公开(公告)号：AT260250T

公开(公告)日：2004-03-15

申请号：AT99968337

申请日：1999-12-01

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： ZELLER MARTIN ,  JEANGUENAT ANDRE ,  LAMBERTH CLEMENS

IPC: C07D295/22 ,  A01N37/44 ,  A01N41/06 ,  C07B61/00 ,  C07C303/34 ,  C07C303/38 ,  C07C303/40 ,  C07C307/06 ,  C07C311/06 ,  C07C311/07 ,  C07C311/11

Abstract: The invention relates to alpha-sulfin- and alpha-sulfonamino acid amides of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinn is a number zero or one;R1 is C1-C12alkyl, C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkenyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR12R13 wherein R12 and R13 are each independently of the other hydrogen or C1-C6-alkyl, or together are tetra- or penta-methylene;R2 and R3 are each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring;R4, R5, R6 and R7 are each independently hydrogen or C1-C4alkyl;R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl;R9, R10, R14, R15, R16 and R17 are each independently hydrogen or C1-C4alkyl;A is optionally substituted phenyl, andto the preparation of those substances and to agrochemical compositions comprising at least one of those compounds as active ingredient. The invention relates also to the preparation of the said compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

公开(公告)号：AU2003251456A1

公开(公告)日：2004-02-16

申请号：AU2003251456

申请日：2003-07-23

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： LAMBERTH CLEMENS ,  ZELLER MARTIN ,  GOEGH TIBOR

IPC: C07D333/24 ,  C07C215/64 ,  C07C215/74 ,  C07C217/74 ,  C07C217/80 ,  C07C235/36 ,  C07C235/38 ,  C07C323/62 ,  C07D213/56 ,  C07D213/61 ,  C07D307/54 ,  C07D333/28 ,  C07F7/18

Abstract: The invention relates to N-bisaryl- and N-aryl-cycloalkylidenyl-a-hydroxy- and a-alkoxy acetic acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R 1 is hydrogen, C 1 -C 12 alkyl; C 2 -C 12 alkenyl; C 2 -C 12 alkynyl; C 1 -C 12 haloalkyl; R 2 is hydrogen; optionally substituted alkyl; optionally substituted alkenyl or optionally substituted alkynyl; R 3 is optionally substituted aryl or optionally substituted heteroaryl; A is an optionally substituted saturated or unsaturated C 3 -C 8 -cycloalkylidene, optionally substituted phenylidene or optionally substituted saturated or unsaturated heterocyclylidene bridge, R 4 and R 5 are each independently hydrogen or an organic radical, and R 6 is hydrogen; tri-C 1 -C 4 alkyl-silyl; di-C 1 -C 4 alkyl-phenylsilyl; C 1 -C 4 alkyl-diphenylsilyl; triphenylsilyl; optionally substituted alkyl; optionally substituted alkenyl or optionally substituted alkynyl. The compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic miroorganism, especially fungi.

公开(公告)号：HK1054368A1

公开(公告)日：2003-11-28

申请号：HK03104881

申请日：2003-07-08

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： LAMBERTH CLEMENS ,  ZELLER MARTIN ,  KUNZ WALTER ,  CEDERBAUM FREDRIK

IPC: A01N37/18 ,  A01N37/30 ,  A01N37/36 ,  A01N41/06 ,  A01N41/12 ,  A01N43/00 ,  A01N43/12 ,  A01N43/30 ,  A01N43/32 ,  A01P3/00 ,  C07C231/02 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C239/12 ,  C07C239/22 ,  C07C313/04 ,  C07C323/56 ,  C07C323/60 ,  C07C323/62 ,  C07D213/02 ,  C07D213/56 ,  C07D215/14 ,  C07D239/02 ,  C07D239/26 ,  C07D241/42 ,  C07D261/08 ,  C07D277/64 ,  C07D307/16 ,  C07D307/79 ,  C07D307/80 ,  C07D317/60 ,  C07D319/18 ,  C07D333/00 ,  C07D333/24 ,  C07D333/28 ,  C07D333/52 ,  C07D333/60 ,  C07C ,  C07D ,  A01N

Abstract: The invention relates to phenyl-propargylether derivatives of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinR1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl,R2 and R3 are each independently hydrogen or alkyl,R4 is alkyl, alkenyl or alkynyl,R5, R6, R7, and R8 are each independently hydrogen or alkyl,R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl,R10 is optionally substituted aryl or optionally substituted heteroaryl, andZ is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

公开(公告)号：HU0301965A2

公开(公告)日：2003-09-29

申请号：HU0301965

申请日：2001-05-15

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： CEDERBAUM FREDRIK ,  KUNZ WALTER ,  LAMBERTH CLEMENS ,  ZELLER MARTIN

