NOVEL N-P-PROPARGYLOXYPHENETHYL-THIOACETIC ACID AMIDES
    3.
    发明申请
    NOVEL N-P-PROPARGYLOXYPHENETHYL-THIOACETIC ACID AMIDES 审中-公开
    新型N-对 - 丙烯酰氧基苯乙酸 - 柠檬酸

    公开(公告)号:WO02081437A3

    公开(公告)日:2003-01-09

    申请号:PCT/EP0203623

    申请日:2002-04-02

    Abstract: The invention relates to N-propargyloxy-phenethyl thioacetic acid amide derivatives of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5, R6, R7 and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is hydroxy, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenysulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl, optionally substituted alkynylsulfonyl or a group -O-CO-R11, -O-CO-O-R11 or -O-CO -CO-O-R11 wherein R11 is hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted heteroaryl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

    Abstract translation: 本发明涉及通式(I)的N-炔丙氧基 - 苯乙基硫代乙酰胺衍生物,其包括其旋光异构体和这些异构体的混合物,其中R 1为氢,烷基,环烷基或任选取代的芳基,R 2和R 3各自独立地为 氢或烷基,R4是烷基,烯基或炔基,R5,R6,R7和R8各自独立地是氢或烷基,R9是氢,任选取代的烷基,任选取代的烯基或任选取代的炔基,R 10是任选取代的芳基或任选取代的 杂芳基,Z是羟基,任选取代的芳氧基,任选取代的烷氧基,任选取代的炔氧基,任选取代的芳硫基,任选取代的烷硫基,任选取代的炔硫基,任选取代的烷基亚磺酰基,任选取代的烯基亚磺酰基,任选取代的炔基亚磺酰基,任选取代的烷基磺酰基, ,选择 取代的炔基磺酰基或基团-O-CO-R11,-O-CO-O-R11或-O-CO-CO-O-R11,其中R11是氢,任选取代的烷基,任选取代的环烷基,任选取代的芳基或任选地 取代的杂芳基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止植物病原微生物特别是真菌侵染植物。

    DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES
    10.
    发明申请
    DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES 审中-公开
    DIAZA-INDOLE DORIVATIVES及其作为FUNGICIDES的用途

    公开(公告)号:WO2010046215A3

    公开(公告)日:2011-04-07

    申请号:PCT/EP2009062673

    申请日:2009-09-30

    CPC classification number: A01N43/90 C07D471/04 C07D487/04

    Abstract: The present invention relates to novel compounds of the formula (I) in which any one of G1, G2 and G3 is N and the other two of G1, G2 and G3 are CR8, CR1 or CR2, such that when G1 is not N, G1 is CR8; when G2 is not N, G2 is CR1; when G3 is not N, G3 is CR2; and X1, X2, R1, R2, R3, R4, R6, R7, and R8 are as defined in the claims. In particular, the invention relates to use of these compounds in methods for the control and/or prevention of fungal infection in plants. The invention also relates to compositions containing these compounds as well as methods for preparing these compounds.

    Abstract translation: 本发明涉及式(I)的新化合物,其中,G1,G2和G3中的任一个为N,而G1,G2和G3中的任一个为CR8,CR1或CR2,使得当G1不为N时, G1是CR8; 当G2不是N时,G2是CR1; 当G3不为N时,G3为CR2; 并且X 1,X 2,R 1,R 2,R 3,R 4,R 6,R 7和R 8如权利要求中所定义。 特别地,本发明涉及这些化合物在控制和/或预防植物真菌感染的方法中的用途。 本发明还涉及含有这些化合物的组合物以及制备这些化合物的方法。

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