公开(公告)号：FI970147A

公开(公告)日：1997-01-14

申请号：FI970147

申请日：1997-01-14

Applicant: BASF AG

Inventor： HELLENDAHL BEATE ,  LANSKY ANNEGRET ,  MUNSCHAUER RAINER ,  BIALOJAN SIEGFRIED ,  UNGER LILIANE ,  TESCHENDORF HANS-JUERGEN ,  WICKE KARSTEN ,  DRESCHER KARLA

IPC: C07D249/08 ,  A61K31/41 ,  A61K31/435 ,  A61K31/4427 ,  A61K31/445 ,  A61K31/505 ,  A61K31/53 ,  A61P1/08 ,  A61P25/18 ,  A61P25/20 ,  A61P25/24 ,  A61P25/26 ,  C07D249/12 ,  C07D249/14 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D

Abstract: PCT No. PCT/EP95/02781 Sec. 371 Date Jan. 14, 1997 Sec. 102(e) Date Jan. 14, 1997 PCT Filed Jul. 14, 1995 PCT Pub. No. WO96/02520 PCT Pub. Date Feb. 1, 1996The present invention relates to triazole compounds of the following formula: where R1, R2, A, B and Ar have the meanings stated in the description. The compounds according to the invention have a high affinity for the dopamine D3 receptor and can therefore be used to treat disorders which respond to dopamine D3 ligands.

公开(公告)号：FI945488A

公开(公告)日：1995-01-18

申请号：FI945488

申请日：1994-11-22

Applicant: BASF AG

Inventor： HELLENDAHL BEATE ,  SCHLECKER RAINER ,  ROEHL FRANZ ,  ZIPPLIES MATTHIAS ,  RASCHACK MANFRED ,  HAFNER MATTHIAS

IPC: A61K31/47 ,  A61K31/472 ,  A61P9/00 ,  A61P31/04 ,  C07D217/04 ,  C07D217/06 ,  C07D

公开(公告)号：NO944476D0

公开(公告)日：1994-11-22

申请号：NO944476

申请日：1994-11-22

Applicant: BASF AG

Inventor： HELLENDAHL BEATE ,  SCHLECKER RAINER ,  ROEHL FRANZ ,  ZIPPLIES MATTHIAS ,  RASCHACK MANFRED ,  HAFNER MATTHIAS

IPC: A61K31/47 ,  C07D217/04 ,  C07D217/06

公开(公告)号：AU6062894A

公开(公告)日：1994-10-27

申请号：AU6062894

申请日：1994-04-21

Applicant: BASF AG

Inventor： WINGERT HORST ,  HELLENDAHL BEATE ,  SAUTER HUBERT ,  LORENZ GISELA

IPC: A01N43/18 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  A01N43/836 ,  C07D207/337 ,  C07D209/12 ,  C07D213/55 ,  C07D213/56 ,  C07D213/61 ,  C07D215/14 ,  C07D235/20 ,  C07D261/08 ,  C07D263/32 ,  C07D263/56 ,  C07D271/10 ,  C07D271/107 ,  C07D277/10 ,  C07D277/22 ,  C07D277/30 ,  C07D277/64 ,  C07D277/66 ,  C07D285/12 ,  C07D307/54 ,  C07D307/81 ,  C07D333/20 ,  C07D333/24 ,  C07D333/58 ,  C07D413/04 ,  A01N43/76

Abstract: Diaryl derivatives of the general formula I in which A denotes =CHOR , =CHSR , =CHR , =CHCl or =NOR , B denotes OR , SR or NR R , Het denotes a mono-, di- or trinuclear aromatic five-membered or six-membered heterocycle which can optionally be substituted by R, R R , R , R , R are identical or different and denote hydrogen or alkyl and U, V, and W are identical or different and denote halogen, alkyl or alkoxy, and fungicides containing these compounds.A

公开(公告)号：HU9401168D0

公开(公告)日：1994-07-28

申请号：HU9401168

申请日：1994-04-22

Applicant: BASF AG

Inventor： SAUTER HUBERT ,  LORENZ GISELA ,  WINGERT HORST ,  HELLENDAHL BEATE

IPC: A01N43/18 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  A01N43/836 ,  C07D207/337 ,  C07D209/12 ,  C07D213/55 ,  C07D213/56 ,  C07D213/61 ,  C07D215/14 ,  C07D235/20 ,  C07D261/08 ,  C07D263/32 ,  C07D263/56 ,  C07D271/10 ,  C07D271/107 ,  C07D277/10 ,  C07D277/22 ,  C07D277/30 ,  C07D277/64 ,  C07D277/66 ,  C07D285/12 ,  C07D307/54 ,  C07D307/81 ,  C07D333/20 ,  C07D333/24 ,  C07D333/58 ,  C07D413/04

