公开(公告)号：EP0810998B1

公开(公告)日：2000-04-26

申请号：EP96902272.2

申请日：1996-02-14

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  ENGEL, Stefan ,  OTTEN, Martina ,  VOSSEN, Marcus ,  PLATH, Peter ,  RANG, Harald ,  HARREUS, Albrecht ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D261/08 ,  C07D277/30 ,  A01N43/80 ,  A01N43/78 ,  C07D333/24 ,  C07D307/54 ,  C07D275/02 ,  C07D213/57 ,  C07D263/32 ,  C07D277/66 ,  C07D231/12 ,  C07D215/12

CPC classification number: C07D207/327 ,  A01N43/78 ,  A01N43/80 ,  C07D213/57 ,  C07D213/647 ,  C07D213/70 ,  C07D213/74 ,  C07D215/12 ,  C07D231/12 ,  C07D231/14 ,  C07D235/18 ,  C07D239/26 ,  C07D239/38 ,  C07D249/08 ,  C07D261/08 ,  C07D261/18 ,  C07D263/32 ,  C07D271/06 ,  C07D271/107 ,  C07D275/02 ,  C07D277/30 ,  C07D277/32 ,  C07D277/34 ,  C07D277/36 ,  C07D277/66 ,  C07D279/06 ,  C07D285/08 ,  C07D285/125 ,  C07D307/54 ,  C07D317/30 ,  C07D319/06 ,  C07D333/24 ,  C07D333/28 ,  C07D339/06 ,  C07D339/08

Abstract: Phenyldiketone derivatives have the formula (I), in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy optionally substituted by 1 to 5 halogen atoms or C1-C4 alkoxy, halogen, cyano, nitro, a group -(Y)n-S(O)mR7 or a group -(Y)¿n-CO-R?8; Z is a 5 or 6 membered saturated or unsaturated heterocyclic rest that contains 1 to 3 heteroatoms selected from the group that includes oxygen, sulphur or nitrogen, optionally substituted by halogen, cyano, nitro, a group -CO-R8, C1-C4 alkyl, C1-C4 halogen alkyl, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 halogen alkylthio, di-C1-C4-alkylamino or an optionally substituted phenyl ring, and that forms a bicyclic system together with a condensed carbon cycle or a second condensed heterocycle; Y is O, NR9; n equals 0 or 1; m equals 0, 1 or 2; R7 is C1-C4 alkyl, C1-C4 halogen alkyl or NR?9R10; R8 is C¿1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy or NR?9R10; R9¿ is hydrogen or C¿1?-C4 alkyl; R?10 is C¿1-C4 alkyl; and R1 is cyclopropyl, 1-methylcyclopropyl, 1-methylthiocyclopropyl or tertiary butyl. Also disclosed are the salts of compounds (I) usually utilized in agriculture.

公开(公告)号：EP0802905B1

公开(公告)日：1998-09-09

申请号：EP96900897.8

申请日：1996-01-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  KLINTZ, Ralf ,  KÖNIG, Hartmann ,  HARREUS, Albrecht ,  GÖTZ, Norbert ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D213/61 ,  A01N43/40 ,  C07D405/12

