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1.SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME 有权
Title translation: 白细胞介素-1β转化酶的琥珀酰胺抑制剂公开(公告)号:EP1082127A4
公开(公告)日:2002-10-09
申请号:EP99918930
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , GALATSIS PAUL , THOMAS ANTHONY JEROME
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
CPC classification number: C07D257/04 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C2602/42 , C07D209/16 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D307/33 , C07D311/14 , C07D405/12
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公开(公告)号:AU758120B2
公开(公告)日:2003-03-13
申请号:AU3673099
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , GALATSIS PAUL , THOMAS ANTHONY JEROME
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:EE200000644A
公开(公告)日:2002-04-15
申请号:EEP200000644
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: THOMAS ANTHONY JEROME , CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , GALATSIS PAUL
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:AU738341B2
公开(公告)日:2001-09-13
申请号:AU4902397
申请日:1997-10-09
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: ALBRECHT HANS P , ALLEN HAMISH JOHN , BRADY KENNETH DALE , CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , THOMAS ANTHONY JEROME , WALKER NIGEL
IPC: C07D233/34 , A61K31/22 , A61K31/222 , A61K31/341 , A61K31/343 , A61K31/381 , A61K31/40 , A61K31/405 , A61K31/4164 , A61K31/4166 , A61K31/428 , A61K31/44 , A61K31/4409 , A61K31/4412 , A61K31/472 , A61K31/505 , A61K38/00 , A61P1/00 , A61P25/28 , A61P29/00 , A61P31/10 , A61P43/00 , C07C233/47 , C07C233/50 , C07C233/51 , C07C271/22 , C07C275/16 , C07C275/60 , C07C311/03 , C07C311/06 , C07C311/19 , C07C317/04 , C07C317/44 , C07C323/52 , C07C327/32 , C07D207/08 , C07D207/16 , C07D207/26 , C07D207/27 , C07D207/28 , C07D207/48 , C07D209/08 , C07D209/18 , C07D211/34 , C07D211/76 , C07D211/96 , C07D213/55 , C07D213/75 , C07D217/24 , C07D233/36 , C07D233/64 , C07D239/10 , C07D277/64 , C07D307/68 , C07D307/79 , C07D307/80 , C07D333/22 , C07D333/24 , C07D333/38 , C07D333/54 , C07D333/60 , C07K5/00 , C07K5/02 , C07K5/093
Abstract: The present invention relates to compounds that are inhibitors of interleukin-1 beta converting enzyme that have formula (I). This invention also relates to a method of treatment of stroke, inflammatory diseases, reperfusion injury, Alzheimer's disease, and shigellosis, and to a pharmaceutically acceptable composition that contains a compound that is an inhibitor of interleukin-1 beta converting enzyme.
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公开(公告)号:NO20005537A
公开(公告)日:2000-12-20
申请号:NO20005537
申请日:2000-11-02
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , GALATSIS PAUL , GILMORE JOHN LODGE , THOMAS ANTHONY JEROME , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHRINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
CPC classification number: C07D257/04 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C2602/42 , C07D209/16 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D307/33 , C07D311/14 , C07D405/12
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公开(公告)号:CA2327507A1
公开(公告)日:1999-11-11
申请号:CA2327507
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: GALATSIS PAUL , LUNNEY ELIZABETH ANN , THOMAS ANTHONY JEROME , KOSTLAN CATHERINE ROSE , GILMORE JOHN LODGE , HAYS SHERYL JEANNE , HARTER WILLIAM GLEN , KNAPP KRISTEN MICHELE , PARA KIMBERLY SUZANNE , CAPRATHE BRADLEY WILLIAM
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:ZA200006881B
公开(公告)日:2002-05-25
申请号:ZA200006881
申请日:2000-11-23
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , HARTER WILLIAM GLEN , KNAPP KRISTEN MICHELE , LUNNEY ELIZABETH ANN , GALATSIS PAUL , GILMORE JOHN LODGE , HAYS SHERYL JEANNE , KOSTLAN CATHERINE ROSE , PARA KIMBERLEY , THOMAS ANTHONY JEROME
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12 , A61K , C07D
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:HU0101963A2
公开(公告)日:2001-10-28
申请号:HU0101963
申请日:1999-04-30
Applicant: BASF AG , WARNER LAMBERT CO
Inventor: CAPRATHE BRADLEY WILLIAM , GALATSIS PAUL , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , THOMAS ANTHONY JEROME
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:SK16732000A3
公开(公告)日:2001-06-11
申请号:SK16732000
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE , GALATSIS PAUL , THOMAS ANTHONY JEROME
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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公开(公告)号:TR200003252T2
公开(公告)日:2001-04-20
申请号:TR200003252
申请日:1999-04-30
Applicant: WARNER LAMBERT CO , BASF AG
Inventor: CAPRATHE BRADLEY WILLIAM , GILMORE JOHN LODGE , HARTER WILLIAM GLEN , HAYS SHERYL JEANNE , KNAPP KRISTEN MICHELE , KOSTLAN CATHERINE ROSE , LUNNEY ELIZABETH ANN , PARA KIMBERLY SUZANNE
IPC: A61K31/197 , A61K31/277 , A61K31/352 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/41 , A61K31/416 , A61K31/4164 , A61K31/4178 , A61K31/4184 , A61K31/4192 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/443 , A61K31/47 , A61K38/05 , A61P1/04 , A61P9/02 , A61P9/08 , A61P9/10 , A61P19/02 , A61P25/00 , A61P25/28 , A61P29/00 , A61P31/04 , A61P43/00 , C07C233/47 , C07C255/29 , C07C311/10 , C07C311/13 , C07C323/59 , C07D209/08 , C07D209/16 , C07D211/14 , C07D213/40 , C07D215/12 , C07D231/56 , C07D233/54 , C07D233/64 , C07D235/06 , C07D235/08 , C07D249/18 , C07D257/04 , C07D265/28 , C07D307/33 , C07D311/14 , C07D405/12
Abstract: The present invention provides compounds of Formula (I), pharmaceutical compositions comprising a compound of Formula (I), and methods of treatment of stroke; inflammatory diseases such as rheumatoid arthritis or inflammatory bowel disease; septic shock; reperfusion injury; Alzheimer's disease; shigellosis; and multiple sclerosis.
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