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公开(公告)号:EP0892797A4
公开(公告)日:2004-10-20
申请号:EP97906761
申请日:1997-02-24
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: DING CHARLES Z , HUNT JOHN T , KIM SOONG-HOON , MITT TOOMIS , BHIDE RAJEEV , LEFTHERIS KATERINA
IPC: C07D401/14 , A61K31/00 , A61K31/35 , A61K31/4178 , A61K31/495 , A61K31/498 , A61K31/55 , A61K31/551 , A61K31/5513 , A61K31/675 , A61P35/00 , A61P43/00 , C07D20060101 , C07D243/14 , C07D245/06 , C07D401/04 , C07D401/10 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/14 , C07D407/14 , C07D409/14 , C07D413/06 , C07D413/12 , C07D413/14 , C07D417/04 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D487/04 , C07D491/044 , C07D491/048 , C07D495/04 , C07D497/04 , C07D513/04 , C07F9/645
CPC classification number: C07D243/14 , C07D401/14 , C07D403/06 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D473/00 , C07D487/04 , C07D495/04
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公开(公告)号:EP0994856A4
公开(公告)日:2000-12-06
申请号:EP98930299
申请日:1998-06-16
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: BHIDE RAJEEV S , DING CHARLES Z , HUNT JOHN T , KIM SOONG-HOON , LEFTHERIS KATERINA
IPC: C07D403/08 , A61K31/4709 , A61K31/55 , A61P35/00 , A61P37/02 , A61P43/00 , C07D233/54 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/12 , C07D403/14 , C07D409/14 , C07D233/02 , C07D233/04 , C07D235/02 , C07D249/00 , C07D249/16 , C07D257/04 , C07D257/10 , C07D403/00 , C07D403/02
CPC classification number: C07D401/06 , C07D403/06 , C07D403/12 , C07D409/14
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23.
公开(公告)号:EP1617840A4
公开(公告)日:2008-08-20
申请号:EP04760683
申请日:2004-05-03
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: DYCKMAN ALARIC , DAS JAGABANDHU , LEFTHERIS KATERINA , LIU CHUNJIAN , MOQUIN ROBERT V , WROBLESKI STEPHEN T
IPC: C07D231/14 , A61K20060101 , A61K31/415 , A61K31/4152 , A61K31/4155 , A61K31/416 , A61K31/4439 , A61K31/497 , A61K31/501 , A61K31/506 , A61K31/535 , A61K31/675 , A61P37/00 , C07D20060101 , C07D231/04 , C07D231/18 , C07D401/04 , C07D401/12 , C07D403/04 , C07D405/12 , C07D413/12 , C07D413/14
CPC classification number: C07D231/14 , C07D231/12 , C07D231/40 , C07D401/12 , C07D413/12
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24.ARYL KETONE PYRROLO-TRIAZINE COMPOUNDS USEFUL AS KINASE INHIBITORS 有权
Title translation: 芳基酮吡咯烷三嗪化合物适合作为激酶抑制剂公开(公告)号:EP1503996A4
公开(公告)日:2006-05-17
申请号:EP03718493
申请日:2003-04-18
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: DYCKMAN ALARIC , LEFTHERIS KATERINA , HYNES JOHN
IPC: A61K31/53 , A61P1/04 , A61P3/10 , A61P9/10 , A61P11/00 , A61P11/06 , A61P17/06 , A61P19/02 , A61P19/06 , A61P19/08 , A61P19/10 , A61P29/00 , A61P37/06 , A61P43/00 , C07D253/10 , C07D401/06 , C07D403/06 , C07D487/04
CPC classification number: C07D487/04
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25.