Abstract: Diaryl derivatives of the general formula I in which A denotes =CHOR , =CHSR , =CHR , =CHCl or =NOR , B denotes OR , SR or NR R , Het denotes a mono-, di- or trinuclear aromatic five-membered or six-membered heterocycle which can optionally be substituted by R, R R , R , R , R are identical or different and denote hydrogen or alkyl and U, V, and W are identical or different and denote halogen, alkyl or alkoxy, and fungicides containing these compounds.A

公开(公告)号：AU4066993A

公开(公告)日：1993-12-30

申请号：AU4066993

申请日：1993-05-12

Applicant: BASF AG

Inventor： HELLENDAHL BEATE ,  ROEHL FRANZ ,  RASCHACK MANFRED ,  HAFNER MATTHIAS

IPC: C07C211/49 ,  C07C215/50 ,  C07C217/58 ,  C07C219/28 ,  C07C233/43 ,  A61K31/135 ,  A61K31/16 ,  C07C215/64

公开(公告)号：CA2136449A1

公开(公告)日：1993-12-09

申请号：CA2136449

申请日：1993-05-13

Applicant: BASF AG

Inventor： HELLENDAHL BEATE ,  SCHLECKER RAINER ,  ROEHL FRANZ ,  ZIPPLIES MATTHIAS ,  RASCHACK MANFRED ,  HAFNER MATTHIAS

IPC: A61K31/47 ,  A61K31/472 ,  A61P9/00 ,  A61P31/04 ,  C07D217/04 ,  C07D217/06 ,  C07D217/02

Abstract: 2136449 9324461 PCTABS00028 Medicament for oral administration which contains as active substance per individual dose, besides the customary galenic auxiliaries, 10 to 1000 mg of a compound of general formula (I) or (II) in which W is a carbonyl group or a single bond, R1 is a hydrogen atom or a group of the general formula R3CO in which R3 is a lower alkyl, lower alkoxy, mono lower alkylamino or di lower alkylamino group, R2 is an alkyl residue with 3 to 20 carbon atoms which may be branched or unbranched and contain 1 to 3 double bonds, a saturated cycle of 3 to 7 carbon atoms integrated into the chain or as substituent, or may be substituted by one or more aromatic rings or contain an oxygen or sulphur atom, as a racemate and as isolated enantiomers; or the addition salt thereof with a physiologically acceptable acid, and the active substances themselves insofar as they are novel.

公开(公告)号：ZA921186B

公开(公告)日：1993-08-19

申请号：ZA921186

申请日：1992-02-19

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  HARREUS ALBRECHT ,  SAUTER HUBERT ,  HELLENDAHL BEATE ,  DOETZER REINHARD ,  AMMERMANN EBERHARD ,  LORENZ GISELA

IPC: A01N37/50 ,  A01N43/54 ,  A01N43/58 ,  A01N43/76 ,  A01N43/836 ,  C07C69/65 ,  C07C69/653 ,  C07C69/734 ,  C07C69/738 ,  C07C251/48 ,  C07C251/50 ,  C07C251/52 ,  C07C251/54 ,  C07C251/56 ,  C07C251/58 ,  C07C251/60 ,  C07C251/86 ,  C07C255/15 ,  C07C255/57 ,  C07C255/58 ,  C07C255/62 ,  C07D213/77 ,  C07D239/42 ,  C07D241/20 ,  C07D263/32 ,  C07D333/28 ,  C07C ,  A01N

Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).

公开(公告)号：AU1103792A

公开(公告)日：1992-08-27

申请号：AU1103792

申请日：1992-02-19

Applicant: BASF AG

Inventor： HARREUS ALBERT ,  SAUTER HUBERT ,  HELLENDAHL BEATE ,  DOETZER REINHARD ,  AMMERMANN EBERHARD ,  LORENZ GISELA

IPC: A01N37/50 ,  A01N43/54 ,  A01N43/58 ,  A01N43/76 ,  A01N43/836 ,  C07C69/65 ,  C07C69/653 ,  C07C69/734 ,  C07C69/738 ,  C07C251/48 ,  C07C251/50 ,  C07C251/52 ,  C07C251/54 ,  C07C251/56 ,  C07C251/58 ,  C07C251/60 ,  C07C251/86 ,  C07C255/15 ,  C07C255/57 ,  C07C255/58 ,  C07C255/62 ,  C07D213/77 ,  C07D239/42 ,  C07D241/20 ,  C07D263/32 ,  C07D333/28 ,  A01N33/26 ,  A01N33/16 ,  C07D213/30 ,  C07D213/61 ,  C07D213/26 ,  C07D213/80 ,  C07D213/50 ,  C07D241/12 ,  C07D241/42 ,  C07D237/08 ,  C07D207/14 ,  C07D333/56 ,  C07D261/08 ,  C07D261/10 ,  C07D209/12 ,  C07D213/42 ,  C07D303/36 ,  C07D303/48 ,  C07D303/08 ,  C07D285/10 ,  C07D285/12 ,  C07D239/26 ,  C07D239/74

Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).