CPC classification number: C07D405/10 ,  A01N43/40 ,  C07D213/61 ,  C07D405/12

Abstract: The invention concerns substituted 2-phenylpyridines of formula (I), in which: n = 0, 1; R?1, R3 and R4¿ represent H, OH, SH, NO¿2?, NH2, CN, COOH, CONH2, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl amino, dialkyl amino, alkyl thio, alkyl thio halide, alkoxy carbonyl, amino carbonyl, alkylamino carbonyl, dialkylamino carbonyl; R?2¿ represents H, OH, SH, NO¿2?, NH2, CN, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkyl thio halide, alkyl sulphinyl, alkyl sulphinyl halide, alkylsulphonyl, alkyl halide sulphonyl; R?5¿ represents H, CN or halogen; R6, R8 represent H or halogen; R7 represents H, OH, NO¿2?, CN, CF3-SO2-O-, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide; X represents -CO-, -O-C(R?9, R10¿)-CO-, -S-(R9, R10)-CO-, -CH¿2?-CH(R?11¿)-CO-, -CH=C(R11)-CO-; R9, R10 represent H or alkyl; R11 represents H, halogen or alkyl; Z represents optionally substituted tetrahydrofurane-3-yl or -C(R?15, COR16)-CH¿2-COR17; R15 represents H or alkyl; R?16 and R17¿ represent OH, NH¿2?, pyrrolidinyl, piperidinyl, morpholinyl, alkoxy, alkenyloxy, alkinyloxy, alkoxyalkoxy, cycloalkyloxy, alkylamino, dialkylamino, cycloalkylamino, dicycloalkylamino, alkenylamino, alkinylamino, or alternatively together represent -N(R?18)-N(R19¿)-, -N(R?20)-; R18, R19¿ represent H or alkyl; R20 represents H, alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy. The invention also concerns salts of these compounds and the use of the compounds and salts as herbicides and for drying out and defoliating plants.

Abstract translation: 本发明涉及式（I）的取代的2-苯基吡啶，其中：n = 0,1; R 1，R 3和R 4代表H，OH，SH，NO 2，NH 2，CN，COOH，CONH 2，卤素，烷基，烷基卤，烷氧基，烷氧基卤，烷基氨基，二烷基氨基，烷基硫代， 硫代卤化物，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基; R 2 2代表H，OH，SH，NO 2，NH 2，CN，卤素，烷基，烷基卤，烷氧基，烷氧基卤，烷硫基，烷基硫代卤化物，烷基亚磺酰基，烷基亚磺酰基卤，烷基磺酰基， ; R 5'代表H，CN或卤素; R6，R8代表H或卤素; R7表示H，OH，NO2，CN，CF3-SO2-O-，卤素，烷基，烷基卤，烷氧基，烷氧基卤化物; X表示-CO-，-OC（R 9，R 10）-CO - ， - S-（R 9，R 10）-CO-，-CH 2， CH = C（R11）-CO-; R9，R10代表H或烷基; R11代表H，卤素或烷基; Z代表任选取代的四氢呋喃-3-基或-C（R 15，COR 16）-CH 2 -OCR 17; R15代表H或烷基; R16和R17代表OH，NH2，吡咯烷基，哌啶基，吗啉基，烷氧基，烯氧基，炔氧基，烷氧基烷氧基，环烷氧基，烷基氨基，二烷基氨基，环烷基氨基，二环烷基氨基，烯基氨基， -N（R 19） - ， - N（R 20） - ; R18，R19'代表H或烷基; R20代表H，烷基，烯基，炔基，烷氧基，烯氧基。 本发明还涉及这些化合物的盐以及这些化合物和盐作为除草剂和用于干燥和脱叶植物的用途。

公开(公告)号：EP0802904B1

公开(公告)日：1998-09-09

申请号：EP96900563.6

申请日：1996-01-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  KLINTZ, Ralf ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D213/61 ,  A01N43/40

CPC classification number: A01N43/40 ,  C07D213/61

Abstract: The invention concerns substituted 2-phenylpyridines of formula (I), in which: n = 0, 1; R?1, R3 and R4¿ represent H, OH, SH, NO¿2?, NH2, CN, COOH, CONH2, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkyl amino, dialkyl amino, alkyl thio, alkyl thio halide, alkoxy carbonyl, amino carbonyl, alkylamino carbonyl, dialkylamino carbonyl; R?2¿ represents H, OH, SH, NO¿2?, NH2, CN, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, alkyl sulphinyl, alkyl sulphinyl halide, alkylsulphonyl, alkylsulphonyl halide; R?5¿ represents H, CN or halogen; R6, R13 represent H or halogen; X represents -CH¿2?- or -CO-; R?7, R8, R9, R10¿ represent H, NO¿2?, CN, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide; R?11¿ represents H, OH, NO¿2?, NH2, NHOH, CN, CHO, COOH, COCL, CONH2, 1-pyrrolidinyl carbonyl, 1-piperidinyl carbonyl, 4-morpholinyl carbonyl, 2-hydroxy carbonyl-pyrrolidine-1-yl-carbonyl, halogen or various organic groups; R?12¿ represents H, NO¿2?, NH2, NHOH, alkylsulphonyl amino, dialkylsulphonyl amino, alkylsulphonyl amino halide, alkoxy carbonyl-alkyl halide, alkoxycarbonyl-alkenyl halide. The invention also concerns salts of these compounds. Excluded are variants of formula (I) in which R?5, R7, R11 and R13¿ all represent hydrogen or R?7 and R8 or R10 and R11¿ represent fluorine. The said compounds can be used as herbicides and for drying out and defoliating plants.

