

公开(公告)号：EP1001939A1

公开(公告)日：2000-05-24

申请号：EP98942612.7

申请日：1998-07-23

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： ENGEL, Stefan ,  RHEINHEIMER, Joachim ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  MAYER, Guido ,  MISSLITZ, Ulf ,  WAGNER, Oliver ,  WITSCHEL, Matthias ,  OTTEN, Martina ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07D231/20 ,  C07D401/12 ,  A01N43/56

CPC classification number: C07D231/12 ,  A01N43/56 ,  C07D231/20 ,  C07D233/56 ,  C07D249/08 ,  C07D401/12

Abstract: The invention relates to substituted 4-benzoyl-pyrazole of formula (I), in which the substituents have the meaning indicated in the description, the agriculturally usable salts thereof, the production and the intermediary products used for obtaining compounds of formula (I), agents containing said compounds, the use of formula (I), as well as agents containing said compounds for pest control.

公开(公告)号：EP0810998B1

公开(公告)日：2000-04-26

申请号：EP96902272.2

申请日：1996-02-14

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  ENGEL, Stefan ,  OTTEN, Martina ,  VOSSEN, Marcus ,  PLATH, Peter ,  RANG, Harald ,  HARREUS, Albrecht ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D261/08 ,  C07D277/30 ,  A01N43/80 ,  A01N43/78 ,  C07D333/24 ,  C07D307/54 ,  C07D275/02 ,  C07D213/57 ,  C07D263/32 ,  C07D277/66 ,  C07D231/12 ,  C07D215/12

CPC classification number: C07D207/327 ,  A01N43/78 ,  A01N43/80 ,  C07D213/57 ,  C07D213/647 ,  C07D213/70 ,  C07D213/74 ,  C07D215/12 ,  C07D231/12 ,  C07D231/14 ,  C07D235/18 ,  C07D239/26 ,  C07D239/38 ,  C07D249/08 ,  C07D261/08 ,  C07D261/18 ,  C07D263/32 ,  C07D271/06 ,  C07D271/107 ,  C07D275/02 ,  C07D277/30 ,  C07D277/32 ,  C07D277/34 ,  C07D277/36 ,  C07D277/66 ,  C07D279/06 ,  C07D285/08 ,  C07D285/125 ,  C07D307/54 ,  C07D317/30 ,  C07D319/06 ,  C07D333/24 ,  C07D333/28 ,  C07D339/06 ,  C07D339/08

Abstract: Phenyldiketone derivatives have the formula (I), in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy optionally substituted by 1 to 5 halogen atoms or C1-C4 alkoxy, halogen, cyano, nitro, a group -(Y)n-S(O)mR7 or a group -(Y)¿n-CO-R?8; Z is a 5 or 6 membered saturated or unsaturated heterocyclic rest that contains 1 to 3 heteroatoms selected from the group that includes oxygen, sulphur or nitrogen, optionally substituted by halogen, cyano, nitro, a group -CO-R8, C1-C4 alkyl, C1-C4 halogen alkyl, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 halogen alkylthio, di-C1-C4-alkylamino or an optionally substituted phenyl ring, and that forms a bicyclic system together with a condensed carbon cycle or a second condensed heterocycle; Y is O, NR9; n equals 0 or 1; m equals 0, 1 or 2; R7 is C1-C4 alkyl, C1-C4 halogen alkyl or NR?9R10; R8 is C¿1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy or NR?9R10; R9¿ is hydrogen or C¿1?-C4 alkyl; R?10 is C¿1-C4 alkyl; and R1 is cyclopropyl, 1-methylcyclopropyl, 1-methylthiocyclopropyl or tertiary butyl. Also disclosed are the salts of compounds (I) usually utilized in agriculture.

公开(公告)号：EP0783487B1

公开(公告)日：2000-02-09

申请号：EP95932774.3

申请日：1995-09-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： KAST, Jürgen ,  VOSSEN, Marcus ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  OTTEN, Martina ,  PLATH, Peter ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07C317/24 ,  C07C49/84 ,  C07C245/08 ,  C07D319/06 ,  C07D339/08 ,  A01N41/10 ,  A01N35/02 ,  A01N43/28 ,  A01N43/32

CPC classification number: A01N35/06 ,  A01N41/10 ,  C07C205/45 ,  C07C245/08 ,  C07C317/24 ,  C07C2601/16 ,  C07D317/14 ,  C07D319/06

公开(公告)号：EP0960100A1

公开(公告)日：1999-12-01

申请号：EP97954936.0

申请日：1997-12-19

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HILL, Regina, Luise ,  KARDORFF, Uwe ,  RACK, Michael ,  GÖTZ, Norbert ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  MAYER, Guido ,  OTTEN, Martina ,  REINHEIMER, Joachim ,  WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: A01N ,  C07D ,  C07D231 ,  A01N43 ,  C07D409

CPC classification number: A01N43/56 ,  C07D231/24

Abstract: The invention concerns 4-benzoyl-pyrazoles of formula (I), in which the variables have the following meanings: R1, R2 stand for hydrogen, nitro, halogen, cyano, rhodano, alkyl, halogen alkyl, alkoxyalkyl, alkenyl, alkinyl, -OR?5, -OCOR6¿, -OSO¿2R?6, -SH, -S(O)¿n?R?7, -SO¿2OR5, -SO2NR?5R8, -NR8SO¿2R?6 or -NR8COR6; R3¿ stands for hydrogen, cyano, alkyl, halogen alkyl, -OR?7, -SR7 or -NR7R10; R4¿ stands for hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkinyl, -COR9, -CO2R?9, -COSR9¿ or -CONR8R9; X stands for oxygen or NR8; n equals 0, 1 or 2; R5 stands for hydrogen, alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R6 stands for alkyl or halogen alkyl; R7 stands for alkyl, halogen alkyl, alkoxyalkyl, alkenyl or alkinyl; R8 stands for hydrogen or alkyl; R9 stands for alkyl, alkenyl, alkinyl, phenyl or benzyl; R10 stands for alkyl, halogen alkyl, alkenyl or alkinyl; Q stands for optionally substituted pyrazol linked in position 4. Also disclosed are the salts of these compounds useful in agriculture; processes and intermediate products for preparing the compounds of formula (I), agents containing the same and the use of these derivatives or agents containing the same for controlling undesirable plants.

