公开(公告)号：JPS5549359A

公开(公告)日：1980-04-09

申请号：JP12427779

申请日：1979-09-28

Applicant: BASF AG

Inventor： RENTZEA COSTIN ,  SAUTER HUBERT ,  ZEEH BERND ,  HEILEN GERD ,  JUNG JOHANN

IPC: A01N43/64 ,  A01N43/653 ,  C07D249/08 ,  C07D405/06 ,  C07D409/06 ,  C07D521/00

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9920615A3

公开(公告)日：1999-06-24

申请号：PCT/EP9806299

申请日：1998-10-05

Applicant: BASF AG ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： BAYER HERBERT ,  GEWEHR MARKUS ,  GROTE THOMAS ,  MUELLER BERND ,  SAUTER HUBERT ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  PTOCK ARNE ,  GOETZ ROLAND ,  RACK MICHAEL ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  HARRIES VOLKER ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/82 ,  A01N43/836 ,  C07C259/14 ,  C07C265/12 ,  C07D271/06 ,  C07D271/07 ,  C07D413/12 ,  C07C239/12 ,  C07C251/38 ,  C07D413/14

CPC classification number: C07D271/07 ,  A01N43/82 ,  C07C259/14 ,  C07C265/12 ,  C07D413/12

Abstract: The invention relates to substituted phenyl carbamates of formula (I), wherein E represents a group A or B, # characterises the bond with the phenyl ring, and R , R , Y, n, T, and Z have the meanings given in the description.

Abstract translation: 本发明涉及式（I），其中E是基团A或B，其中＃为键合到苯基环的特征的取代的苯基氨基甲酸酯，且R <阿尔法>，R <克（B）>，Y，N，T 和Z具有描述中给出的含义。

公开(公告)号：WO9608969A3

公开(公告)日：1996-06-06

申请号：PCT/EP9503557

申请日：1995-09-09

Applicant: BASF AG ,  RETZLAFF GUENTER ,  KOEHLE HARALD ,  SAUTER HUBERT ,  BAYER HERBERT ,  KIRSTGEN REINHARD

Inventor： RETZLAFF GUENTER ,  KOEHLE HARALD ,  SAUTER HUBERT ,  BAYER HERBERT ,  KIRSTGEN REINHARD

IPC: A01N35/10 ,  A01N37/38 ,  A01N37/50 ,  A01N61/00 ,  A01N37/10 ,  A01N37/18 ,  A01N37/36 ,  A01N37/44 ,  A01N43/02 ,  A01N43/36 ,  A01N43/40 ,  A01N43/48 ,  A01N43/64 ,  A01N43/66 ,  A01N47/20 ,  A01N47/30

CPC classification number: A01N35/10 ,  A01N37/38 ,  A01N37/50 ,  A01N61/00

Abstract: A process is disclosed for increasing agricultural plant harvests. The plants are treated with an active substance that inhibits the mitochondrial breathing chain at the level of the b/c1 complex.

公开(公告)号：WO0195721A3

公开(公告)日：2002-04-25

申请号：PCT/EP0106686

申请日：2001-06-13

Applicant: BASF AG ,  GRAMMENOS WASILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

Inventor： GRAMMENOS WASILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMAN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIGFRIED

IPC: A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22 ,  C07C233/69

CPC classification number: A01N37/36 ,  A01N37/18 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22

Abstract: The invention relates to the use of phenethyl acrylamides of formula (I) for controlling phytopathogenic fungi, wherein the substituents of said phenethyl acrylamides have the following significations: X signifies halogen, alkyl, halogenalkyl, alkoxy halogenalkoxy and -O-C(Ra, Rb)-C C-R?6; Ra, Rb and Rc¿ have the signification given in the description; m, n independently signify 1 to 4, the radicals X or Y being potentially different if m or n is higher than 1; Y signifies halogen, nitro, cyano, alkyl, CF¿3?, alkoxy and phenyl; R?1, R2¿ independently signify hydrogen, halogen, alkyl, alkoxy, halogenalkoxy and CF¿3?; R?3, R4, R5, and R6¿ independently signify hydrogen, alkyl and alkoxy, or R?3 and R4¿ together form a cyclopropyl ring, whereby the C-R5 and C-R6 bonds can be in position E or Z in relation to each other. The invention also relates to novel phenethyl acrylamides, a method for the production thereof, and agents containing the same.