Abstract translation: PCT No.PCT / EP96 / 00022 Sec。 371日期：1997年6月18日 102（e）日期1996年6月18日PCT提交1996年1月4日PCT公布。 WO96 / 21647 PCT出版物 日期1996年7月18日其中所有变量如本说明书中所定义的取代的2-苯基吡啶I用作除草剂和植物的干燥/脱叶。

公开(公告)号：EP0775137A1

公开(公告)日：1997-05-28

申请号：EP95927735.0

申请日：1995-07-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： PLATH, Peter ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  KARDORFF, Uwe ,  KÖNIG, Hartmann ,  RANG, Harald ,  GERBER, Matthias ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: A01N43 ,  C07D275 ,  C07D417

CPC classification number: C07D275/06 ,  A01N43/80 ,  C07D417/06

Abstract: The invention concerns saccharine derivatives of formula (I) in which the substituents are defined as follows: L, M hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, chlorine, cyano, methylsulphonyl, nitro or trifluoromethyl; Z hydrogen, C1-C4 alkyl, C3-C8 cycloalkyl, C3-C6 alkenyl, C3-C5 alkinyl, C1-C4 acyl, benzyl or phenyl, wherein any of the phenyl rings may be substituted by halogen or C1-C4 alkyl; Q a T-J group, T being a carbonyl (CO) group or the -CHY group, J being an isoxazole ring of formula (II) bonded at the 4-position and in which R1 is hydrogen or C¿1?-C4 alkyl, R?2 is C¿1-C4 alkyl, cyclopropyl, 1-methylcyclopropyl or 1-methylthiocyclopropyl, Y is an OH-group, a hydroxy group acylated with C2-C4 acyl, or a chlorine atom. The invention also concerns salts of such compounds usually used in agriculture.

公开(公告)号：EP0758322B1

公开(公告)日：2001-09-05

申请号：EP95918603.2

申请日：1995-04-25

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OBERDORF, Klaus ,  KÖNIG, Hartmann ,  MÜLLER, Bernd ,  KIRSTGEN, Reinhard ,  GRAMMENOS, Wassilios ,  SAUTER, Hubert ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  HARRIES, Volker

IPC: C07D231/20 ,  C07D231/08 ,  C07D401/04 ,  C07D403/04 ,  A01N43/56

CPC classification number: C07D401/04 ,  A01N43/56 ,  C07D231/08 ,  C07D231/20 ,  C07D403/04

Abstract: α-phenylbutenic acid methyl esters of formula (I) are disclosed, wherein -- represents a single or double bond and the index and substituents have the following meanings: n is 0, 1, 2, 3, or 4; R1 represents nitro, cyano, halogen, alkyl, alkyl halide or alkoxy; R2 represents hydrogen, nitro, cyano, halogen, alkyl, alkyl halide, alkoxy, alkylthio or alkoxycarbonyl; R3 represents optionally substituted alkyl, alkenyl or alkinyl; an optionally substituted saturated or mono or biunsaturated ring which in addition to carbon atoms can contain 1-3 heteroatoms chosen from oxygen, sulphur and nitrogen, as ring members, or an optionally, substituted mono or binuclear aromatic group which in addition to carbon atoms can contain 1-4 nitrogen atoms or one or two nitrogen atoms and an oxygen or sulphur atom or an oxygen or sulphur atom as ring members. Also disclosed is a process for the production of the claimed compounds and the use thereof against harmful fungi or animal pests.