Abstract translation: 本发明涉及式（I）的4-苯甲酰基 - 吡唑，其中各变量具有以下含义：R 1，R 2表示氢，硝基，卤素，氰基，rhodano，烷基，卤素烷基，烷氧基烷基，烯基，炔基， - OR 5，-OCOR 6，-OSO 2 R 6，-SH，-S（O）n R 7，-SO 2 OR 5，-SO 2 NR 5 R 8，-NR 8 SO 2 R 6或-NR 8 COR 6; R3代表氢，氰基，烷基，卤代烷基，-OR 7，-SR 7或-NR 7 R 10; R 4代表氢，任选取代的烷基，环烷基，烯基，环烯基，炔基，-COR 9，-CO 2 R 9，-COSR 9或-CONR 8 R 9; X代表氧或NR8; n等于0,1或2; R5代表氢，烷基，卤素烷基，烷氧基烷基，烯基或炔基; R6代表烷基或卤素烷基; R7代表烷基，卤代烷基，烷氧基烷基，烯基或炔基; R8代表氢或烷基; R9代表烷基，烯基，炔基，苯基或苄基; R10代表烷基，卤代烷基，烯基或炔基; Q表示在4位连接的任选取代的吡唑。还公开了用于农业的这些化合物的盐; 用于制备式（I）化合物的方法和中间产物，含有它们的试剂以及这些衍生物的用途或含有它们的试剂用于防治不希望的植物。

公开(公告)号：EP0958292A1

公开(公告)日：1999-11-24

申请号：EP98907930.0

申请日：1998-01-08

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  BAUMANN, Ernst ,  ENGEL, Stefan ,  MAYER, Guido ,  RHEINHEIMER, Joachim ,  WITSCHEL, Matthias ,  MISSLITZ, Ulf ,  WAGNER, Oliver ,  OTTEN, Martina ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07D277 ,  A01N43 ,  C07D231 ,  C07D261 ,  C07D263 ,  C07D273 ,  C07D291 ,  C07D401 ,  C07D403 ,  C07D405 ,  C07D409 ,  C07D411 ,  C07D413 ,  C07D417 ,  C07D419 ,  C07D498

CPC classification number: C07D231/20 ,  C07D261/04 ,  C07D261/20 ,  C07D413/10 ,  C07D417/10

Abstract: The invention concerns 4-(3-heterocyclyl-1-benzoyl)pyrazoles of formula (I) in which the variables have the following meanings: R1, R3: hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, alkylsulphinyl, alkylsulphinyl halide, alkylsulphonyl, alkylsulphonyl halide, aminosulphonyl, N-alkylaminosulphonyl, N,N-dialkylaminosulphonyl, N-alkylsulphonylamino, N-alkylsulphonylamino halide, N-alkyl-N-alkylsulphonylamino or N-alkyl-N-alkylsulphonylamino halide; R2: an optionally substituted 5- or 6-member heterocyclyl group containing between 1 and 4 identical or different heteroatoms selected from the group comprising oxygen, sulphur or nitrogen; R4: hydrogen, halogen or alkyl; R5: substituted pyrazole bonded in position 4. The invention also concerns: the salts of these 4-(3-heterocyclyl-1-benzoyl)pyrazoles which can be used for agricultural purposes; processes for preparing these substances; agents containing them; and the use as herbicides of these derivatives or agents containing them.

公开(公告)号：EP0958291A1

公开(公告)日：1999-11-24

申请号：EP98905274.0

申请日：1998-01-08

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  BAUMANN, Ernst ,  ENGEL, Stefan ,  MAYER, Guido ,  WITSCHEL, Matthias ,  RACK, Michael ,  GÖTZ, Norbert ,  GEBHARDT, Joachim ,  MISSLITZ, Ulf ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  OTTEN, Martina ,  RHEINHEIMER, Joachim

IPC: C07D277 ,  A01N43 ,  C07D231 ,  C07D261 ,  C07D263 ,  C07D273 ,  C07D291 ,  C07D403 ,  C07D413 ,  C07D417 ,  C07D419 ,  C07D498 ,  C07D237 ,  C07D311

CPC classification number: C07D413/10 ,  A01N43/76 ,  A01N43/80 ,  C07D231/20 ,  C07D261/04 ,  C07D261/20 ,  C07D403/12 ,  C07D417/10

Abstract: The invention concerns benzoyl derivatives of formula (I) in which the variables have the following meanings: R1, R2: hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, alkylsulphinyl, alkylsulphinyl halide, alkylsulphonyl, or C¿1?-C6 alkylsulphonyl halide; R?3¿: hydrogen, halogen or alkyl; R4, R5: hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, wherein the six last-mentioned groups can be substituted; X: O, S, NR9, CO or CR10R11; Y: O, S, NR12, CO or CR?13R14; R15¿: optionally substituted pyrazole which is bonded in position 4 and carries a hydroxy or sulphonyloxy group in position 5. The invention also concerns: the salts of these 3-heterocyclyl-substituted benzoyl derivatives which can be used for agricultural purposes; processes and intermediate products for preparing these substances; agents containing them; and the use as herbicides of these derivatives or agents containing them.