公开(公告)号：WO9959982A3

公开(公告)日：2000-03-16

申请号：PCT/EP9903003

申请日：1999-05-04

Applicant: BASF AG ,  BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

Inventor： BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

IPC: C07C251/38 ,  A01N37/40 ,  C07C49/303 ,  C07C251/42 ,  C07C251/50 ,  C07C251/52 ,  C07C251/60 ,  A01N37/50 ,  C07C49/35

CPC classification number: C07C251/60 ,  C07C2601/14

Abstract: The invention relates to bisoximether derivatives of formula (I) in which the variables have the following meanings: R represents halogen, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or C1-C4 alkoxy halide; n is 1 to 5, whereby the radicals R can be different if n is not equal to 1; R represents C1-C4 alkyl, C3-C6 alkenyl or C3-C6 alkynyl, whereby these groups can be partially or completely halogenated; Q represents C(=CHOCH3)-COOCH3, C(=CHCH3)-COOCH3, C(=NOCH3)-COOCH3 or C(=NOCH3)-CONHCH3. The invention also relates to the salts of the bisoximether derivatives, to methods and intermediate products for the production of these compounds and to their use for combating animal pests and fungicidal pests.

Abstract translation: 式（I），其中各变量具有以下含义的双肟醚衍生物，R <1>为卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基; n为1至5，其中基团可以是与R <1>不同的，当n不为1; [R <2> C1-C4烷基，C3-C6链烯基或C3-C6炔基，其中这些基团可以部分或完全被卤代; Q为C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3）-COOCH 3或C（= NOCH 3）-CONHCH 3; 和它们的盐，方法和中间体制备这些化合物和它们用于控制动物害虫和有害真菌中的用途。

公开(公告)号：WO9010006A3

公开(公告)日：1990-11-01

申请号：PCT/EP9000280

申请日：1990-02-20

Applicant: BASF AG

Inventor： DAUM LOTHAR ,  KEILHAUER GERHARD ,  SAUTER HUBERT ,  BERTRAM GUNDA ,  ANKE TIMM ,  WEBER WOLFGANG ,  STEGLICH WOLFGANG

IPC: C07D319/14 ,  A61K31/335 ,  A61K31/357 ,  A61P31/04 ,  C07D407/12 ,  C07D493/10

CPC classification number: C07D407/12 ,  C07D493/10

Abstract: β-methoxyacrylates of formula (I), in which R?1, R2 and R3¿ have the meanings given in the description, are useful for treating diseases. Their production is also described.

公开(公告)号：WO0238565A3

公开(公告)日：2003-10-09

申请号：PCT/EP0112977

申请日：2001-11-09

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.

Abstract translation: 7-（R）式（I）的-aminotriazolopyrimidine其中取代基和指数具有以下含义：R t <1>是氢或甲基; [R <2>是甲基; [R <3> C2-C10烷基，C1-C4烷氧基，C3-C10环烷基; [R <4>为卤素，C1-C4烷基，C1-C4卤代烷基或C1-C4烷氧基; n是从1到5的数; Y是卤素，氰基，C1-C4烷基或C1-C4烷氧基; 其中*是R构型的手性中心。 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9940082A3

公开(公告)日：1999-10-21

申请号：PCT/EP9900470

申请日：1999-01-26

Applicant: BASF AG ,  PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

Inventor： PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D401/12 ,  C07D401/14 ,  A01N43/48

CPC classification number: C07D401/12 ,  A01N43/56

Abstract: The present invention relates to compounds of the general formula (I) and to the salts thereof, wherein the substituents and the n index have the following values: Q represents -C(=CHCH3)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-CONH(CH3); R represents hydrogen, halogen, C1-C4 alkyl, C1-C2 halogenalkyl, C1-C4 alkoxy or C1-C2 halogenalkoxy; R represents halogen, C1-C4 alkyl, C1-C2 halogenalkyl or C1-C4 alkoxy; n is 0, 1 or 2, wherein the R substituents can be different when n = 2; and R represents phenyl, pyridyle or pyrimidyle. This invention also relates to agents containing these compounds as well as to the use of said compounds (I) and agents against noxious fungi and animal parasites.

Abstract translation: 通式（I）和它们的盐，其中取代基和指数n具有以下含义的化合物：Q是-C（= CHCH 3）-COOCH 3，-C（= CHOCH 3）-COOCH 3，C（= NOCH 3） - COOCH 3或-C（= NOCH 3）-CONH（CH 3）; R 1是氢，卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基或C 1 -C 2卤代烷氧基; R 2是卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基; n是0,1或2，其中当n = 2时取代基R 2可以不同; R 3苯基，吡啶基或嘧啶基，含有它们的试剂以及化合物（I）和防治有害真菌和动物害虫的试剂的用途。

公开(公告)号：WO9521154A2

公开(公告)日：1995-08-10

申请号：PCT/EP9500007

申请日：1995-01-03

Applicant: BASF AG ,  BAYER HERBERT ,  SAUTER HUBERT ,  MUELLER RUTH ,  GRAMMENOS WASSILIOS ,  HARREUS ALBRECHT ,  KIRSTGEN REINHARD ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA

Inventor： BAYER HERBERT ,  SAUTER HUBERT ,  MUELLER RUTH ,  GRAMMENOS WASSILIOS ,  HARREUS ALBRECHT ,  KIRSTGEN REINHARD ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA

IPC: C07D249/08 ,  A01N37/50 ,  A01N37/52 ,  A01N43/06 ,  A01N43/36 ,  A01N43/40 ,  A01N43/54 ,  A01N43/80 ,  A01N43/82 ,  A01N43/824 ,  A01P3/00 ,  A01P7/04 ,  C07C251/38 ,  C07C251/40 ,  C07C251/48 ,  C07C251/54 ,  C07C251/56 ,  C07C251/58 ,  C07C255/11 ,  C07C327/44 ,  C07C327/48 ,  C07C327/58 ,  C07D207/32 ,  C07D207/333 ,  C07D207/36 ,  C07D213/30 ,  C07D213/53 ,  C07D213/62 ,  C07D213/64 ,  C07D213/79 ,  C07D233/64 ,  C07D237/14 ,  C07D239/34 ,  C07D239/46 ,  C07D241/18 ,  C07D261/08 ,  C07D261/10 ,  C07D263/32 ,  C07D263/34 ,  C07D271/06 ,  C07D271/10 ,  C07D277/24 ,  C07D307/42 ,  C07D333/32 ,  C07D521/00 ,  C07C251/44 ,  C07C251/52 ,  C07D261/12 ,  C07D263/18 ,  C07D307/58

CPC classification number: C07D207/333 ,  A01N37/50 ,  A01N37/52 ,  A01N43/06 ,  A01N43/36 ,  A01N43/40 ,  A01N43/54 ,  A01N43/80 ,  A01N43/82 ,  C07C251/58 ,  C07C255/11 ,  C07C327/48 ,  C07C327/58 ,  C07D213/53 ,  C07D213/64 ,  C07D239/34 ,  C07D261/08 ,  C07D263/32 ,  C07D271/06 ,  C07D277/24 ,  C07D307/42

Abstract: Phenyl acetic acid derivatives of formula (I) in which the substituents and index have the following meanings: X is oxygen or sulphur; R is hydrogen and alkyl; R is hydrogen and alkyl; R is cyano, nitro, trifluoromethyl, halogen, alkyl and alkoxy; m is 0, 1 ou 2, in which the radicals R may be different if m is 2; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, halogen alkyl, alkoxy, halogen alkoxy, alkylthio, alkylamino or dialkylamino; R is hydrogen, cyano, nitro, hydroxy, amino, halogen, possibly substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkinyl, alkinyloxy, alkinylthio, alkinylamino, N-alkinyl-N-alkylamino; optionally substituted cycloalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocylcyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, n-aryl-n-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetarylamino, N-hetaryl-N-alkylamino; R is hydrogen, optionally substituted alkyl, cycloalkyl, alkenyl, alkinyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl or alkylsulfonyl; optionally substituted aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl or hetarylsulphonyl; and their salts, process and intermediate products for their production, and their use.

Abstract translation: 式I其中取代基和指数具有以下含义的苯乙酸衍生物：X是氧或硫; R是氢和烷基; [R <1>是氢和烷基; [R <2>氰基，硝基，三氟甲基，卤素，烷基和烷氧基; m是0，1或2，其中基团可以是与R <2>中，当m是2不同; [R <3>是氢，氰基，硝基，羟基，氨基，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷基氨基或二烷基氨基; [R <4>为氢，氰基，硝基，羟基，氨基，卤素，未取代或取代的。 烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，烯基，烯氧基，烯硫基，链烯基，N-链烯基 - N-烷基氨基，炔基，炔氧基，炔硫基，炔基氨基，N-炔基 - N-烷基氨基; 未取代的或取代的。 环烷基，环烷氧基，环烷硫基，环烷基氨基，N-环烷基-N-烷基氨基，环烯基，环烯氧基，环烯硫基，cycloalkenylamino，N-环烯基-N-烷基氨基，杂环基，杂环氧基，杂环硫基，杂环基氨基，N-Heterocylcyl-N-烷基氨基，芳基， 芳氧基，芳硫基，芳基氨基，N-芳基-N-烷基氨基，杂芳基，杂芳氧基，杂芳硫基，Hetarylamino，N-杂芳基的N-烷基氨基; [R <5>氢，未取代或取代的。 烷基，环烷基，烯基，炔基，烷基羰基，烯基羰基，炔基羰基或烷基磺酰基; 未取代的或取代的。 芳基，芳基羰基，芳基磺酰基，杂芳基，或hetarylcarbonyl hetarylsulfonyl; 和它们的盐，过程和它们的制备方法和它们的使用的中间体。