公开(公告)号：EP0966452A1

公开(公告)日：1999-12-29

申请号：EP98904041.0

申请日：1998-01-08

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： RHEINHEIMER, Joachim ,  VON DEYN, Wolfgang ,  GEBHARDT, Joachim ,  HILL, Regina, Luise ,  RACK, Michael ,  KÖNIG, Hartmann ,  GÖTZ, Norbert ,  MAYWALD, Volker ,  KARDORFF, Uwe

IPC: C07D231 ,  C07D261 ,  C07D413 ,  C07D417

CPC classification number: C07D413/10 ,  C07D231/20 ,  C07D261/04 ,  C07D261/20 ,  C07D417/10

Abstract: The invention concerns a process for preparing sulphurous 2-chloro-3-(4,5-dihydroisoxazol-3-yl)-benzoic acids of general formula (I) in which the substituents have the meanings given in the description.

公开(公告)号：EP0804421B1

公开(公告)日：1998-09-16

申请号：EP95924888.1

申请日：1995-06-21

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  KÖNIG, Hartmann ,  KIRSTGEN, Reinhard ,  OBERDORF, Klaus ,  RÖHL, Franz ,  GÖTZ, Norbert ,  SAUTER, Hubert ,  LORENZ, Gisela ,  AMMERMANN, Eberhard

IPC: C07D231/22 ,  A01N43/56 ,  C07D231/20 ,  C07D401/04 ,  C07D403/04 ,  C07C239/10 ,  C07C271/28 ,  C07C271/58

CPC classification number: C07D401/04 ,  A01N47/24 ,  A01N47/30 ,  C07D231/08 ,  C07D231/20 ,  C07D231/22 ,  C07D403/04

公开(公告)号：EP0810998A1

公开(公告)日：1997-12-10

申请号：EP96902272.0

申请日：1996-02-14

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  ENGEL, Stefan ,  OTTEN, Martina ,  VOSSEN, Marcus ,  PLATH, Peter ,  RANG, Harald ,  HARREUS, Albrecht ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: A01N43 ,  C07D207 ,  C07D213 ,  C07D215 ,  C07D231 ,  C07D235 ,  C07D239 ,  C07D249 ,  C07D261 ,  C07D263 ,  C07D271 ,  C07D275 ,  C07D277 ,  C07D279 ,  C07D285 ,  C07D307 ,  C07D317 ,  C07D319 ,  C07D333 ,  C07D339

CPC classification number: C07D207/327 ,  A01N43/78 ,  A01N43/80 ,  C07D213/57 ,  C07D213/647 ,  C07D213/70 ,  C07D213/74 ,  C07D215/12 ,  C07D231/12 ,  C07D231/14 ,  C07D235/18 ,  C07D239/26 ,  C07D239/38 ,  C07D249/08 ,  C07D261/08 ,  C07D261/18 ,  C07D263/32 ,  C07D271/06 ,  C07D271/107 ,  C07D275/02 ,  C07D277/30 ,  C07D277/32 ,  C07D277/34 ,  C07D277/36 ,  C07D277/66 ,  C07D279/06 ,  C07D285/08 ,  C07D285/125 ,  C07D307/54 ,  C07D317/30 ,  C07D319/06 ,  C07D333/24 ,  C07D333/28 ,  C07D339/06 ,  C07D339/08

