FUNGICIDAL MIXTURES
    2.
    发明申请
    FUNGICIDAL MIXTURES 审中-公开
    真菌混合物

    公开(公告)号:WO2008148859A3

    公开(公告)日:2009-09-17

    申请号:PCT/EP2008057027

    申请日:2008-06-05

    Abstract: The present invention relates to mixtures comprising, as active components, 1) a fungicidal compound of formula (I) wherein: R1 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; or heteroaryl; R2 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; heteroaryl; 5-pyrimidinyl; or 2-or 5-thiazolyl; R3 is H; alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryloxyalkyl; arylthioalkyl; aryl; heteroaryl; or alkylsilyl; R4 is H; acyl; haloacyl, alkoxycarbonyl; aryloxycarbonyl; alkylaminocarbonyl; or dialkylaminocarbonyl; or a salt thereof; and 2) a fungicidal compound II selected from azoles, strobilurins, carboxamides, heterocylic compounds, carbamates, and other active compounds in synergistically effective amounts.

    Abstract translation: 本发明涉及包含作为活性成分的1)式(I)的杀真菌化合物的混合物,其中:R 1是烷基; 烷氧基; 卤代; 芳; 芳基; 或杂芳基; R2是烷基; 烷氧基; 卤代; 芳; 芳基; 杂; 5-嘧啶基; 或2-或5-噻唑基; R3为H; 烷基; 烷氧基; 卤代; 芳; 芳氧; 芳硫基; 芳基; 杂; 或烷基甲硅烷基; R4是H; 酰基; 卤代酰基,烷氧基羰基; 芳氧羰基; 烷基氨基; 或二烷基氨基羰基; 或其盐; 和2)协同有效量的选自唑类,嗜球半胱氨酸,羧酰胺,杂环化合物,氨基甲酸酯和其它活性化合物的杀真菌化合物II。

    SUBSTITUTED 5-HETARYL-4-AMINOPYRIMIDINES
    5.
    发明申请
    SUBSTITUTED 5-HETARYL-4-AMINOPYRIMIDINES 审中-公开
    取代的5-杂芳基-4-氨基嘧啶

    公开(公告)号:WO2007110418A3

    公开(公告)日:2008-11-20

    申请号:PCT/EP2007052888

    申请日:2007-03-26

    CPC classification number: A01N43/54

    Abstract: The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and of their salts for controlling phytopathogenic fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to plant protection compositions which contain at least one such compound as active component. Het represents an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 hetero atoms as ring members which are selected among nitrogen, oxygen and sulphur, where the 5- or 6-membered heteroaromatic radical can have 1, 2, 3 or 4 identical or different substituents L; R 1 , R 2 represent inter alia hydrogen, C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four hetero atoms from the series O, N or S as ring members; or together form a ring; R 3 represents, inter alia, hydrogen, OH, halogen, cyano, NR 31 R 32 , C 1 -C 8 -alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulphinyl, C 1 -C 8 -alkyl-sulphonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkynyl; and R 4 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -haloalkylthio, or represents a radical of the formulae C(=Z)OR 41 , C(=Z)NR 42 R 43 , C(=Z)NR 44 -NR 42 R 43 , C(=Z)R 45 , CR 46 R 47 -OR 48 , CR 46 R 47 -NR 42 R 43 , ON(=CR 49 R 50 ), O-C(=Z)R 45 , NR 42 R 43a , NR 51 (C(=Z)R 45 ), NR 51 (C(=Z)OR 41 ), NR 51 (C(=Z)-NR 42 R 43 ), NR 52a (N=CR 49 R 50 ), NR 52 NR 42 R 43 , NR 52 OR 41 , or C(=N-X-R 45 )SR 41 .

    Abstract translation: 本发明涉及使用5-杂芳基-4-氨基嘧啶式I及其盐用于防治植物破坏性真菌。 本发明还涉及新的5-杂芳基-4-氨基嘧啶和含有至少一个这样的化合物作为有效成分的杀虫剂。 Het代表任选substituerten 5-或6-元芳族杂环,其具有1,2,3或4个氮,氧和选定的作为环成员的硫杂原子,其中所述5元或6元杂芳族残基1,2,3 可以包括或4个相同或不同的取代基L,R 1 ,R 2 除其他外,氢,C 1 -C 8 < / SUB>烷基,C 3 -C 8 环烷基,C 5 -C 10 二环烷基, ç 2 -C 8 烯基,C 4 -C 10 链二烯基,C 3 < / SUB> -C 6 环烯基,C 2 -C 8 炔基,苯基,萘基或五 - 或六元饱和的,部分 含有一个,具有从所述组的两个,三个或四个杂原子的不饱和或芳族杂环O,N或S作为环成员; 或一起形成一个环; [R 3 除其他外,氢,OH,卤素,氰基,NR 31 - [R 32 ,C 1 -C < SUB> 8 烷基,C 1 -C 8 烷氧基,C 1 -C 8 烷硫基,C 1 -C 8 烷基亚磺酰基,C 1 -C 8 烷基磺酰基,C < SUB> 2 -C 8 链烯基或C 2 -C 8 装置-Alkiny,且R 4 < / SUP>表示卤素,氰基,羟基,巯基,N 3 ,C 1 -C 6 烷基,C 2 < / SUB> -C 8 烯基,C 2 -C 8 炔基,C 1 -C < SUB> 6 卤代烷基,C 1 -C 6 烷氧基,C 3 -C 8 烯,C 3 -C 8 炔氧基,C 1 -C 6 卤代烷氧基,C < SUB> 1 -C 6 烷硫基,C 3 -C 8 烯,C 3 -C 8 炔硫基,C 1 -C 6 卤代烷硫基,或一个基团,式C(= Z)或 41 ,C(= Z)NR 42 ř 43 ,C(= Z)NR 44 -NR 42 - [R 43 ,C(= Z)R < SUP> 45 ,CR 46 - [R 47 为-OR 48 ,CR 46 - [R 47 -NR 42 - [R 43 ,ON(= CR 49 - [R 50 ),OC( = Z)R 45 ,NR 42 - [R 43A ,NR 51 (C(= Z)R 45 ),NR 51 (C(= Z)OR 41 ),NR 51 (C(= Z) - NR 42 - [R 43 ),NR 52A (N = CR 49 - [R 50 ),NR 52 NR 42 - [R 43 ,NR 52 41 ,或 C(= NXR 45 )SR 41 是。

