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    N-ACYLIMINO HETEROCYCLIC COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS
    11.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS 审中-公开

    公开(公告)号：US20180179177A1

    公开(公告)日：2018-06-28

    申请号：US15128625

    申请日：2015-03-26

    Applicant: BASF SE

    Inventor： Birgit GOCKEL ,  Martin John McLAUGHLIN ,  Karsten KOERBER ,  Wolfgang VON DEYN ,  Jochen DIETZ ,  Matthias POHLMAN ,  Kenichi KOJIMA

    IPC: C07D401/06 ,  C07D405/06 ,  C07D417/06 ,  A01N43/40 ,  A01N43/78 ,  A61P33/00

    CPC classification number: C07D401/06 ,  A01N43/40 ,  A01N43/78 ,  A61P33/00 ,  C07D405/06 ,  C07D411/06 ,  C07D417/06

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. or R3 and R4a may also form a double bound, R5 may be hydrogen, halogen, CN, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl, C2-C6-alkenyl, C2-C6-alkynyl, C2-C6-alkenylthio, C2-C6-alkenylsulfinyl, C2-C6-alkenylsulfonyl, C2-C6-alkynyl, C2-C6-alkynylthio, C2-C6-alkynylsulfinyl, C2-C6-alkynylsulfonyl, etc. R3 and R5 together may also form with the carbon atom they are bound to, a 3-, 4-, 5- or 6-membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Process for Preparing Sulfimines and Their in-situ Conversion into N-(1-Amino-Benzoyl)-Sulfimines
    19.
    发明申请
    Process for Preparing Sulfimines and Their in-situ Conversion into N-(1-Amino-Benzoyl)-Sulfimines 审中-公开
    制备亚磺酰亚胺及其原位转化成N-（1-氨基 - 苯甲酰基） - 亚磺酰胺的方法

    公开(公告)号：US20160046572A1

    公开(公告)日：2016-02-18

    申请号：US14778771

    申请日：2014-03-27

    Applicant: BASF SE

    Inventor： Timo FRASSETTO ,  Harald JOCKERS ,  Christopher KORADIN ,  Thomas ZIERKE ,  Karsten KOERBER

    IPC: C07C381/10 ,  C07D401/04

    CPC classification number: C07C381/10 ,  A01N37/28 ,  A01N43/56 ,  C07C2601/02 ,  C07D401/04 ,  C07D409/14

    Abstract: The present invention relates to a process for preparing a compound of the formulae (Ia) or (Ib), or a mixture thereof, wherein R1 and R2 independently of one another are hydrogen, C1-C10-alkyl, C1-C10-haloalkyl, C3-C10-cycloalkyl, C3-C10-halocycloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl or together represent an aliphatic chain, or the like; A− is HSO4− or 1/2 SO42−; the process comprising the reaction of a sulfide of formula SR1R2 with hydroxylamineO-sulfonic acid of formula; wherein the reaction is carried out in an aqueous medium in the presence of a base. The present invention also relates to a process for preparing a compound of the formula (IV), wherein R3 is halogen, cyano, C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C2-C8-alkenyl, C2-C8-haloalkenyl, C1-C8-alkoxy, phenyl, or the like; R4 is hydrogen, C1-C10-alkyl, C1-C10-haloalkyl, C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl, phenyl, or the like; p is 0, 1, 2, 3 or 4; the process comprising: (i) providing the compound of the formulae (Ia) or (Ib), or a mixture thereof, (ii) reacting a compound of the formulae (Ia) or (Ib), or a mixture thereof, obtained in step (i) with a compound of the formula (V) in the presence of a base,

    Abstract translation: 本发明涉及制备式（Ia）或（Ib）化合物或其混合物的方法，其中R 1和R 2彼此独立地是氢，C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基， C 3 -C 10 - 环烷基，C 3 -C 10 - 卤代环烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基或一起代表脂族链等; A-是HSO4-或1/2 SO42-; 该方法包括式SR 1 R 2的硫化物与式的羟胺O-磺酸的反应; 其中反应在碱的存在下在水性介质中进行。 本发明还涉及制备式（IV）化合物的方法，其中R 3是卤素，氰基，C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代环烷基， C 2 -C 8 - 烯基，C 2 -C 8 - 卤代烯基，C 1 -C 8 - 烷氧基，苯基等; R4是氢，C1-C10-烷基，C1-C10-卤代烷基，C3-C8-环烷基，C3-C8-卤代环烷基，C2-C10-烯基，C2-C10-卤代烯基，苯基等; p是0，1，2，3或4; 该方法包括：（i）提供式（Ia）或（Ib）化合物或其混合物，（ii）使式（Ia）或（Ib）化合物或其混合物 步骤（i）与式（Ⅴ）化合物在碱的存在下反应，

    PROCESS FOR PREPARATION OF BENZYLIC AMIDES
    20.
    发明申请
    PROCESS FOR PREPARATION OF BENZYLIC AMIDES 审中-公开

    公开(公告)号：US20190382362A1

    公开(公告)日：2019-12-19

    申请号：US16480407

    申请日：2018-01-16

    Applicant: BASF SE

    Inventor： Martin John MCLAUGHLIN ,  Karsten KOERBER ,  Birgit GOCKEL ,  Devendra VYAS ,  Arun NARINE

    IPC: C07D307/79

    Abstract: The present invention relates to a process for preparing benzylic amides of formula I wherein the variables have the meaning as defined in the description, by reductive amidation of a nitrile of formula II wherein the variables have the meanings given for formula I, with an activated carbonyl compound of formula III, and which nitrile is obtained by reaction of a compound of formula IV with a halogen compound of formula V, wherein X is a halogen atom, preferably bromo, which halogen compound V in turn is obtained by Sandmeyer reaction of an aniline derivative of formula VI novel compounds of formula I, and processes for preparing compounds of formula XII wherein the variables have the meaning as defined in the description by condensing compounds of formula I with compounds of formula X and subjecting the resulting α,β-unsaturated ketone of formula XI to a reaction with hydroxylamine to yield compounds of formula XII.

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