-
公开(公告)号:ZA955868B
公开(公告)日:1997-01-14
申请号:ZA955868
申请日:1995-07-14
Applicant: BASF AG
Inventor: HELLENDAHL BEATE , LANSKY ANNEGRET , MUNSCHAUER RAINER , BIALOJAN SIEGFRIED , UNGER LILIANE , TESCHENDORF HANS-JUERGEN , WICKE KARSTEN , DRESCHER KARLA
IPC: C07D239/26 , A61K31/505 , A61K31/506 , A61P25/16 , A61P25/24 , A61P25/26 , C07D239/38 , C07D239/46 , C07D239/56 , C07D239/60 , C07D401/00 , C07D401/12 , C07D , A61K
Abstract: The present invention relates to the use of pyrimidine compounds of the following formula:wherein R1, R2, R3, A, B and Ar have the meanings indicated in the description. The compounds according to the invention have a high affinity for the dopamine D3 receptor and can therefore be used to treat disorders which respond to dopamine D3 ligands.
-
公开(公告)号:ZA9505867B
公开(公告)日:1997-01-14
申请号:ZA9505867
申请日:1995-07-14
Applicant: BASF AG
Inventor: HELLENDAHL BEATE , LANSKY ANNEGRET , MUNSCHAUER RAINER , BIALOJAN SIEGFRIED , UNGER LILIANE , TESCHENDORF HANS-JUERGEN , WICKE KARSTEN , DRESCHER KARLA
IPC: C07D249/08 , A61K31/41 , A61K31/435 , A61K31/4427 , A61K31/445 , A61K31/505 , A61K31/53 , A61P1/08 , A61P25/18 , A61P25/20 , A61P25/24 , A61P25/26 , C07D249/12 , C07D249/14 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D , A61K
CPC classification number: C07D403/12 , C07D249/12
-
公开(公告)号:FI970148A0
公开(公告)日:1997-01-14
申请号:FI970148
申请日:1997-01-14
Applicant: BASF AG
Inventor: HELLENDAHL BEATE , LANSKY ANNEGRET , RENDENBACH-MUELLER BEATRICE , BACH ALFRED , UNGER LILIANE , TESCHENDORF HANS-JUERGEN , WICKE KARSTEN
IPC: C07D233/84 , A61K31/33 , A61K31/415 , A61K31/44 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/4425 , A61K31/445 , A61K31/495 , A61K31/496 , A61P25/18 , A61P25/20 , A61P25/24 , A61P25/26 , C07D213/56 , C07D213/64 , C07D213/65 , C07D213/70 , C07D213/73 , C07D213/79 , C07D213/81 , C07D233/90 , C07D307/79 , C07D333/24 , C07D333/28 , C07D333/38 , C07D471/18 , A61K
Abstract: PCT No. PCT/EP95/02782 Sec. 371 Date Jan. 14, 1997 Sec. 102(e) Date Jan. 14, 1997 PCT Filed Jul. 14, 1995 PCT Pub. No. WO96/02246 PCT Pub. Date Feb. 1, 1996The present invention relate to the use of heterocyclic compounds of the following formula:Het-A-B-Arwhere Het, A, B and Ar have the meanings stated in the description. The compounds according to the invention have a high affinity for the dopamine D3 receptor and can therefore be used to treat disorders which respond to dopamine D3 ligands.
-
公开(公告)号:FI970147A0
公开(公告)日:1997-01-14
申请号:FI970147
申请日:1997-01-14
Applicant: BASF AG
Inventor: HELLENDAHL BEATE , LANSKY ANNEGRET , MUNSCHAUER RAINER , BIALOJAN SIEGFRIED , UNGER LILIANE , TESCHENDORF HANS-JUERGEN , WICKE KARSTEN , DRESCHER KARLA
IPC: C07D249/08 , A61K31/41 , A61K31/435 , A61K31/4427 , A61K31/445 , A61K31/505 , A61K31/53 , A61P1/08 , A61P25/18 , A61P25/20 , A61P25/24 , A61P25/26 , C07D249/12 , C07D249/14 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D
Abstract: PCT No. PCT/EP95/02781 Sec. 371 Date Jan. 14, 1997 Sec. 102(e) Date Jan. 14, 1997 PCT Filed Jul. 14, 1995 PCT Pub. No. WO96/02520 PCT Pub. Date Feb. 1, 1996The present invention relates to triazole compounds of the following formula: where R1, R2, A, B and Ar have the meanings stated in the description. The compounds according to the invention have a high affinity for the dopamine D3 receptor and can therefore be used to treat disorders which respond to dopamine D3 ligands.
-
公开(公告)号:NZ260366A
公开(公告)日:1995-12-21
申请号:NZ26036694
申请日:1994-04-21
Applicant: BASF AG
Inventor: WINGERT HORST , HELLENDAHL BEATE , SAUTER HUBERT , LORENZ GISELA
IPC: A01N43/18 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/824 , A01N43/836 , C07D207/337 , C07D209/12 , C07D213/55 , C07D213/56 , C07D213/61 , C07D215/14 , C07D235/20 , C07D261/08 , C07D263/32 , C07D263/56 , C07D271/10 , C07D271/107 , C07D277/10 , C07D277/22 , C07D277/30 , C07D277/64 , C07D277/66 , C07D285/12 , C07D307/54 , C07D307/81 , C07D333/20 , C07D333/24 , C07D333/58 , C07D413/04 , C07D277/28 , C07D307/52 , C07D333/22 , C07D333/60 , C07D233/64 , C07D235/18 , C07D207/335 , C07D215/12 , C07D263/57 , C07D409/10 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/36 , A01N43/40 , A01N43/42 , A01N43/50 , A01N43/52 , A01N43/76
Abstract: Diaryl derivatives of the general formula I in which A denotes =CHOR , =CHSR , =CHR , =CHCl or =NOR , B denotes OR , SR or NR R , Het denotes a mono-, di- or trinuclear aromatic five-membered or six-membered heterocycle which can optionally be substituted by R, R R , R , R , R are identical or different and denote hydrogen or alkyl and U, V, and W are identical or different and denote halogen, alkyl or alkoxy, and fungicides containing these compounds.A
-
公开(公告)号:HU211107B
公开(公告)日:1995-10-30
申请号:HU9200537
申请日:1992-02-19
Applicant: BASF AG
Inventor: AMMERMANN EBERHARD , HARREUS ALBRECHT , SAUTER HUBERT , DOETZER REINHARD , LORENZ GISELA , GRAMMENOS WASSILIOS , HELLENDAHL BEATE
IPC: A01N37/50 , A01N43/54 , A01N43/58 , A01N43/76 , A01N43/836 , C07C69/65 , C07C69/653 , C07C69/734 , C07C69/738 , C07C251/48 , C07C251/50 , C07C251/52 , C07C251/54 , C07C251/56 , C07C251/58 , C07C251/60 , C07C251/86 , C07C255/15 , C07C255/57 , C07C255/58 , C07C255/62 , C07D213/77 , C07D239/42 , C07D241/20 , C07D263/32 , C07D333/28 , A01N43/40 , A01N43/74 , A01N43/82 , C07C251/32 , C07C255/66 , C07C249/16 , C07C69/73
Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).
-
公开(公告)号:NZ248276A
公开(公告)日:1995-03-28
申请号:NZ24827693
申请日:1993-07-29
Applicant: BASF AG
Inventor: WINGERT HORST , HELLENDAHL BEATE , KIRSTGEN REINHARD , SAUTER HUBERT , AMMERMANN EBERHARD , LORENZ GISELA
IPC: A01N37/42 , A01N37/10 , A01N37/34 , A01N37/36 , A01N37/50 , A01N43/10 , A01N43/40 , A01N43/78 , A01N43/80 , A01N43/84 , A01N55/00 , C07C69/618 , C07C69/734 , C07C69/738 , C07C69/76 , C07C205/56 , C07C233/31 , C07C233/54 , C07C251/48 , C07C255/23 , C07C255/62 , C07C323/57 , C07C323/60 , C07D213/54 , C07D213/55 , C07D213/56 , C07D215/12 , C07D217/16 , C07D231/12 , C07D233/92 , C07D261/08 , C07D271/10 , C07D271/107 , C07D277/20 , C07D277/22 , C07D277/58 , C07D277/66 , C07D285/12 , C07D307/54 , C07D307/71 , C07D317/60 , C07D319/18 , C07D333/24 , C07D333/28 , C07D333/38 , C07D333/42 , C07D413/12 , C07D521/00 , C07F7/10 , C07F7/22 , C07D295/04 , A01N43/06 , A01N43/72
Abstract: Acetylene derivatives of the general formula I in which U, V and W denote hydrogen, halogen, nitro, cyano, alkyl and alkoxy, A denotes alkylidene, alkoxymethylidene, alkylthiomethylidene and alkoximino, B denotes OH, alkoxy and alkylamino and R denotes hydrogen, halogen, cyano, CF3, alkyl, cycloalkyl, haloalkyl, aryl, alkenyl, alkinyl, heterocyclyl, heteroaryl, arylalkyl, arylalkenyl, arylethinyl, heteroaryl-C1-C4-alkyl, C1-C4-alkoxy-C1-C4-alkyl, aryloxyalkyl, heteroaryloxyalkyl, arylamino-alkyl, arylthiomethyl, heteroarylthiomethyl, C(O)R , C(O)NR R , C(S)NR R , C(O)SR , C(S)OR , C(S)SR , CH(OH)R )R , SiR R R , SnR R R , C(OR)R , C(=N-OR )R , and the radicals R -R , R and R denote hydrogen, alkyl, aryl, heteroaryl, arylalkyl and heteroarylalkyl, and fungicides containing these compounds.
-
公开(公告)号:ZA935787B
公开(公告)日:1995-02-10
申请号:ZA935787
申请日:1993-08-10
Applicant: BASF AG
Inventor: WINGERT HORST , HELLENDAHL BEATE , KIRSTGEN REINHARD , SAUTER HUBERT , AMMERMANN EBERHARD , LORENZ GISELA
IPC: A01N20060101 , C07C20060101 , C07C , A01N
-
公开(公告)号:ZA9305787B
公开(公告)日:1995-02-10
申请号:ZA9305787
申请日:1993-08-10
Applicant: BASF AG
Inventor: WINGERT HORST , HELLENDAHL BEATE , KIRSTGEN REINHARD , SAUTER HUBERT , AMMERMANN EBERHARD , LORENZ GISELA
IPC: A01N20060101 , C07C20060101 , C07C , A01N
-
公开(公告)号:NZ241638A
公开(公告)日:1994-04-27
申请号:NZ24163892
申请日:1992-02-18
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS , HARREUS ALBRECHT , SAUTER HUBERT , HELLENDAHL BEATE , DOETZER REINHARD , AMMERMANN EBERHARD , LORENZ GISEL
IPC: A01N37/50 , A01N43/54 , A01N43/58 , A01N43/76 , A01N43/836 , C07C69/65 , C07C69/653 , C07C69/734 , C07C69/738 , C07C251/48 , C07C251/50 , C07C251/52 , C07C251/54 , C07C251/56 , C07C251/58 , C07C251/60 , C07C251/86 , C07C255/15 , C07C255/57 , C07C255/58 , C07C255/62 , C07D213/77 , C07D239/42 , C07D241/20 , C07D263/32 , C07D333/28 , C07C255/63 , C07D237/20 , A01N43/40
Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).
-
-
-
-
-
-
-
-
-