N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS
    4.
    发明申请
    N-SUBSTITUTED IMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-取代的IMINO杂环化合物

    公开(公告)号:US20160326153A1

    公开(公告)日:2016-11-10

    申请号:US15105239

    申请日:2014-12-17

    Applicant: BASF SE

    Abstract: The present invention relates to N-substituted imino compound of formula (I): wherein Y is a radical Y1, Y2, Y3, Y4 or Y5, where Y1 is O—C(═X)—R3; Y2 is S—C(═X)—R3; Y3 is N(R5)—C(═X)—R3; Y4 is N(R5)—S(═O)—R4; Y5 is N(R5)—S(═O)2—R4; and where X is O or S; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, C1-C6-alkyl etc.; and where R3, R4 and R5 are as defined herein. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS
    5.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS 有权
    N-乙酰氨基杂环化合物

    公开(公告)号:US20160297793A1

    公开(公告)日:2016-10-13

    申请号:US15038272

    申请日:2014-11-21

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; Y is a single bond, O, S or NR5; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, etc.; R3 may be hydrogen, CN, C1-C6-alkyl, etc.; R4 may be of hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, Q-phenyl, Q′-O-phenyl, Q′-S-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, and the moieties Q-Het#, Q′-O-Het# and Q′-S-Het# where Het# represents a heterocyclic radical and where Q and Q′ are C1-C6-alkandiyl, C2-C6-alkendiyl, or C2-C6-alkyndiyl, and where Q may also be a single bond; R3 and R4 together may also may also a bivalent radical, selected from the group consisting of C2-C5-alkandiyl, C2-C5-alkendiyl, Q″-C1-C4-alkandiyl and Q″-C2-C4-alkendiyl, where Q″ is O or S. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明还涉及N-酰基亚氨基杂环化合物,其立体异构体,其互变异构体及其盐的用途,用于防治无脊椎动物害虫。 此外,本发明还涉及防治无脊椎害虫的方法,其包括施用这样的化合物。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS

    公开(公告)号:US20180179177A1

    公开(公告)日:2018-06-28

    申请号:US15128625

    申请日:2015-03-26

    Applicant: BASF SE

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1—W2—W3—W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. or R3 and R4a may also form a double bound, R5 may be hydrogen, halogen, CN, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl, C2-C6-alkenyl, C2-C6-alkynyl, C2-C6-alkenylthio, C2-C6-alkenylsulfinyl, C2-C6-alkenylsulfonyl, C2-C6-alkynyl, C2-C6-alkynylthio, C2-C6-alkynylsulfinyl, C2-C6-alkynylsulfonyl, etc. R3 and R5 together may also form with the carbon atom they are bound to, a 3-, 4-, 5- or 6-membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Pyrazoles for Controlling Invertebrate Pests
    8.
    发明申请
    Pyrazoles for Controlling Invertebrate Pests 有权
    吡唑类用于控制无脊椎动物害虫

    公开(公告)号:US20160345581A1

    公开(公告)日:2016-12-01

    申请号:US15114974

    申请日:2015-01-30

    Applicant: BASF SE

    CPC classification number: A01N43/58 A01N43/36 A01N43/56 C07D403/12

    Abstract: The present invention relates to novel pyrazoles of formula I. Moreover, the invention relates to processes and intermediates for preparing the pyrazoles of formula I, and also to active compound combinations comprising them, to compositions comprising them, and to their use for protecting growing plants from attack or infestation by invertebrate pests. Furthermore, the invention relates to methods of applying such compounds. The present invention also relates to seed comprising such compounds.

    Abstract translation: 本发明涉及式I的新的吡唑。此外,本发明涉及制备式I的吡唑的方法和中间体,还涉及包含它们的活性化合物组合物,包含它们的组合物及其用于保护生长植物的用途 来自无脊椎害虫的攻击或感染。 此外,本发明涉及应用这些化合物的方法。 本发明还涉及包含这种化合物的种子。

    PROCESS FOR PREPARATION OF BENZYLIC AMIDES
    9.
    发明申请

    公开(公告)号:US20190382362A1

    公开(公告)日:2019-12-19

    申请号:US16480407

    申请日:2018-01-16

    Applicant: BASF SE

    Abstract: The present invention relates to a process for preparing benzylic amides of formula I wherein the variables have the meaning as defined in the description, by reductive amidation of a nitrile of formula II wherein the variables have the meanings given for formula I, with an activated carbonyl compound of formula III, and which nitrile is obtained by reaction of a compound of formula IV with a halogen compound of formula V, wherein X is a halogen atom, preferably bromo, which halogen compound V in turn is obtained by Sandmeyer reaction of an aniline derivative of formula VI novel compounds of formula I, and processes for preparing compounds of formula XII wherein the variables have the meaning as defined in the description by condensing compounds of formula I with compounds of formula X and subjecting the resulting α,β-unsaturated ketone of formula XI to a reaction with hydroxylamine to yield compounds of formula XII.

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