公开(公告)号:EP1590335A4
公开(公告)日:2006-03-08
申请号:EP04708546
申请日:2004-02-05
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: CHEN BANG-CHI , ZHAO RULIN , SUNDEEN JOSEPH EDWARD , LEFTHERIS KATERINA , HYNES JOHN , WROBLESKI STEPHEN T
IPC: A61K31/53 , A61P29/00 , C07D20060101 , C07D253/08 , C07D487/04
CPC classification number: C07D487/04
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公开(公告)号:EP1406875A4
公开(公告)日:2005-05-04
申请号:EP02746724
申请日:2002-06-26
Applicant: SQUIBB BRISTOL MYERS CO , PHARMACOPEIA INC
Inventor: AHMED GULZAR , METZGER AXEL , WROBLESKI STEPHEN T , HENDERSON IAN , WEN JAMES , DILLER DAVID J , LEFTHERIS KATERINA
IPC: A61K31/44 , A61K31/505 , A61K31/506 , A61K31/551 , A61K31/56 , A61P1/02 , A61P1/04 , A61P1/16 , A61P1/18 , A61P3/10 , A61P7/02 , A61P7/04 , A61P7/06 , A61P9/00 , A61P9/04 , A61P9/10 , A61P11/00 , A61P13/12 , A61P17/00 , A61P17/02 , A61P17/06 , A61P19/02 , A61P19/06 , A61P19/08 , A61P19/10 , A61P21/04 , A61P25/00 , A61P25/02 , A61P25/16 , A61P25/28 , A61P27/02 , A61P29/00 , A61P29/02 , A61P31/00 , A61P31/12 , A61P31/18 , A61P35/00 , A61P35/04 , A61P37/02 , A61P37/04 , A61P37/06 , A61P37/08 , A61P43/00 , C07D213/85 , C07D239/48 , C07D239/50 , C07D401/12 , C07D403/12 , C07D403/14 , C07D409/12 , C07D239/42
CPC classification number: C07D239/48 , C07D213/85 , C07D239/47 , C07D239/50 , C07D401/12 , C07D403/12
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27.TRICYCLIC-HETEROARYL COMPOUNDS USEFUL AS KINASE INHIBITORS 有权
Title translation: 作为激酶抑制剂TRIZYKLISCHEM杂有用的链接公开(公告)号:EP1778693A4
公开(公告)日:2009-11-11
申请号:EP05803757
申请日:2005-06-30
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: LIN JAMES , WROBLESKI STEPHEN T , LIU CHUNJIAN , LEFTHERIS KATERINA
IPC: C07D487/14 , A61K31/53 , A61P3/10 , A61P9/04 , A61P19/02
CPC classification number: C07D487/14
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公开(公告)号:EP1620108A4
公开(公告)日:2008-08-27
申请号:EP04760705
申请日:2004-05-03
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: DYCKMAN ALARIC , DAS JAGABANDHU , LEFTHERIS KATERINA , LIU CHUNJIAN , MOQUIN ROBERT V , WROBLESKI STEPHEN T
IPC: C07D231/14 , A61K20060101 , A61K31/415 , A61K31/4152 , A61K31/4155 , A61K31/416 , A61K31/4439 , A61K31/497 , A61K31/501 , A61K31/506 , A61K31/535 , A61K31/675 , A61P29/00 , C07D20060101 , C07D231/04 , C07D231/18 , C07D231/38 , C07D231/40 , C07D401/04 , C07D401/12 , C07D403/04 , C07D405/12 , C07D413/12 , C07D413/14
CPC classification number: C07D231/14 , C07D231/12 , C07D231/40 , C07D401/12 , C07D413/12
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29.ARYL-SUBSTITUTED PYRAZOLE-AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS 有权
Title translation: 作为激酶抑制剂的合适的芳PYRAZOLAMIDVERBINDUNGEN公开(公告)号:EP1618092A4
公开(公告)日:2008-08-20
申请号:EP04751133
申请日:2004-05-03
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: DYCKMAN ALARIC , DAS JAGABANDHU , LEFTHERIS KATERINA , LIU CHUNJIAN , ZHAO RULIN , CHEN BANG-CHI , WROBLESKI STEPHEN T
IPC: C07D231/18 , A61K20060101 , A61K31/415 , A61K31/4152 , A61K31/4155 , A61K31/416 , A61K31/4439 , A61K31/497 , A61K31/501 , A61K31/506 , A61K31/535 , A61K31/675 , A61P37/00 , C07D20060101 , C07D231/04 , C07D231/14 , C07D401/04 , C07D401/12 , C07D403/04 , C07D405/12 , C07D413/12 , C07D413/14
CPC classification number: C07D231/14 , C07D231/12 , C07D231/40 , C07D401/12 , C07D413/12
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30.METHODS FOR THE PREPARATION OF PYRROLOTRIAZINE COMPOUNDS USEFUL AS KINASE INHIBITORS 有权
Title translation: 用于生产VONPYRROLOTRIAZINVERBINDUNGEN引致的,激酶抑制剂适合...公开(公告)号:EP1562949A4
公开(公告)日:2007-09-12
申请号:EP03781756
申请日:2003-11-03
Applicant: SQUIBB BRISTOL MYERS CO
Inventor: GODFREY JOLLIE DUAINE JR , HYNES JOHN JR , DYCKMAN ALARIC J , LEFTHERIS KATERINA , SHI ZHONGPING , WROBLESKI STEPHEN T , DOUBLEDAY WENDEL WILLIAM , GROSSO JOHN A
IPC: A61P11/06 , A61P19/02 , A61P19/10 , C07D207/50 , C07D487/04 , C07D519/00 , A61K31/53
CPC classification number: C07D487/04 , C07D207/50
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