公开(公告)号：AU778913B2

公开(公告)日：2004-12-23

申请号：AU7056401

申请日：2001-06-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

公开(公告)号：ZA200210070B

公开(公告)日：2003-12-12

申请号：ZA200210070

申请日：2002-12-12

Applicant: BASF AG

Inventor： HEFFERNAN GAVIN ,  PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR

IPC: A01N20060101 ,  A01N43/54 ,  C07D20060101 ,  C07D239/48 ,  C07D401/04 ,  C07D ,  A01N

公开(公告)号：HU0300649A2

公开(公告)日：2003-07-28

申请号：HU0300649

申请日：2001-06-11

Applicant: BASF AG

Inventor： HEFFERNAN GAVIN ,  PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

公开(公告)号：SK17452002A3

公开(公告)日：2003-06-03

申请号：SK17452002

申请日：2001-06-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

公开(公告)号：CZ20024041A3

公开(公告)日：2003-04-16

申请号：CZ20024041

申请日：2001-06-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

公开(公告)号：BR0111594A

公开(公告)日：2003-04-15

申请号：BR0111594

申请日：2001-06-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

公开(公告)号：AU7056401A

公开(公告)日：2001-12-24

申请号：AU7056401

申请日：2001-06-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.