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    PROCEDIMIENTO PARA LA PREPARACION DE AMIDAS Y ESTERES HETEROARIL-CARBOXILICOS.
    13.
    发明专利
    PROCEDIMIENTO PARA LA PREPARACION DE AMIDAS Y ESTERES HETEROARIL-CARBOXILICOS. 未知

    公开(公告)号：ES2241102T3

    公开(公告)日：2005-10-16

    申请号：ES98306530

    申请日：1998-08-17

    Applicant: BASF AG

    Inventor： KNELL MARCUS ,  BRINK MONIKA ,  WEVERS JAN HENDRIK ,  HEINZ WILLI

    IPC: C07D213/79 ,  C07D20060101 ,  C07D213/00 ,  C07D213/02 ,  C07D213/04 ,  C07D213/60 ,  C07D213/78 ,  C07D213/80 ,  C07D213/803 ,  C07D213/81 ,  C07D213/82 ,  C07D401/12 ,  C07D401/14 ,  C07D403/00

    Abstract: LA PRESENTE INVENCION SE REFIERE A UN PROCEDIMIENTO DE PREPARACION DE AMIDAS Y ESTERES HETEROARILCARBOXILICOS DE FORMULA I: DONDE DESDE A 1 HASTA A 5 , R 1 , HAL Y X REPRESENTAN: UNO O DOS DE LOS GRUPOS ENTRE A 1 , A 2 , A SUP,3 , A 4 Y A 5 REPRESENTAN UN ATOMO DE NITROGENO Y LOS DEMAS GRUPOS, CADA UNO INDEPENDIENTEMENTE, REPRESENTAN CR 3 , HAL REPRESENTA UN ATOMO DE HALOGENO, X REPRESENTA OX IGENO O NR 2 , R 1 REPRESENTA UN GRUPO CICLOALQUILO, HETEROARILO, ARILO O ALQUILO, OPCIONALMENTE SUSTITUIDO, R 2 REPRESENTA UN ATOMO DE HIDROGENO O UN GRUPO ALQUILO, O R SUP,1 Y R 2 FORMAN CONJUNTAMENTE CON EL CICLO INTERYACENTE, UN GRUPO HETEROCICLICO, Y R 3 CADA UNO INDEPENDIENTEMENTE, REPRESENTA UN ATOMO DE HIDROGENO O UN GRUPO ALQUILO, DICHO PROCEDIMIENTO CONSISTE EN CALENTAR LA MEZCLA, COMPUESTA FUNDAMENTALMENTE POR UN COMPUESTO HETEROARILTRICLOROMETANO DE FORMULA II: EN LA QUE DE A 1 A A 5 Y HAL, SON TAL Y COMO SE LOS DESCRIBIO ANTERIORMENTE, Y DE 1,0 A 1,5 EQUIVALENTES DE ACIDO SULFURICO CONCENTRADO, Y HACIENDO REACCIONAR EL PRODUCTO INTERMEDIO RESULTANTE CON UN ALCOHOL O AMINA DE FORMULA III: OPCIONALMENTE EN PRESENCIA DE UN DILUYENTE Y/O UNA BASE.

    14.
    发明专利
    未知

    公开(公告)号：DK0899262T3

    公开(公告)日：2005-06-20

    申请号：DK98306530

    申请日：1998-08-17

    Applicant: BASF AG

    Inventor： BRINK MONIKA ,  KNELL MARCUS ,  WEVERS JAN HENDRIK ,  HEINZ WILLI

    IPC: C07D213/79 ,  C07D20060101 ,  C07D213/00 ,  C07D213/02 ,  C07D213/04 ,  C07D213/60 ,  C07D213/78 ,  C07D213/80 ,  C07D213/803 ,  C07D213/81 ,  C07D213/82 ,  C07D401/12 ,  C07D401/14 ,  C07D403/00