IPC: A01N37/18 ,  A01N37/30 ,  A01N37/36 ,  A01N41/06 ,  A01N41/12 ,  A01N43/00 ,  A01N43/12 ,  A01N43/30 ,  A01N43/32 ,  A01P3/00 ,  C07C231/02 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C239/12 ,  C07C239/22 ,  C07C313/04 ,  C07C323/56 ,  C07C323/60 ,  C07C323/62 ,  C07D213/02 ,  C07D213/56 ,  C07D215/14 ,  C07D239/02 ,  C07D239/26 ,  C07D241/42 ,  C07D261/08 ,  C07D277/64 ,  C07D307/16 ,  C07D307/79 ,  C07D307/80 ,  C07D317/60 ,  C07D319/18 ,  C07D333/00 ,  C07D333/24 ,  C07D333/28 ,  C07D333/52 ,  C07D333/60

Abstract: The invention relates to phenyl-propargylether derivatives of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinR1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl,R2 and R3 are each independently hydrogen or alkyl,R4 is alkyl, alkenyl or alkynyl,R5, R6, R7, and R8 are each independently hydrogen or alkyl,R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl,R10 is optionally substituted aryl or optionally substituted heteroaryl, andZ is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

公开(公告)号：ES2191422T3

公开(公告)日：2003-09-01

申请号：ES99911707

申请日：1999-02-25

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： JEANGUENAT ANDRE ,  ZELLER MARTIN

IPC: C07D295/14 ,  A01N41/02 ,  A01N41/06 ,  C07C237/08 ,  C07C307/06 ,  C07C311/06 ,  C07C311/19 ,  C07C323/63 ,  C07D209/20 ,  C07D213/56 ,  C07D235/16 ,  C07D277/64 ,  C07D307/54 ,  C07D311/80 ,  C07D317/60 ,  C07D333/24 ,  C07D333/28

Abstract: Novel alpha-amino acid amides of formula (I) as well as possible isomers and mixtures of isomers thereof, wherein the substituents are defined as follows: n is the number zero or one; R1 is optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl; or a group NRaRb wherein Ra and Rb are each independently of the other hydrogen, alkyl or form together an alkylene bridge; R2 is hydrogen or alkyl; R3 is optionally substituted aryl or heteroaryl; A is alkylene; and B is optionally substituted aryl; with the exception of the following compounds 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methylphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-chlorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-nitrolphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methoxyphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-fluorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-phenyl-sulfonylamino-acetamide and 2-phenyl-N-(1-phenyl-ethyl)-2-methane-sulfonylamino-acetamide. The novel compounds have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms, in particular fungi.

公开(公告)号：CA2461438A1

公开(公告)日：2003-05-22

申请号：CA2461438

申请日：2002-11-15

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： LAMBERTH CLEMENS ,  VETTIGER THOMAS ,  ZELLER MARTIN ,  FABER DOMINIK

IPC: C07C231/02 ,  C07C213/02 ,  C07C231/00 ,  C07C233/00 ,  C07C235/08 ,  C07C235/32 ,  C07C235/34 ,  C07D213/56

Abstract: The invention concerns a novel process for the preparation of 2-phenyl-2- hydroxy-N-[2-(3-alkoxy-4-hydroxyphenyl)-ethyl]-acetamides of the formula (I) , wherein R1 is alkyl, R2 and R3 are each independently hydrogen or alkyl, and R4 is optionally substituted aryl or optionally substituted heteroaryl, whic h process comprises reacting a 2-(3-alkoxy-4-hydroxyphenyl)-ethylamine of the formula (II), wherein R1 R2 and R3 are as defined above with a .alpha.- hydoxycarboxylic acid ester of the formula (III) or a dioxolanone of the formula (III)a, wherein R4 is as defined above, and R5, R6 and R7 independently of each other are lower alkyl. The compounds of formula (I) ar e important intermediates for a novel group of fungicides derived from mandeli c acid amides.

公开(公告)号：BR0107770A

公开(公告)日：2003-04-29

申请号：BR0107770

申请日：2001-01-23

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： CRAIG GERALD WAYNE ,  EBERLE MARTIN ,  ZELLER MARTIN ,  BONDY STEVEN SCOTT ,  COMER DANIEL DENNIS ,  CHENG SOAN ,  PENZOTTI JULIE ELIZABETH ,  GROOTENHUIS PETER DIEDERIK JAN ,  EHRLER JUERG

IPC: A01N37/34 ,  A01N37/38 ,  A01N37/40 ,  A01N37/48 ,  A01P13/00 ,  C07C17/14 ,  C07C43/215 ,  C07C43/225 ,  C07C43/23 ,  C07C47/575 ,  C07C49/84 ,  C07C69/734 ,  C07C69/736 ,  C07C69/76 ,  C07C205/35 ,  C07C205/37 ,  C07C217/48 ,  C07C217/60 ,  C07C217/76 ,  C07C251/48 ,  C07C255/37 ,  C07C255/46 ,  C07C255/54 ,  C07D209/48 ,  C07C43/00