    PYRAZINE COMPOUNDS
    7.
    发明申请
    PYRAZINE COMPOUNDS 审中-公开
    吡嗪化合物

    公开(公告)号:WO2008107398A3

    公开(公告)日:2008-10-23

    申请号:PCT/EP2008052515

    申请日:2008-02-29

    CPC classification number: C07D403/04

    Abstract: The present invention relates to novel pyrazine compounds of formula (I), N-oxides or agriculturally useful salts thereof, to their use for controlling harnful fungi, to their use in the treatment of cancer and to fungicidal or pharmaceutical compositions comprising at least one of these compounds as active component.

    Abstract translation: 本发明涉及新颖的式(I)吡嗪化合物,其N-氧化物或农业上可用的盐,用于控制恶性真菌,用于治疗癌症,以及杀真菌剂或药物组合物,其包含至少一种 这些化合物作为活性成分。

    FUNGICIDAL MIXTURES II
    10.
    发明申请
    FUNGICIDAL MIXTURES II 审中-公开
    真菌混合物II

    公开(公告)号:WO2009063075A3

    公开(公告)日:2010-05-06

    申请号:PCT/EP2008065604

    申请日:2008-11-14

    Abstract: The present invention relates to mixtures of fungicidally active compounds comprising at least one substituted 3-hydroxyl-3-(3-pyridyl)propanoate compound of the formula (I) X1 and X2 are hydrogen or X1 together with X2 form a covalent bond; R1 is H, CN, C1-C6-alkyl, C2-C6-alkynyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6- alkylthio-C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, aryl-C1-C4-alkyl, ary- loxy-C1-C4-alkyl, arylthio-C1-C4-alkyl, aryl, hetaryl-C1-C4-alkyl, hetaryloxy- C1-C4-alkyl, hetarylthioC1-C4-alkyl or heteroaryl, wherein the cyclic moieties of the last eight radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-alkylsulfinyl, C1-C4-alkylsulfonyl, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano and nitro; A is a covalent bond or Ci-C4-alkylen, which is unsubstituted or which may carry a substitutent selected from Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and cyano; Ar is aryl or heteroaryl, wherein the cyclic moieties of the aromatic radicals are unsubstituted or substituted with 1, 2 or 3 radicals Ra, where the radicals Ra are identical or different and selected from halogen, C1-C4-alkyl, C2-C4- alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano, nitro, aryl, hetaryl, aryloxy, hetaryloxy, aryloxy-C1-C4-alkyl and hetaryloxy-C1-C4-alkyl, wherein the cyclic moieties of the six last mentioned radicals are unsbsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, cyano and nitro; or a tautomer or a salt thereof. and at least one further fungicidally active compound II.

    Abstract translation: 本发明涉及杀真菌活性化合物的混合物,其包含至少一种式(I)的取代的3-羟基-3-(3-吡啶基)丙酸酯化合物,X 1和X 2是氢或X 1与X 2一起形成共价键; R 1是H,CN,C 1 -C 6烷基,C 2 -C 6炔基,C 1 -C 6烷氧基-C 1 -C 6烷基,C 1 -C 6烷基硫代-C 1 -C 6烷基,C 1 -C 6卤代烷基, C 1 -C 4 - 烷氧基,芳基-C 1 -C 4 - 烷基,芳氧基-C 1 -C 4 - 烷基,芳硫基-C 1 -C 4 - 烷基,芳基,杂芳基-C 1 -C 4烷基,苯氧基-C 1 -C 4烷基, C4-烷基或杂芳基,其中最后八个基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 2 -C 4 - 炔基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4烷基亚磺酰基,C 1 -C 4烷基磺酰基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基和硝基; A是共价键或C 1 -C 4亚烷基,其是未取代的或可以携带选自C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基和氰基的取代基; Ar是芳基或杂芳基,其中芳族基团的环状部分是未取代的或被1,2或3个基团R a取代,其中基团R a相同或不同并且选自卤素,C 1 -C 4烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基,硝基,芳基,杂芳基,芳氧基, 芳氧基-C 1 -C 4 - 烷基和芳基氧基-C 1 -C 4 - 烷基,其中六个最后提到的基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 1 -C 4 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,氰基和硝基; 或其互变异构体或其盐。 和至少一种其它杀真菌活性化合物II。

Patent Agency Ranking