    Abstract: The invention relates to a process for the preparation of heteroarylcarboxylic amides and esters of formula I in which A through A , R , Hal and X one or two of the groups A , A , A , A and A represent a nitrogen atom and the other groups each independently represent CR , Hal represents a halogen atom, X represents oxygen or NR , R1 represents an optionally substituted alkyl, aryl, heteroaryl or cycloalkyl group, R represents a hydrogen atom or an alkyl group, or R and R together with the interjacent ring form a heterocyclic group, and R each independently represent a hydrogen atom or an alkyl group, which comprises: heating a mixture consisting essentially of heteroaryltrichloromethane compound of formula II, in which A through A and Hal are as hereinbefore defined, and 1.0 to 1.5 equivalents of concentrated sulfuric acid, and reacting the resulting intermediate product with an alcohol or amine of formula III HXR optionally in the presence of a diluent and/or a base.

    15.
    发明专利
    未知

    公开(公告)号：DE69829613D1

    公开(公告)日：2005-05-12

    申请号：DE69829613

    申请日：1998-08-17

    Applicant: BASF AG

    Inventor： KNELL MARCUS ,  BRINK MONIKA ,  WEVERS JAN HENDRIK ,  HEINZ WILLI

    IPC: C07D213/79 ,  C07D20060101 ,  C07D213/00 ,  C07D213/02 ,  C07D213/04 ,  C07D213/60 ,  C07D213/78 ,  C07D213/80 ,  C07D213/803 ,  C07D213/81 ,  C07D213/82 ,  C07D401/12 ,  C07D401/14 ,  C07D403/00

    Abstract: The invention relates to a process for the preparation of heteroarylcarboxylic amides and esters of formula I in which A through A , R , Hal and X one or two of the groups A , A , A , A and A represent a nitrogen atom and the other groups each independently represent CR , Hal represents a halogen atom, X represents oxygen or NR , R1 represents an optionally substituted alkyl, aryl, heteroaryl or cycloalkyl group, R represents a hydrogen atom or an alkyl group, or R and R together with the interjacent ring form a heterocyclic group, and R each independently represent a hydrogen atom or an alkyl group, which comprises: heating a mixture consisting essentially of heteroaryltrichloromethane compound of formula II, in which A through A and Hal are as hereinbefore defined, and 1.0 to 1.5 equivalents of concentrated sulfuric acid, and reacting the resulting intermediate product with an alcohol or amine of formula III HXR optionally in the presence of a diluent and/or a base.

    16.
    发明专利
    未知

    公开(公告)号：DE69829613T2

    公开(公告)日：2005-09-15

    申请号：DE69829613

    申请日：1998-08-17

    Applicant: BASF AG

    Inventor： KNELL MARCUS ,  BRINK MONIKA ,  WEVERS JAN HENDRIK ,  HEINZ WILLI

    IPC: C07D213/79 ,  C07D20060101 ,  C07D213/00 ,  C07D213/02 ,  C07D213/04 ,  C07D213/60 ,  C07D213/78 ,  C07D213/80 ,  C07D213/803 ,  C07D213/81 ,  C07D213/82 ,  C07D401/12 ,  C07D401/14 ,  C07D403/00

    Abstract: The invention relates to a process for the preparation of heteroarylcarboxylic amides and esters of formula I in which A through A , R , Hal and X one or two of the groups A , A , A , A and A represent a nitrogen atom and the other groups each independently represent CR , Hal represents a halogen atom, X represents oxygen or NR , R1 represents an optionally substituted alkyl, aryl, heteroaryl or cycloalkyl group, R represents a hydrogen atom or an alkyl group, or R and R together with the interjacent ring form a heterocyclic group, and R each independently represent a hydrogen atom or an alkyl group, which comprises: heating a mixture consisting essentially of heteroaryltrichloromethane compound of formula II, in which A through A and Hal are as hereinbefore defined, and 1.0 to 1.5 equivalents of concentrated sulfuric acid, and reacting the resulting intermediate product with an alcohol or amine of formula III HXR optionally in the presence of a diluent and/or a base.

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