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    AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES
    1.
    发明申请
    AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES 审中-公开
    氨基取代的苯并（杂环）环状衍生物

    公开(公告)号：WO2004080170A3

    公开(公告)日：2004-11-04

    申请号：PCT/EP2004001677

    申请日：2004-02-20

    Applicant: BASF AG ,  STEINER GERD ,  SCHMIDT THOMAS ,  KORDES MARKUS ,  DEYN WOLFGANG VON ,  HOFMANN MICHAEL ,  BAUMANN ERNEST ,  PUHL MICHAEL ,  HEFFERNAN GAVIN ,  CULBERTSON DEBORAH L ,  TREACY MICHAEL F

    Inventor： STEINER GERD ,  SCHMIDT THOMAS ,  KORDES MARKUS ,  VON DEYN WOLFGANG ,  HOFMANN MICHAEL ,  BAUMANN ERNEST ,  PUHL MICHAEL ,  HEFFERNAN GAVIN ,  CULBERTSON DEBORAH L ,  TREACY MICHAEL F

    IPC: A01N43/60 ,  A01N43/72

    CPC classification number: A01N43/72 ,  A01N43/60

    Abstract: Use of compounds Formula (I), A = a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R = OH, SH, NH2, CN, NO2, halogen, C1-C6-alkyl, C1-C6-haloalkyl; C1-C6- alkoxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C2-C6-alkenyl, C2-C6-alkenyloxy, C2-C6-alkenylthio, C2-C6-alkynyl, C2-C6­alkynyloxy, C2-C6-alkynylthio, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C2-C6-alkenylsulfonyl, C2-C6-alkynylsulfoxyl, C1-C6-alkylcarbonyl, C1-C6- alkoxycarbonyl, C1-C6-alkylcarbonyloxy; R = C1-C6-alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C1-C6-alkylene or C1-C6-alkyleneoxy linkage to A or fused to A and which may be substituted; R , R = H, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylamino, C1-C6-alkoxy, C3-C6 cycloalkyl, or R and R together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system con-taining 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitro-gen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R and R together form the chains -(CH2)2N (O-)(CH2)2- or -(CH2)3N (O )(CH2)2 ; m = 0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.

    Abstract translation: 式（I）化合物的用途，A =可含有1-3个杂原子且可以是饱和或部分或完全不饱和的5至7元环; R 1 = OH，SH，NH 2，CN，NO 2，卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基; C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基，C 1 -C 6卤代烷硫基，C 2 -C 6烯基，C 2 -C 6烯氧基，C 2 -C 6烯硫基， C 1 -C 6烷基磺酰基，C 1 -C 6烷基亚磺酰基，C 2 -C 6烯基磺酰基，C 2 -C 6炔基亚磺酰基，C 1 -C 6烷基羰基，C 1 -C 6烷氧基羰基， R 2 = C 1 -C 6烷基或可含有1至4个杂原子并且直接键合或通过O，S，C 1 -C 6亚烷基键合的单环或双环5至10元芳环体系或 与A相连的C1-C6-亚烷氧基键或者与A相连并可以被取代的; R 3，R 4 = H，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷基氨基，C 1 -C 6烷氧基，C 3 -C 6环烷基或R 3和 R 4与它们所连接的氮原子一起形成饱和或部分饱和的含有1至3个杂原子的5至10元环系统或含有1至4个硝基的5元杂芳基 其中环系统中的碳和/或氮原子可以被取代或者可以被取代的苯基或苄基; 或者R 3和R 4一起形成链 - （CH 2）2 N +（O-）（CH 2）2 - 或 - （CH 2）3 N +（O-）（CH 2）2 < - >; m = 0至4; n是0至4; 以及用于防治昆虫，蛛形纲动物或线虫的对映异构体，非对映异构体，顺式/反式异构体或其盐，控制这些害虫的方法以及通过施用农药有效量的式（I）化合物来保护生长中的植物对这些害虫的侵袭或侵染 （I），制备它们的方法以及包含它们的组合物。

    FUNGICIDAL 5-PHENYL SUBSTITUTED 2-(CYANOAMINO) PYRIMIDINES
    2.
    发明专利
    FUNGICIDAL 5-PHENYL SUBSTITUTED 2-(CYANOAMINO) PYRIMIDINES 未知

    公开(公告)号：CA2412010A1

    公开(公告)日：2001-12-20

    申请号：CA2412010

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： PEES KLAUS-JUERGEN ,  HEFFERNAN GAVIN ,  PFRENGLE WALDEMAR

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

    Abstract: Pyrimidines of formula (I) in which R1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- o r 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to fo ur nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxycarbonyl, wherein R1 groups are unsubstituted or substituted as defined in the specification; R2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstitute d or substituted; R4 represents hydrogen or alkyl, alkenyl or alkynyl; which a re unsubstituted or substituted; and X represents O, S, NR5 or a single bond, wherein R5 represents hydrogen or alkyl; or R1 and R5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

    3.
    发明专利
    未知

    公开(公告)号：DE60113104D1

    公开(公告)日：2005-10-06

    申请号：DE60113104

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04 ,  C07D39/48 ,  C07D01/04

    Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

    2-(CIANOAMINO)PIRIMIDINAS SUBSTITUIDAS CON 5-FENILO FUNGICIDAS.
    4.
    发明专利
    2-(CIANOAMINO)PIRIMIDINAS SUBSTITUIDAS CON 5-FENILO FUNGICIDAS. 未知

    公开(公告)号：MXPA02012073A

    公开(公告)日：2003-04-25

    申请号：MXPA02012073

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： HEFFERNAN GAVIN

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

    Abstract: Las pirimidinas de la formula I; (Ver formula) en la cual R1 representa hidrogeno o alquilo, haloalquilo, alquenilo, alquinilo, alcadienilo, alcoxi, cicloalquilo, fenilo, o heteroarilo con 6 o 5 miembros o heterociclilo con 6 o 5 miembros, que contiene uno a cuatro atomos de nitrogeno o uno a tres atomos de nitrogeno y un atomo de azufre o un atomo de oxigeno, o tri-alquilo-sililo, formilo o alcoxicarbonilo, en donde los grupos R1 estan no sustituidos o sustituidos como se define en la descripcion; R2 representa fenilo, cicloalquilo o heteroarilo con 5 o 6 miembros, que contiene uno a cuatro atomos de nitrogeno o uno a tres atomos de nitrogeno y un atomo de azufre o atomo de oxigeno, los cuales son no sustituidos o sustituidos; R3 representa hidrogeno, halogeno o alquilo, alcoxi, alquiltio, alquilamino o di-alquilamino; los cuales estan no sustituidos o sustituidos; R4 representa hidrogeno o alquilo, alquenilo o alquinilo, los cuales estan no sustituidos o sustituidos, y X representa O, S, NR5 o un enlace unico, en donde R5 representa hidrogeno o alquilo; o R1 y R5 junto con el atomo de nitrogeno interyacente forman un anillo heterociclico; procesos e intermediarios para preparar estos compuestos, a composiciones que los comprenden y a su uso para controlar hongos nocivos.

    2-(CIANOAMINO)PIRIMIDINAS 5-FENIL-SUSTITUIDAS FUNGICIDAS.
    5.
    发明专利
    2-(CIANOAMINO)PIRIMIDINAS 5-FENIL-SUSTITUIDAS FUNGICIDAS. 未知

    公开(公告)号：ES2246330T3

    公开(公告)日：2006-02-16

    申请号：ES01949398

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

    Abstract: Pirimidinas de **fórmula** en donde R1 representa alquilo C1-C10, haloalquilo C1-C10, alquenilo C2-C6, alquinilo C2-C6, alcadienilo C4-C8, alcoxi C1-C10, cicloalquilo C3-C8, fenilo o heteroarilo de 5 o 6 miembros o heterociclilo de 5 o 6 miembros, que contiene de uno a cuatro átomos de nitrógeno o de uno a tres átomos de nitrógeno y un átomo de azufre u oxígeno, o tri-alquil(C1-C6)-sililo, formilo o alcoxi(C1- C10)carbonilo; en donde los grupos R1 están insustituidos o sustituidos por uno a tres grupos Ra Ra es halógeno, nitro, ciano, hidroxi o alquilo C1-C10, cicloalquilo C3-C6, cicloalquenilo C3-C6, haloalquilo C1-C10, halocicloalquilo C3-C6, alcoxi C1-C10, haloalcoxi C1-C10, alcoxi(C1- C6)carbonilo, tri-alquil(C1-C4)-sililo, fenilo, halo- o dihalo-fenilo o heteroarilo de 5 o 6 miembros, que contiene de uno a cuatro átomos de nitrógeno o de uno a tres átomos de nitrógeno y un átomo de azufre u oxígeno; R2 representa fenilo, cicloalquilo C3-C6 o heteroarilo de 5 o 6 miembros, que contienede uno a cuatro átomos de nitrógeno o de uno a tres átomos de nitrógeno o un átomo de azufre u oxígeno que están insustituidos o sustituidos por uno a tres grupos Ra.

    FUNGICIDAL 5-PHENYL SUBSTITUTED 2-(CYANOAMINO) PYRIMIDINES
    6.
    发明专利
    FUNGICIDAL 5-PHENYL SUBSTITUTED 2-(CYANOAMINO) PYRIMIDINES 未知

    公开(公告)号：PL362551A1

    公开(公告)日：2004-11-02

    申请号：PL36255101

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

    Abstract: Pyrimidines of formula I in which R 1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R 1 groups are unsubstituted or substituted as defined in the specification; R 2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R 3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R 4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR 5 or a single bond, wherein R 5 represents hydrogen or alkyl; or R 1 and R 5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.

    8.
    发明专利
    未知

    公开(公告)号：BRPI0408188A

    公开(公告)日：2006-04-04

    申请号：BRPI0408188

    申请日：2004-02-20

    Applicant: BASF AG

    Inventor： STEINER GERD ,  SCHMIDT THOMAS ,  KORDES MARKUS ,  DEYN WOLFGANG VON ,  HOFMANN MICHAEL ,  BAUMANN ERNST ,  PUHL MICHAEL ,  HEFFERNAN GAVIN ,  CULBERTSON DEBORAH L ,  TREACY MICHAEL F

    IPC: A01N43/60 ,  A01N43/72

    Abstract: Use of compounds Formula (I), A=a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R 1 -OH, SH, NH 2 , CN, NO 2 , halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl; C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, C 2 -C 6 -alkenyl, C 2 -C 6 alkenyloxy, C 2 -C 6 -alkenylthio, C 2 -C 6 -alkynyl, C 2 -C 6 -alkynyloxy, C 2 -C 6 -alkynylthio, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 -alkylsulfoxyl, C 2 -C 6 -alkenylsulfonyl, C 2 -C 6 -alkylsulfoxyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkoxycarbonyl, C 1 -C 6 -aklylcarbonyloxy; R 2 -C 1 -C 6 -alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C 1 -C 6 -alkylene or C 1 -C 6 -alkyleneoxy linkage to A or fused to A and which may be substituted; R 3 , R 4 -H, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkyl-amino, C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl, or R 3 and R 4 together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system containing 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitrogen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R 3 and R 4 together form the chains -(CH 2 ) 2 N + (O-)(CH 2 ) 2 - or -(CH 2 ) 3 N + (O - )(CH 2 ) 2 -; m=0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.

    ФУНГИЦИДНЫЕ 5-ФЕНИЛ-ЗАМЕЩЕННЫЕ 2-(ЦИАНОАМИНО)ПИРИМИДИНЫ
    10.
    发明专利
    ФУНГИЦИДНЫЕ 5-ФЕНИЛ-ЗАМЕЩЕННЫЕ 2-(ЦИАНОАМИНО)ПИРИМИДИНЫ 未知

    公开(公告)号：EA005927B1

    公开(公告)日：2005-08-25

    申请号：EA200201253

    申请日：2001-06-11

    Applicant: BASF AG

    Inventor： PEES KLAUS-JUERGEN ,  PFRENGLE WALDEMAR ,  HEFFERNAN GAVIN

    IPC: C07D239/42 ,  A01N43/54 ,  A01N47/40 ,  A61K31/519 ,  C07D239/48 ,  C07D401/04 ,  C07D409/12 ,  C07D487/04

    Abstract: Пиримидиныформулы (I)вкоторой Rозначает C-C-алкил, C-C-галоалкил, C-C-алкенил, C-C-алкинил, C-C-алкадиенил, C-C-алкокси, C-C-циклоалкил, фенилилитри-C-C-алкилсилил, формилили C-C-алкоксикарбонил;причемгруппы Rнезамещеныилизамещены 1-3 группами R, приэтом Rозначаетгалоген, нитрогруппу, цианогруппу, гидроксигруппуили C-C-алкил, C-C-циклоалкил, C-C-циклоалкенил, C-C-галоалкил, C-C-галоциклоалкил, C-C-алкокси, C-C-галоалкокси, C-C-алкоксикарбонил, три-C-C-алкилсилил, фенил, гало- илидигалофенилили 5- или 6-членныйгетероарил, содержащий 1-4 атомаазотаили 1-3 атомаазотаи одинатомсерыиликислорода;Rозначаетфенил, необязательнозамещенный 1-3 группами, выбраннымиизгалогена, C-C-алкилаи C-C-алкокси;Rозначаетгалоген;Rозначает C-C-алкил, C-C-алкенилили C-C-алкинил, незамещенныеилизамещенные 1-3 группами R; иХозначаетО, S, NRилипростуюсвязь, причем Rпредставляетсобойводородили C-C-алкил; илиRи Rвместес размещенныммеждунимиатомомазотаобразуютгетероцикл, такойкакпиперидинилиазепан, необязательнозамещенныеоднойилинесколькими C-C-алкильнымигруппами.Визобретениитакжеописаныспособыи промежуточныесоединениядляполученияданныхсоединений, композиции, содержащиеданныесоединения, иприменениеданныхсоединенийдляборьбыс фитопатогеннымигрибами.

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