Abstract: Compounds of general formula (I) wherein the substituents are as defined in claim 1 are suitable for use as herbicides

公开(公告)号：AT231489T

公开(公告)日：2003-02-15

申请号：AT99911707

申请日：1999-02-25

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： JEANGUENAT ANDRE ,  ZELLER MARTIN

IPC: C07D295/14 ,  A01N41/02 ,  A01N41/06 ,  C07C237/08 ,  C07C307/06 ,  C07C311/06 ,  C07C311/19 ,  C07C323/63 ,  C07D209/20 ,  C07D213/56 ,  C07D235/16 ,  C07D277/64 ,  C07D307/54 ,  C07D311/80 ,  C07D317/60 ,  C07D333/24 ,  C07D333/28

Abstract: Novel alpha-amino acid amides of formula (I) as well as possible isomers and mixtures of isomers thereof, wherein the substituents are defined as follows: n is the number zero or one; R1 is optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl; or a group NRaRb wherein Ra and Rb are each independently of the other hydrogen, alkyl or form together an alkylene bridge; R2 is hydrogen or alkyl; R3 is optionally substituted aryl or heteroaryl; A is alkylene; and B is optionally substituted aryl; with the exception of the following compounds 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methylphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-chlorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-nitrolphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-methoxyphenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-(4-fluorophenyl)-sulfonylamino-acetamide, 2-phenyl-N-(1-phenyl-ethyl)-2-phenyl-sulfonylamino-acetamide and 2-phenyl-N-(1-phenyl-ethyl)-2-methane-sulfonylamino-acetamide. The novel compounds have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms, in particular fungi.

公开(公告)号：BR0110810A

公开(公告)日：2003-02-11

申请号：BR0110810

申请日：2001-05-15

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： LAMBERTH CLEMENS ,  ZELLER MARTIN ,  KUNZ WALTER ,  CEDERBAUM FREDRIK

IPC: A01N37/18 ,  A01N37/30 ,  A01N37/36 ,  A01N41/06 ,  A01N41/12 ,  A01N43/00 ,  A01N43/12 ,  A01N43/30 ,  A01N43/32 ,  A01P3/00 ,  C07C231/02 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C239/12 ,  C07C239/22 ,  C07C313/04 ,  C07C323/56 ,  C07C323/60 ,  C07C323/62 ,  C07D213/02 ,  C07D213/56 ,  C07D215/14 ,  C07D239/02 ,  C07D239/26 ,  C07D241/42 ,  C07D261/08 ,  C07D277/64 ,  C07D307/16 ,  C07D307/79 ,  C07D307/80 ,  C07D317/60 ,  C07D319/18 ,  C07D333/00 ,  C07D333/24 ,  C07D333/28 ,  C07D333/52 ,  C07D333/60

Abstract: The invention relates to phenyl-propargylether derivatives of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinR1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl,R2 and R3 are each independently hydrogen or alkyl,R4 is alkyl, alkenyl or alkynyl,R5, R6, R7, and R8 are each independently hydrogen or alkyl,R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl,R10 is optionally substituted aryl or optionally substituted heteroaryl, andZ is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

公开(公告)号：PT1003719E

公开(公告)日：2002-10-31

申请号：PT98946275

申请日：1998-08-04

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： ZELLER MARTIN ,  JEANGUENAT ANDRE

IPC: C07D239/26 ,  A01N41/06 ,  A01N43/10 ,  A01P3/00 ,  A01P13/00 ,  C07C217/60 ,  C07C237/08 ,  C07C307/06 ,  C07C311/06 ,  C07C311/09 ,  C07C311/10 ,  C07C311/11 ,  C07C311/14 ,  C07C313/06 ,  C07D213/30 ,  C07D213/61 ,  C07D215/14 ,  C07D231/12 ,  C07D277/64 ,  C07D333/16 ,  C07D333/24 ,  C07C311/00

Abstract: The invention relates to novel pesticidally active compounds of the general formula Ias well as possible isomers and mixtures of isomers thereof,whereinn is a number zero or one; andR1 is C1-C12alkyl that is unsubstituted or may be substituted by C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or by C3-C6alkynyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl: or a group NR11R12 wherein R11 and R12 are each independently of the other hydrogen or C1-C8alkyl, or together are tetra- or penta-methylene;R2 and R3 are each independently of the other hydrogen; C1-C8alkyl; C1-C8alkyl substituted by hydroxy, C1-C4alkoxy, mercapto or by C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered ring;R4, R5, R6 and R7 are identical or different and are each independently of the others hydrogen or C1-C4alkyl;R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl;A is C1-C6alkylene; andB is optionally mono- or poly-nuclear, unsubstituted or substituted aryl; optionally mono- or poly-nuclear, unsubstituted or substituted heteroaryl; C4-C12alkyl; or C3-C8cycloalkyl.The novel compounds have plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms.