NOVEL PYRIDOPYRAZINE N-OXIDES
    3.
    发明申请
    NOVEL PYRIDOPYRAZINE N-OXIDES 审中-公开
    新型吡咯烷腈氧化物

    公开(公告)号:WO2008031566A3

    公开(公告)日:2008-09-18

    申请号:PCT/EP2007007912

    申请日:2007-09-11

    CPC classification number: C07D471/04 A01N43/90

    Abstract: The present invention relates to novel N -oxide derivatives of pyridopyrazines of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity :wherein X is N + -O" and Y is N; or X is N and Y is N + -O"; or X and Y are both N + -O"; R is for example H, halo, cyano, C 1-6 alkyl or C 1-6 alkoxy; R 1 is optionally substituted aryl or heteroaryl; R 2 is for example halo, C 1-8 alkyl, C 3-8 CycloaIkyI, aryl, or heteroaryl; R 3 and R 4 independently of each other are for example H, C 1-8 alkyl, halo(d-8)alkyl, C 2-8 alkenyl, C 2-8 alkynyl or aryl; or R 3 and R 4 together with the nitrogen atom to which they are attached form a C 3-10 alkylene chain or C 3-7 alkenylene chain optionally substituted with halo, C 1-4 alkyl, C 1-4 haloalkyl, C1-4 alkoxy; or R 3 and R 4 together with the nitrogen atom to which they are attached form for example a morpholine, thiomorpholine or thiomorpholine S-oxide ring; or R 3 and R 4 together with the nitrogen atom to which they are attached form a bicyclic annelated or fused ring; and R 7 and R 8 independently of each other are for example H, halo, cyano, C 1-4 alkyl, C 1-4 aIkoxy or halo(C 1-4 )alkyl.

    Abstract translation: 本发明涉及式(I)吡啶并吡嗪的新型N-氧化物衍生物作为具有杀微生物活性,特别是杀真菌活性的活性成分:其中X为N + O,Y为N; 或X为N且Y为N + O“; 或X和Y均为N + O-O“; R为例如H,卤素,氰基,C 1-6烷基或C 1-6烷基, R 1是任选取代的芳基或杂芳基; R 2是例如卤素,C 1-8烷基,C 1-4烷基, 环烷基,芳基或杂芳基; R 3和R 4彼此独立地是例如H,C 1〜 烷基,卤代(C 1-8)烷基,C 2-8链烯基,C 2-8炔基或芳基;或R 3, R 4和R 4与它们所连接的氮原子一起形成C 3-10亚烷基链或C 3-7亚烷基, 任选被卤素取代的亚烯基链,C 1-4烷基,C 1-4卤代烷基,C 1-4烷氧基或R 3和R 3 与它们所连接的氮原子一起形成例如吗啉,硫代吗啉或硫代吗啉S-氧化物环;或R 3和R 4, SUP与它们所连接的氮原子一起形成a 双环环或稠环; R 7和R 8彼此独立地是例如H,卤素,氰基,C 1-4烷基,C 1 -C 4烷基, 1-4烷氧基或卤代(C 1-4烷基)烷基。

    PESTICIDAL HETEROCYCLIC DIHALOALLYL COMPOUNDS
    4.
    发明申请
    PESTICIDAL HETEROCYCLIC DIHALOALLYL COMPOUNDS 审中-公开
    杀虫剂杂环二氢化合物

    公开(公告)号:WO2005068445A3

    公开(公告)日:2005-09-22

    申请号:PCT/EP2005000094

    申请日:2005-01-07

    Abstract: The invention relates to compounds of formula (I) wherein Het, A1, A2, A3, A4, D, W, T, Q, Y, X1, X2, R1, R2, R3, R4, k and m are as defined hereinabove, and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, to a process for the preparation of and to the use of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, to pesticidal compositions in which the active ingredient has been selected from those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in agrochemically usable salt form, to a process for the preparation of and to the use of those compositions, to plant propagation material treated with those compositions, to a method of controlling pests, to intermediates and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, for the preparation of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, and to a process for the preparation of and to the use of those intermediates and, where applicable, possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof.

    Abstract translation: 本发明涉及式(I)化合物,其中Het,A1,A2,A3,A4,D,W,T,Q,Y,X1,X2,R1,R2,R3,R4,k和m如上所定义 ,以及(如适用)可能的E / Z异构体,E / Z异构体和/或其互变异构体的混合物,在每种情况下为游离形式或盐形式,用于制备和使用这些化合物的方法 ,E / Z异构体,E / Z异构体和/或互变异构体的混合物,其中活性成分选自那些化合物,E / Z异构体,E / Z异构体和/或互变异构体的混合物的农药组合物 游离形式或农业可用盐形式的情况,制备和使用这些组合物的方法,用这些组合物处理的繁殖材料,控制害虫的方法,中间体以及在适用的情况下 可能的E / Z异构体,E / Z异构体和/或其互变异构体的混合物,在每种情况下为游离形式或盐形式,用于制备那些 磅,E / Z异构体,E / Z异构体和/或互变异构体的混合物,以及制备和使用那些中间体的方法,以及可能的E / Z异构体,E / Z异构体的混合物 和/或其互变异构体。

    NOVEL INSECTICIDES
    6.
    发明申请
    NOVEL INSECTICIDES 审中-公开
    新型杀虫剂

    公开(公告)号:WO2005085234A2

    公开(公告)日:2005-09-15

    申请号:PCT/EP2005002204

    申请日:2005-03-02

    Abstract: Compounds of the formula (I) in which Z, is an oxygen atom; or a sulfur atom; Z2 is an oxygen atom; or a sulfur atom; R, is an aryl or heteroaryl group, which is unsubstituted or substituted; R2 is hydrogen; or an organic substituent; R3 is hydrogen; or an organic substituent; R4 is hydrogen; or an organic substituent; or R3 and R4, taken together, form, together with the nitrogen atom, to which they are attached, a ring, which is unsubstituted or substituted; R5 is hydrogen; or an unsubstituted or substituted alkyl group; or forms, taken together with R8 or with a monovalent substituent attached to that atom of R6, via which atom R6 is directly connected with the carbon atom, shown in the formula I, which carries R5, one additional bond; R6 and R7, taken together, form, together with the two carbon atoms, shown in the formula I, to which atoms they are attached, a bicyclic ring system, which ring system is carbocyclic or heterocyclic, which ring system is substituted, in the manner shown in the formula I, by the four substituents -N(R2)-C(=Z1)-R,, -C(=Z2)-N(R3)-R4, R5 and R8, and which ring system is optionally further substituted; and R8 is hydrogen; or an unsubstituted or substituted alkyl group; or forms, taken together with R5 or with a monovalent substituent attached to that atom of R7, via which atom R7 is directly connected with the carbon atom, shown in the formula I, which carries R8, one additional bond, and, where appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

    Abstract translation: 其中Z为氧原子的式(I)化合物; 或硫原子; Z2是氧原子; 或硫原子; R 1是未取代或取代的芳基或杂芳基; R2是氢; 或有机取代基; R3是氢; 或有机取代基; R4是氢; 或有机取代基; 或者R 3和R 4一起与它们所连接的氮原子一起形成未被取代或被取代的环, R5是氢; 或未取代或取代的烷基; 或其形式,与R8一起或与R6的该原子连接的一价取代基,其中原子R6直接与碳原子连接,如式I所示,其携带R5,另外一个键; R6和R7一起与式I中所示的两个碳原子一起形成,其中连接有它们的原子,双环体系,该环系是碳环或杂环,该环系被取代,在 通式为四种取代基-N(R 2)-C(= Z 1)-R 1 -C(= Z 2)-N(R 3)-R 4,R 5和R 8,并且该环系是任选的 进一步取代; R8是氢; 或未取代或取代的烷基; 或其形式与R5一起或与R7的原子连接的一价取代基,其中原子R7与碳原子直接连接,如式I所示,其携带R8,一个附加键,并且在适当的情况下, 互变异构体,以游离形式或盐形式,可以用作农业化学活性成分,并且可以以本身已知的方式制备。

    FUNGICIDAL COMPOUNDS AND COMPOSITIONS
    9.
    发明申请
    FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
    杀真菌化合物和组合物

    公开(公告)号:WO2008014955A3

    公开(公告)日:2008-04-17

    申请号:PCT/EP2007006720

    申请日:2007-07-30

    CPC classification number: C07D237/12 A01N43/58

    Abstract: The present invention relates, inter alia, to a compound having the formula (I):-wherein (R)n is selected from the group consisting of 4-Br, 4-OCH 2 CH 3 , 4-OCH 2 CF 3 , 2-CH 3 -4-C1, 2-CH 3 -4-OCH 3 , 2-CH 3 -4-OCF 3 , 2-F-4-Br, 2-F-4-CF 3 , 3-CH 3 -4-Br, 3-F-4-C1, 3-F-4-CH 3 , 3-F-4-Br, 3-F-4-OCH 3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I) - and also to fungicidal compositions comprising compounds having the formula (II) and/or (III):Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.

    Abstract translation: 本发明特别涉及具有式(I)的化合物:其中(R)n选自4-Br,4-OCH 2 CH 2, 3,4-OCH 2,CF 3,2-CH 3,-S-3,-S-,2-CH 3 4-OCH 3,2-CH 3 -OR-3-N,2-F-4-Br,2 -F-4-CF 3,3-CH 3〜4-Br,3-F-4-C1,3-F-4-CH 3 3-F-4-Br,3-F-4-OCH 3 3和3-F-4-F。 本发明还涉及包含具有式(I)的化合物的杀真菌组合物,以及包含具有式(II)和/或(III)的化合物的杀真菌组合物:此外,本发明涉及用于控制致病性的方法 使用组合物的生物体。

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