Abstract: Phenyldiketone derivatives have the formula (I), in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy optionally substituted by 1 to 5 halogen atoms or C1-C4 alkoxy, halogen, cyano, nitro, a group -(Y)n-S(O)mR7 or a group -(Y)¿n-CO-R?8; Z is a 5 or 6 membered saturated or unsaturated heterocyclic rest that contains 1 to 3 heteroatoms selected from the group that includes oxygen, sulphur or nitrogen, optionally substituted by halogen, cyano, nitro, a group -CO-R8, C1-C4 alkyl, C1-C4 halogen alkyl, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 halogen alkylthio, di-C1-C4-alkylamino or an optionally substituted phenyl ring, and that forms a bicyclic system together with a condensed carbon cycle or a second condensed heterocycle; Y is O, NR9; n equals 0 or 1; m equals 0, 1 or 2; R7 is C1-C4 alkyl, C1-C4 halogen alkyl or NR?9R10; R8 is C¿1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy or NR?9R10; R9¿ is hydrogen or C¿1?-C4 alkyl; R?10 is C¿1-C4 alkyl; and R1 is cyclopropyl, 1-methylcyclopropyl, 1-methylthiocyclopropyl or tertiary butyl. Also disclosed are the salts of compounds (I) usually utilized in agriculture.

Abstract translation: 苯基二酮衍生物具有式（I），其中取代基具有以下含义：L，M为氢，C 1 -C 6烷基，C 2 -C 6烯基，C 2 -C 6炔基，任选被1至5个卤素取代的C 1 -C 4烷氧基 （Y）nS（O）m R 7或基团 - （Y）n -CO-R 8的原子或C1-C4烷氧基，卤素，氰基，硝基， Z是含有1至3个选自包括氧，硫或氮的杂原子，任选被卤素，氰基，硝基，基团-CO-R 8，C 1 -C 4烷基或C 1 -C 4烷氧基取代的5或6元饱和或不饱和杂环基 ，C1-C4卤素烷基，C3-C8环烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4烷硫基，C1-C4卤代烷硫基，二-C1-C4-烷基氨基或任选取代的苯基环， 与稠合碳环或第二稠合杂环一起形成双环体系; Y是O，NR 9; n等于0或1; m等于0,1或2; R7是C1-C4烷基，C1-C4卤代烷基或NR9R10; R 8是C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基或NR 9 R 10; R9是氢或C1-C4烷基; R 10是C 1 -C 4烷基; R1是环丙基，1-甲基环丙基，1-甲基硫代环丙基或叔丁基。 还公开了通常用于农业的化合物（I）的盐。

公开(公告)号：EP0769010B1

公开(公告)日：2000-08-30

申请号：EP95924301.5

申请日：1995-06-21

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MÜLLER, Bernd ,  SAUTER, Hubert ,  GÖTZ, Norbert ,  KÖNIG, Hartmann ,  RÖHL, Franz ,  LORENZ, Gisela ,  AMMERMANN, Eberhard

IPC: C07D249/12 ,  C07D401/04 ,  C07D403/04 ,  A01N43/653 ,  A01N47/08 ,  C07C239/08 ,  C07C271/06

CPC classification number: C07D401/04 ,  A01N43/653 ,  A01N47/24 ,  A01N47/30 ,  C07C239/10 ,  C07C271/06 ,  C07D249/12 ,  C07D403/04

Abstract: The invention concerns 2-[1',2',4'-triazol-3'-yloxymethylene]-anilides of the formula (I) in which the subscript and substituents are as follows: n stands for 0, 1, 2, 3, or 4; X stands for a direct bond, oxygen or NRa, Ra being hydrogen, alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl; R1 nitro, cyano, halogen or optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy; R2 hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, heterocyclyl, aryl or heteroaryl; R4 hydrogen or optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, alkylcarbonyl or alkoxycarbonyl; R5 hydrogen, alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl. The invention also concerns methods of preparing such compounds, intermediates used in their preparation and their use in the control of animal and fungal pests.

公开(公告)号：EP0802903B1

公开(公告)日：1998-09-09

申请号：EP96900557.8

申请日：1996-01-04

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： SCHÄFER, Peter ,  HAMPRECHT, Gerhard ,  HEISTRACHER, Elisabeth ,  KLINTZ, Ralf ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D213/61 ,  A01N43/40

CPC classification number: C07D405/12 ,  A01N43/40 ,  C07D213/61 ,  C07D409/12