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公开(公告)号:BR0010699A
公开(公告)日:2002-02-05
申请号:BR0010699
申请日:2000-04-26
Applicant: BAYER AG
Inventor: GREIF GIESELA , HABERKORN AXEL , BAASNER BERND , LIEB FOLKER , MARHOLD ALBRECHT , STOELTING JOERN
IPC: C07D491/048 , A01N43/28 , A01N43/52 , A01N43/90 , A61K31/4184 , A61P33/02 , C07D405/06 , C07D491/04 , C07D491/056
Abstract: The present invention relates to a new substituted benzimidazoles, their preparation and their use as agents against parasitic protazoa.
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22.
公开(公告)号:CZ20003871A3
公开(公告)日:2001-01-17
申请号:CZ20003871
申请日:1999-04-07
Applicant: BAYER AG
Inventor: STOLTEFUSS JUERGEN , GOLDMANN SIEGFRIED , KRAEMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF , STOELTING JOERN
IPC: C07D213/78 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/04 , C07D401/14 , C07D417/14 , A61K31/495
Abstract: The invention relates to compounds of the formule
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公开(公告)号:BR9909730A
公开(公告)日:2000-12-19
申请号:BR9909730
申请日:1999-04-07
Applicant: BAYER AG
Inventor: STOLTEFUSS JUERGEN , GOLDMANN SIEGFRIED , KRAEMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF , STOELTING JOERN
IPC: C07D213/78 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/04 , C07D401/14 , C07D417/14
Abstract: The invention relates to compounds of the formule
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公开(公告)号:DE19920551A1
公开(公告)日:2000-11-09
申请号:DE19920551
申请日:1999-05-05
Applicant: BAYER AG
Inventor: GREIF GISELA , HABERKORN AXEL , BAASNER BERND , LIEB FOLKER , MARHOLD ALBRECHT , STOELTING JOERN
IPC: C07D491/048 , A01N43/28 , A01N43/52 , A01N43/90 , A61K31/4184 , A61P33/02 , C07D405/06 , C07D491/04 , C07D491/056
Abstract: The present invention relates to novel substituted benzimidazoles, the production thereof and the use thereof as means against parasitic protozoa.
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公开(公告)号:PL193898B1
公开(公告)日:2007-03-30
申请号:PL34348199
申请日:1999-04-07
Applicant: BAYER AG
Inventor: STOLTEFUSS JUERGEN , GOLDMANN SIEGFRIED , KRAEMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF , STOELTING JOERN
IPC: C07D213/78 , A61K31/505 , C07D401/04 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/14 , C07D417/14
Abstract: The invention relates to compounds of the formule
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公开(公告)号:AT256124T
公开(公告)日:2003-12-15
申请号:AT00938613
申请日:2000-04-26
Applicant: BAYER AG
Inventor: GREIF GIESELA , HABERKORN AXEL , BAASNER BERND , LIEB FOLKER , MARHOLD ALBRECHT , STOELTING JOERN
IPC: C07D491/048 , A01N43/28 , A01N43/52 , A01N43/90 , A61K31/4184 , A61P33/02 , C07D405/06 , C07D491/04 , C07D491/056 , C07D319/00 , C07D235/00
Abstract: The present invention relates to a new substituted benzimidazoles, their preparation and their use as agents against parasitic protazoa.
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公开(公告)号:DK1080086T3
公开(公告)日:2002-12-23
申请号:DK99920603
申请日:1999-04-07
Applicant: BAYER AG
Inventor: STOELTING JOERN , STOLTEFUSS JUERGEN , GOLDMANN SIEGFRIED , KRAEMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF
IPC: C07D213/78 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/04 , C07D401/14 , C07D417/14
Abstract: The invention relates to compounds of the formule
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公开(公告)号:DE10122235A1
公开(公告)日:2002-11-14
申请号:DE10122235
申请日:2001-05-08
Applicant: BAYER AG
Inventor: STOELTING JOERN , HOISCHEN DOROTHEE , ROLAND ANDREE , LINKER KARL-HEINZ , WEINTRITT HOLGER , WROBLOWSKY HEINZ-JUERGEN
IPC: C07D239/60 , C07D239/22 , C07D239/54
Abstract: The invention relates to a novel method for the production of known 1-amino-3-phenyl-uracil derivatives (1-amino-3-phenyl-2,4(1H,3H)pyrimidindione derivatives), in addition to novel 1-amino-6-hydroxy-3-phenyl-dihydro-2,4(1H,3H)pyrimidindione derivatives of formula (II) in intermediate products therefor, and a method for the production thereof.
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公开(公告)号:AT223401T
公开(公告)日:2002-09-15
申请号:AT99920603
申请日:1999-04-07
Applicant: BAYER AG
Inventor: STOELTING JOERN , STOLTEFUSS JUERGEN , GOLDMANN SIEGFRIED , KRAEMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF
IPC: C07D213/78 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/04 , C07D401/14 , C07D417/14
Abstract: The invention relates to compounds of the formule
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公开(公告)号:BG104812A
公开(公告)日:2001-06-29
申请号:BG10481200
申请日:2000-09-29
Applicant: BAYER AG
Inventor: STOELTING JOERN , STOLTEFUSS JURGEN , GOLDMANN SIEGFRIED , KRAMER THOMAS , SCHLEMMER KARL-HEINZ , NIEWOEHNER ULRICH , PAESSENS ARNOLD , GRAEF ERWIN , LOTTMANN STEFAN , DERES KARL , WEBER OLAF
IPC: C07D213/78 , A61K31/506 , A61P1/16 , A61P31/12 , C07D213/00 , C07D213/84 , C07D215/00 , C07D239/00 , C07D239/22 , C07D277/62 , C07D401/04 , C07D401/14 , C07D417/14
Abstract: The compounds are used for the treatment and prevention of hepatitis B. The invention relates to compounds with general formulae wherein the meanings of the substituents are given in the description, to a method for the preparation of these compounds and to their application as medicaments. 16 claims
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